Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTOVSRDMFFEVOJ
|
8.9 | pIC50 | 4 | Yes | |
OCOJLTOWRUXQCT
|
8.9 | pIC50 | 4 | Yes | |
UCTPVBCFMDURFZ
|
8.9 | pIC50 | 4 | Yes | |
XIWROJLPONIAKV
|
8.9 | pIC50 | 4 | Yes | |
XLKOPUNLSAOKDW
|
8.9 | pIC50 | 4 | Yes | |
BVCVYTLOMICPJW
|
8.9 | pIC50 | 4 | Yes | |
WNXGFXISCVUWCA
|
8.9 | pIC50 | 4 | Yes | |
AVCFYGNSQWJCRG
|
8.9 | pIC50 | 3 | Yes | |
DFYOVMKHYAWORB
|
8.9 | pIC50 | 3 | Yes | |
DHRWPORNZCWGED
|
8.9 | pIC50 | 4 | Yes | |
KJKOZLCYQNBBEX
|
8.9 | pIC50 | 3 | Yes | |
NWKCPPJDKLUHDY
|
8.9 | pIC50 | 4 | Yes | |
OVFXCANAVHBWGG
|
8.9 | pIC50 | 4 | Yes | |
PTZCIKOPLAEWTE
|
8.9 | pIC50 | 4 | Yes | |
RLZHDVSWTRNLIA
|
8.9 | pIC50 | 3 | Yes | |
XOIYZMDJFLKIEI
|
8.9 | pIC50 | 5 | Yes | |
YIFNILRPNDYIBP
|
8.9 | pIC50 | 3 | Yes | |
YNNSWQDWQWPZOM
|
8.9 | pIC50 | 3 | Yes | |
OPURNPRECWSMQM
|
8.9 | pIC50 | 4 | Yes | |
BAAILVWEAXFTSF
|
8.8 | pIC50 | 5 | Yes | |
FNSIACDWDZGUHN
|
8.8 | pIC50 | 4 | Yes | |
GBNLUWROABYNBX
|
8.8 | pIC50 | 4 | Yes | |
KOYRLVBQHJNLQX
|
8.8 | pIC50 | 4 | Yes | |
LYJSJVYJLZOMCD
|
8.8 | pIC50 | 4 | Yes | |
MXIFCKWMUUNDJR
|
8.8 | pIC50 | 2 | Yes | |
NZUFHNXGURICPD
|
8.8 | pIC50 | 4 | Yes | |
OSDJMOWFTIFDAM
|
8.8 | pIC50 | 4 | Yes | |
PHEDXBVPIONUQT
|
8.8 | pIC50 | 6 | Yes | |
PXAAAZSWSOSGCM
|
8.8 | pIC50 | 3 | Yes | |
QGSOGWMSZGIIKI
|
8.8 | pIC50 | 3 | Yes | |
QGSOGWMSZGIIKI
|
8.8 | pIC50 | 4 | Yes | |
QXWCRBMAGJJKTO
|
8.8 | pIC50 | 4 | Yes | |
UZRQKIJPXLTOGR
|
8.8 | pIC50 | 3 | Yes | |
MFDCEMLTTQCDTH
|
8.8 | pIC50 | 3 | Yes | |
BLGCEUZOXJETEV
|
8.8 | pIC50 | 6 | Yes | |
BNVBGYDJTSISOS
|
8.8 | pIC50 | 3 | Yes | |
BVVFOLSZMQVDKV
|
8.8 | pIC50 | 4 | Yes | |
DCIBBANBLKPKCU
|
8.8 | pIC50 | 3 | Yes | |
FYYOGLGDZCDBDF
|
8.8 | pIC50 | 3 | Yes | |
GOAGYYXQSDTWIW
|
8.8 | pIC50 | 3 | Yes | |
HKMOWVBBDIDACP
|
8.8 | pIC50 | 3 | Yes | |
KIRCGKZULASNTL
|
8.8 | pIC50 | 3 | Yes | |
OCOJLTOWRUXQCT
|
8.8 | pIC50 | 4 | Yes | |
OLTVRSUIOUTBRQ
|
8.8 | pIC50 | 4 | Yes | |
QZCYXWFWSDBJGL
|
8.8 | pIC50 | 8 | Yes | |
TYSOZDHVMFAZKD
|
8.8 | pIC50 | 4 | Yes | |
URTDYVBTGQDEKN
|
8.8 | pIC50 | 4 | Yes | |
UYBIVRLEZVLKDU
|
8.8 | pIC50 | 4 | Yes | |
UZDRXGWOSNDZDM
|
8.8 | pIC50 | 4 | Yes | |
VUNGWWRBVPWOKS
|
8.8 | pIC50 | 4 | Yes |