Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CTKCIBJHOHRDAM
|
9.0 | pIC50 | 4 | Yes | |
CXNZLOIPQFMHLT
|
9.0 | pIC50 | 4 | Yes | |
DMOIIDXHXUHFJK
|
9.0 | pIC50 | 3 | Yes | |
FAKNYSRJFRSEFB
|
9.0 | pIC50 | 4 | Yes | |
FVFFDKKTXYVCCW
|
9.0 | IC50 | 16 | — | |
HTKQZECDKPTYRG
|
9.0 | pIC50 | 5 | Yes | |
HYSLEZHDLSYQLQ
|
9.0 | pIC50 | 5 | Yes | |
IGMUAHQVBFCVQW
|
9.0 | pIC50 | 6 | Yes | |
IMIUBDGXYBCWQZ
|
9.0 | pIC50 | 3 | Yes | |
IPHSQMSRIWZULE
|
9.0 | Ki | 16 | — | |
JIADIKISVDGGIN
|
9.0 | pIC50 | 3 | Yes | |
KDMMIKQMHNBKAV
|
9.0 | Ki | 17 | — | |
KOVRZNUMIKACTB
|
9.0 | IC50 | 17 | — | |
KYOFSMKRNGJKGT
|
9.0 | pIC50 | 4 | Yes | |
LCGSYJVWLGYWTD
|
9.0 | pIC50 | 4 | Yes | |
LHFFYCSBQXAENY
|
9.0 | pIC50 | 3 | Yes | |
LVOBTCONHRNJJA
|
9.0 | pIC50 | 4 | Yes | |
NMAZHZSPSGSCEM
|
9.0 | pIC50 | 3 | Yes | |
NWZALETXBFNATO
|
9.0 | pIC50 | 3 | Yes | |
ONKCOSCHJAFALI
|
9.0 | pIC50 | 4 | Yes | |
RLFKILXOLJVUNF
|
9.0 | IC50 | 16 | — | |
RVPDXKXWYPPTAL
|
9.0 | pIC50 | 7 | Yes | |
UHZDMCREDJRFHQ
|
9.0 | pIC50 | 4 | Yes | |
UJAZLJYGTKUQPF
|
9.0 | pIC50 | 4 | Yes | |
UONOEOTYMVCADB
|
9.0 | pIC50 | 3 | Yes | |
VZCOCGXPISHVHC
|
9.0 | pIC50 | 3 | Yes | |
WGRVAGIQTHEEQW
|
9.0 | IC50 | 16 | — | |
XGTIAYLYSJBDIA
|
9.0 | pIC50 | 3 | Yes | |
NJVFOFMHUJJIMB
|
9.0 | pIC50 | 4 | Yes | |
AFCXUMJPOGOVIU
|
9.0 | pIC50 | 4 | Yes | |
BRFOVRDNLUKMTR
|
9.0 | pIC50 | 4 | Yes | |
BSBLYLUAUVTSMM
|
9.0 | IC50 | 16 | — | |
CQGQVNKFCSRASR
|
9.0 | pIC50 | 4 | Yes | |
DACGDZLVWJQELB
|
9.0 | pIC50 | 3 | Yes | |
FJEBOUIPWLCERS
|
9.0 | pIC50 | 2 | Yes | |
KGLHEVXFWIJETJ
|
9.0 | pIC50 | 4 | Yes | |
KREZVKKCLKOMEF
|
9.0 | pIC50 | 4 | Yes | |
MKGQECWCAKASNT
|
9.0 | pIC50 | 4 | Yes | |
MKLXMJUHEZXHPX
|
9.0 | pIC50 | 4 | Yes | |
OYUGBGZDLCAQEA
|
9.0 | pIC50 | 4 | Yes | |
SOKFWRPORPTXSA
|
9.0 | pIC50 | 2 | Yes | |
UYRALUALZCKFQB
|
9.0 | pIC50 | 3 | Yes | |
NVBFHJWHLNUMCV
|
8.9 | pIC50 | 4 | Yes | |
OITCYCYIUVYFKQ
|
8.9 | pIC50 | 4 | Yes | |
IWDLFWORFMDTLN
|
8.9 | pIC50 | 4 | Yes | |
KZGJWJJJDKPFMH
|
8.9 | pIC50 | 4 | Yes | |
SYQPAVSGPRYEOO
|
8.9 | pIC50 | 4 | Yes | |
CBNHHPMBIUENPL
|
8.9 | pIC50 | 3 | Yes | |
FCGKZIRRZCVIGR
|
8.9 | pIC50 | 7 | Yes | |
JISNDAMZBNGEAC
|
8.9 | pIC50 | 2 | Yes |