Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WUKDUCCXRVBEIK
|
8.8 | pIC50 | 3 | Yes | |
XEEATOCFEUTHHG
|
8.8 | pIC50 | 3 | Yes | |
XEEATOCFEUTHHG
|
8.8 | pIC50 | 4 | Yes | |
XPVKGTWRXBSJKO
|
8.8 | pIC50 | 4 | Yes | |
XPZCWRLFOWPBIA
|
8.8 | pIC50 | 3 | Yes | |
XXOJIRVATXUFCB
|
8.8 | pIC50 | 3 | Yes | |
ZDUXGHLKBYRGNA
|
8.8 | pIC50 | 3 | Yes | |
ZEDBWMYOHLASAQ
|
8.8 | pIC50 | 3 | Yes | |
ZMSBWTFEDUQTFL
|
8.8 | pIC50 | 4 | Yes | |
IOVFZDQUWQWZBK
|
8.8 | pIC50 | 4 | Yes | |
BXZSQERBAIEVJJ
|
8.8 | pIC50 | 4 | Yes | |
JELDBBFVVGTYRF
|
8.8 | pIC50 | 2 | Yes | |
KBQSRNQTSRTYGN
|
8.8 | pIC50 | 4 | Yes | |
LPDMMXAJXUHKPL
|
8.8 | pIC50 | 4 | Yes | |
MYPYUWTXZVADBB
|
8.8 | pIC50 | 4 | Yes | |
OCILFYQUCSGLEE
|
8.8 | pIC50 | 4 | Yes | |
OIWJQXISVVHHBL
|
8.8 | pIC50 | 4 | Yes | |
SXKLCKROMAELSQ
|
8.8 | pIC50 | 4 | Yes | |
VICPJUSXWWJNBZ
|
8.8 | pIC50 | 3 | Yes | |
XAQTXSHCLKDVCM
|
8.8 | pIC50 | 4 | Yes | |
DASVAQCTVIQROX
|
8.8 | pIC50 | 8 | Yes | |
YSYPJTRKLLMYQR
|
8.8 | pIC50 | 4 | Yes | |
AQSSMEORRLJZLU
|
8.8 | pIC50 | 34 | Yes | |
AWOGCPXUTJBQEG
|
8.8 | pIC50 | 3 | Yes | |
BBBAWACESCACAP
|
8.8 | pIC50 | 5 | Yes | |
BHGXZDRFYWOZFO
|
8.8 | pIC50 | 4 | Yes | |
BMWYPIWSQSWTKG
|
8.8 | pIC50 | 3 | Yes | |
DLFGHUQKLJBNNO
|
8.8 | pIC50 | 2 | Yes | |
GNWBLLYJQXKPIP
|
8.8 | pIC50 | 4 | Yes | |
LOECSGIPISXOPO
|
8.8 | pIC50 | 3 | Yes | |
LTTCWZPUBNOMTJ
|
8.8 | pIC50 | 4 | Yes | |
MLZAWUZXMPRAMY
|
8.8 | pIC50 | 3 | Yes | |
NVSJOASGKCGXBZ
|
8.8 | pIC50 | 16 | Yes | |
OJLYUGSSUKAWJC
|
8.8 | Ki | 16 | — | |
PMSRTLBMXMXKDM
|
8.8 | pIC50 | 4 | Yes | |
QASMLJURBZXYNW
|
8.8 | pIC50 | 4 | Yes | |
QASMLJURBZXYNW
|
8.8 | pIC50 | 4 | Yes | |
RBSPTCQSWKXPGH
|
8.8 | pIC50 | 4 | Yes | |
SFEJKVIUEGSERT
|
8.8 | pIC50 | 3 | Yes | |
WGUNFTKBYUCLEL
|
8.8 | pIC50 | 4 | Yes | |
WFRLFWGASBLYTC
|
8.8 | pIC50 | 15 | Yes | |
CXIZEAWVDWCMQV
|
8.7 | pIC50 | 2 | Yes | |
DJJCBDOVULVMNS
|
8.7 | pIC50 | 4 | Yes | |
HYKBWCOBEOHSMP
|
8.7 | pIC50 | 4 | Yes | |
KVKYGVOAHGNAKZ
|
8.7 | IC50 | 16 | — | |
LZACPHWPRDKUPK
|
8.7 | pIC50 | 5 | Yes | |
NGGIJEYOMPYIIW
|
8.7 | pIC50 | 3 | Yes | |
UYUBFBWOFKSJPT
|
8.7 | pIC50 | 5 | Yes | |
WQNDOASZRAMVMT
|
8.7 | pIC50 | 3 | Yes | |
DUYNJNWVGIWJRI
|
8.7 | pIC50 | 4 | Yes |