Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SUPHGISSSNNOGO
|
9.1 | pIC50 | 4 | Yes | |
UAWFPNAVZNTVLR
|
9.1 | pIC50 | 4 | Yes | |
UPNAHMSJUMHPOR
|
9.1 | pIC50 | 4 | Yes | |
VZKRZUPJCVFVGR
|
9.1 | IC50 | 16 | — | |
WGYZSJCMDOXKNM
|
9.1 | pIC50 | 4 | Yes | |
XMXSDIHLINKFLN
|
9.1 | pIC50 | 4 | Yes | |
ZBNZXTGUTAYRHI
|
9.1 | pIC50 | 102 | Yes | |
ZMYFLSKLOJVQBK
|
9.1 | pIC50 | 3 | Yes | |
DGBIGWXXNGSACT
|
9.1 | Ki | 16 | — | |
IENZQIKPVFGBNW
|
9.1 | pIC50 | 11 | Yes | |
IXTYIAPVUSDHLB
|
9.1 | pIC50 | 4 | Yes | |
NGOHYVFQZPROBG
|
9.1 | pIC50 | 6 | Yes | |
AQFHRIRPLDYFGS
|
9.1 | pIC50 | 3 | Yes | |
ARJOCRMEGRIBFE
|
9.1 | pIC50 | 4 | Yes | |
BZQBJHJYQYGIHL
|
9.1 | pIC50 | 4 | Yes | |
CEVFZHVZMHZPRV
|
9.1 | pIC50 | 4 | Yes | |
CTKCIBJHOHRDAM
|
9.1 | pIC50 | 4 | Yes | |
GZOGYGSYSRTUBF
|
9.1 | pIC50 | 4 | Yes | |
HHOVYYSFRMBKPP
|
9.1 | pIC50 | 3 | Yes | |
HVFXPRVDRFNNGG
|
9.1 | pIC50 | 3 | Yes | |
HWADPEMDUDRDOV
|
9.1 | pIC50 | 4 | Yes | |
IOHWQOBDRDHMNK
|
9.1 | pIC50 | 4 | Yes | |
JQKANSBWFRBIRJ
|
9.1 | pIC50 | 4 | Yes | |
JUMHXAHUWIPRTK
|
9.1 | pIC50 | 4 | Yes | |
KREZVKKCLKOMEF
|
9.1 | pIC50 | 4 | Yes | |
OCNLOXNOURUUDD
|
9.1 | pIC50 | 4 | Yes | |
OFBIFZUFASYYRE
|
9.1 | Ki | 16 | — | |
RHDBRQBCMWHOTA
|
9.1 | pIC50 | 4 | Yes | |
SNURMSXWIAIOCJ
|
9.1 | pIC50 | 4 | Yes | |
VATZWJYBMQBVKJ
|
9.1 | pIC50 | 4 | Yes | |
VEYVECZRBNJMJV
|
9.1 | pIC50 | 4 | Yes | |
WUSQSYLTSUGLKJ
|
9.1 | pIC50 | 3 | Yes | |
XBYJCVDSFWJBSM
|
9.1 | pIC50 | 6 | Yes | |
XMVZTBZRGWZAOZ
|
9.1 | pIC50 | 4 | Yes | |
YJZGQBGGTBIAOP
|
9.1 | IC50 | 16 | — | |
ZZJKKUWYWYKHBB
|
9.1 | pIC50 | 4 | Yes | |
ABWCAVMWLBXQQF
|
9.0 | pIC50 | 4 | Yes | |
JKVAFNSXXFFLKN
|
9.0 | pIC50 | 4 | Yes | |
XTMQXGYZVJVLMD
|
9.0 | pIC50 | 3 | Yes | |
QQYZSCQKDDRJGS
|
9.0 | pIC50 | 3 | Yes | |
OLTPRSGJHXAYBO
|
9.0 | pIC50 | 6 | Yes | |
QAOAUSPEVNTMIF
|
9.0 | pIC50 | 6 | Yes | |
TZACYAAFEOUQNL
|
9.0 | pIC50 | 4 | Yes | |
FABVMONGQZFVFR
|
9.0 | pIC50 | 6 | Yes | |
ABKUNMXQTDTBPW
|
9.0 | pIC50 | 6 | Yes | |
AQKFCEWRKDXGMK
|
9.0 | Ki | 16 | — | |
AQVOTCCORNBNKJ
|
9.0 | pIC50 | 3 | Yes | |
ATYLCJOUAUSNKE
|
9.0 | pIC50 | 4 | Yes | |
BEULGLCETLDRNQ
|
9.0 | pIC50 | 5 | Yes | |
CRCNSYRHGVJFMT
|
9.0 | pIC50 | 4 | Yes |