Target Details
UniProt ACP18505
Gene SymbolGABRB1
Protein NameGamma-aminobutyric acid receptor subunit beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 5,316
  • Clinical molecules 4981
  • Avg pChEMBL 7.5
Top Co-occurrence Targets
Active Molecules (5,316)
InChIKey pChEMBL Type Targets Clinical
AKRKKOYYGGSJRD 9.3 pIC50 4 Yes
ALBKMJDFBZVHAK 9.3 IC50 16
ANWMJUPMEWGUTN 9.3 pIC50 3 Yes
BMQWSLBNOKTRQB 9.3 pIC50 3 Yes
BWFWKLRLHQZLAB 9.3 pIC50 4 Yes
BYMDBFGHCDTBMT 9.3 IC50 16
COJFASLRENZFLP 9.3 pIC50 4 Yes
DGNUOTXXMYEVBK 9.3 pIC50 4 Yes
DLUHBPYUABWXMD 9.3 pIC50 4 Yes
DODQJNMQWMSYGS 9.3 pIC50 4 Yes
FOUMLJPHHOLTNI 9.3 pIC50 4 Yes
FYEARXADVSSUQS 9.3 pIC50 4 Yes
GAZIJXXDYOWMAS 9.3 pIC50 3 Yes
GWRGVEOEXIBMJH 9.3 pIC50 4 Yes
HBPRHKLSAUIZHE 9.3 pIC50 3 Yes
HRVAZKKEGJGZOW 9.3 pIC50 3 Yes
IUHKSTINHDUYRO 9.3 IC50 16
MBHOBWXKVAOSNF 9.3 pIC50 3 Yes
OVEYKEUBLRTYDZ 9.3 pIC50 3 Yes
PJDIJYZHMSPAKC 9.3 pIC50 4 Yes
SAJDFWWOBZTXQE 9.3 pIC50 3 Yes
SFUGTTJDFJMSGN 9.3 pIC50 2 Yes
TYKGMSWZEALPBQ 9.3 pIC50 4 Yes
ULKYBVFYFLCZOX 9.3 pIC50 4 Yes
UNUQONUFWDAEON 9.3 pIC50 3 Yes
UZOOIPXOYYJULJ 9.3 pIC50 4 Yes
VJVAWKPXJCDEQG 9.3 IC50 16
VTXPJLWYFJDDQR 9.3 pIC50 4 Yes
WLGDFYOOSGHIPS 9.3 pIC50 4 Yes
WRXDVVALWQGPMW 9.3 IC50 16
XUTZDXHKQDPUMA 9.3 pIC50 4 Yes
YAGJNFGKXDDDJI 9.3 pIC50 3 Yes
YGIGTTQRWLXDFG 9.3 pIC50 4 Yes
ZRKMLXOVZYKUKU 9.3 pIC50 3 Yes
ZTMDXFVSRFQNLX 9.3 pIC50 4 Yes
ZZLLLCNRSQXFHU 9.3 pIC50 4 Yes
GPFRMIHXGMVMGF 9.3 pIC50 4 Yes
IKZMTNSYXDOFJH 9.3 pIC50 4 Yes
VFJFQJKZWLXQQX 9.3 pIC50 4 Yes
CWBFECUIDZXHBY 9.2 pIC50 3 Yes
BKCXBMXTXLGZCV 9.2 pIC50 3 Yes
BKCXBMXTXLGZCV 9.2 pIC50 3 Yes
BLJPKQXXDFIIFR 9.2 IC50 16
CYGCWJCVIJAEOL 9.2 pIC50 7 Yes
DWSHVVSVJWDKEK 9.2 pIC50 3 Yes
FAGYSQSLIMHWHR 9.2 pIC50 4 Yes
HHUWJVYTBKEMON 9.2 pIC50 5 Yes
HIMQJMWVIJRMHV 9.2 pIC50 4 Yes
IBIQLEWQPHHHEE 9.2 pIC50 4 Yes
JAVIIUAYGNOEAR 9.2 pIC50 4 Yes
2D structure