Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LRADDEITIGOBAG
|
9.2 | pIC50 | 4 | Yes | |
NGOWHFOEQRKCQX
|
9.2 | pIC50 | 3 | Yes | |
NJIYCMKWBWEALF
|
9.2 | pIC50 | 4 | Yes | |
PUGUGQZVQLLOFL
|
9.2 | pIC50 | 4 | Yes | |
QVXLLSDFMNQMLD
|
9.2 | pIC50 | 3 | Yes | |
VMXKZXYUKBFHEP
|
9.2 | pIC50 | 3 | Yes | |
WGYZSJCMDOXKNM
|
9.2 | pIC50 | 4 | Yes | |
WUCDOXDCHOCLCO
|
9.2 | pIC50 | 3 | Yes | |
XJMIBNLJFYSGAR
|
9.2 | IC50 | 16 | — | |
XTLIGSXCHIJPDK
|
9.2 | pIC50 | 4 | Yes | |
YAHPNJWQRCEXRQ
|
9.2 | pIC50 | 3 | Yes | |
ZPMDXAPBRHPDIM
|
9.2 | pIC50 | 3 | Yes | |
ARZNLQCBMDYYDU
|
9.2 | pIC50 | 2 | Yes | |
GBDGTOLMAXSIBD
|
9.2 | pIC50 | 3 | Yes | |
LSMUQPOCAXNDRJ
|
9.2 | pIC50 | 4 | Yes | |
SHUMXHZGMOYSRM
|
9.2 | pIC50 | 4 | Yes | |
OFYCPZYSYANJMI
|
9.2 | pIC50 | 4 | Yes | |
ASXGJMSKWNBENU
|
9.2 | pIC50 | 12 | Yes | |
FSYFYSFYUHBIHE
|
9.2 | pIC50 | 4 | Yes | |
SUXYGJZMCWKJJI
|
9.2 | pIC50 | 26 | Yes | |
WLEXCTJQABXUGS
|
9.2 | pIC50 | 4 | Yes | |
BSVZGMIZZFSSFC
|
9.2 | pIC50 | 4 | Yes | |
CLYUNXJFERDYMU
|
9.2 | pIC50 | 4 | Yes | |
DLCGHEAGXLUOOT
|
9.2 | pIC50 | 4 | Yes | |
FAZOEMRTBCXQLO
|
9.2 | pIC50 | 4 | Yes | |
GCVNOSTYUVURLK
|
9.2 | pIC50 | 3 | Yes | |
GHZHWDWADLAOIQ
|
9.2 | pIC50 | 2 | Yes | |
GTPUHNJIMQQEMY
|
9.2 | pIC50 | 4 | Yes | |
HMUAODOJRHDKMR
|
9.2 | pIC50 | 3 | Yes | |
JBKMRMOTMJVNML
|
9.2 | pIC50 | 11 | Yes | |
NOYGCWVGNBCIJK
|
9.2 | pIC50 | 4 | Yes | |
PKIBTPDYAFKEOS
|
9.2 | pIC50 | 4 | Yes | |
UBPYILGKFZZVDX
|
9.2 | pIC50 | 130 | Yes | |
ZDNCDNWZGWFVKE
|
9.2 | pIC50 | 4 | Yes | |
PFCYQMFWFCEFGN
|
9.1 | pIC50 | 4 | Yes | |
ALXFBXZUXCHLTA
|
9.1 | pIC50 | 4 | Yes | |
GHZHWDWADLAOIQ
|
9.1 | pIC50 | 2 | Yes | |
XHRFFDAZHQMDPM
|
9.1 | pIC50 | 3 | Yes | |
XBLYYDDTTORRLT
|
9.1 | pIC50 | 3 | Yes | |
BZKPWHYZMXOIDC
|
9.1 | pIC50 | 20 | Yes | |
CRLVKJCAHBZLJT
|
9.1 | pIC50 | 4 | Yes | |
GFUKHIMMBLMJDN
|
9.1 | pIC50 | 4 | Yes | |
GHWLNWTTXZKARD
|
9.1 | pIC50 | 3 | Yes | |
GHZHWDWADLAOIQ
|
9.1 | pIC50 | 2 | Yes | |
JFGUJXZLJIUVPZ
|
9.1 | IC50 | 16 | — | |
JZSYDIHQPGCMDN
|
9.1 | pIC50 | 4 | Yes | |
KSIKWQAAQUDISH
|
9.1 | pIC50 | 3 | Yes | |
LYFROTHEKIFZAU
|
9.1 | IC50 | 16 | — | |
QTRPSCXVKWWSNO
|
9.1 | pIC50 | 4 | Yes | |
RYIVVNHBYBYXHF
|
9.1 | IC50 | 16 | — |