Target Details
UniProt ACP18505
Gene SymbolGABRB1
Protein NameGamma-aminobutyric acid receptor subunit beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 5,316
  • Clinical molecules 4981
  • Avg pChEMBL 7.5
Top Co-occurrence Targets
Active Molecules (5,316)
InChIKey pChEMBL Type Targets Clinical
LRADDEITIGOBAG 9.2 pIC50 4 Yes
NGOWHFOEQRKCQX 9.2 pIC50 3 Yes
NJIYCMKWBWEALF 9.2 pIC50 4 Yes
PUGUGQZVQLLOFL 9.2 pIC50 4 Yes
QVXLLSDFMNQMLD 9.2 pIC50 3 Yes
VMXKZXYUKBFHEP 9.2 pIC50 3 Yes
WGYZSJCMDOXKNM 9.2 pIC50 4 Yes
WUCDOXDCHOCLCO 9.2 pIC50 3 Yes
XJMIBNLJFYSGAR 9.2 IC50 16
XTLIGSXCHIJPDK 9.2 pIC50 4 Yes
YAHPNJWQRCEXRQ 9.2 pIC50 3 Yes
ZPMDXAPBRHPDIM 9.2 pIC50 3 Yes
ARZNLQCBMDYYDU 9.2 pIC50 2 Yes
GBDGTOLMAXSIBD 9.2 pIC50 3 Yes
LSMUQPOCAXNDRJ 9.2 pIC50 4 Yes
SHUMXHZGMOYSRM 9.2 pIC50 4 Yes
OFYCPZYSYANJMI 9.2 pIC50 4 Yes
ASXGJMSKWNBENU 9.2 pIC50 12 Yes
FSYFYSFYUHBIHE 9.2 pIC50 4 Yes
SUXYGJZMCWKJJI 9.2 pIC50 26 Yes
WLEXCTJQABXUGS 9.2 pIC50 4 Yes
BSVZGMIZZFSSFC 9.2 pIC50 4 Yes
CLYUNXJFERDYMU 9.2 pIC50 4 Yes
DLCGHEAGXLUOOT 9.2 pIC50 4 Yes
FAZOEMRTBCXQLO 9.2 pIC50 4 Yes
GCVNOSTYUVURLK 9.2 pIC50 3 Yes
GHZHWDWADLAOIQ 9.2 pIC50 2 Yes
GTPUHNJIMQQEMY 9.2 pIC50 4 Yes
HMUAODOJRHDKMR 9.2 pIC50 3 Yes
JBKMRMOTMJVNML 9.2 pIC50 11 Yes
NOYGCWVGNBCIJK 9.2 pIC50 4 Yes
PKIBTPDYAFKEOS 9.2 pIC50 4 Yes
UBPYILGKFZZVDX 9.2 pIC50 130 Yes
ZDNCDNWZGWFVKE 9.2 pIC50 4 Yes
PFCYQMFWFCEFGN 9.1 pIC50 4 Yes
ALXFBXZUXCHLTA 9.1 pIC50 4 Yes
GHZHWDWADLAOIQ 9.1 pIC50 2 Yes
XHRFFDAZHQMDPM 9.1 pIC50 3 Yes
XBLYYDDTTORRLT 9.1 pIC50 3 Yes
BZKPWHYZMXOIDC 9.1 pIC50 20 Yes
CRLVKJCAHBZLJT 9.1 pIC50 4 Yes
GFUKHIMMBLMJDN 9.1 pIC50 4 Yes
GHWLNWTTXZKARD 9.1 pIC50 3 Yes
GHZHWDWADLAOIQ 9.1 pIC50 2 Yes
JFGUJXZLJIUVPZ 9.1 IC50 16
JZSYDIHQPGCMDN 9.1 pIC50 4 Yes
KSIKWQAAQUDISH 9.1 pIC50 3 Yes
LYFROTHEKIFZAU 9.1 IC50 16
QTRPSCXVKWWSNO 9.1 pIC50 4 Yes
RYIVVNHBYBYXHF 9.1 IC50 16
2D structure