Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AKRKKOYYGGSJRD
|
9.3 | pIC50 | 4 | Yes | |
ALBKMJDFBZVHAK
|
9.3 | IC50 | 16 | — | |
ANWMJUPMEWGUTN
|
9.3 | pIC50 | 3 | Yes | |
BMQWSLBNOKTRQB
|
9.3 | pIC50 | 3 | Yes | |
BWFWKLRLHQZLAB
|
9.3 | pIC50 | 4 | Yes | |
BYMDBFGHCDTBMT
|
9.3 | IC50 | 16 | — | |
COJFASLRENZFLP
|
9.3 | pIC50 | 4 | Yes | |
DGNUOTXXMYEVBK
|
9.3 | pIC50 | 4 | Yes | |
DLUHBPYUABWXMD
|
9.3 | pIC50 | 4 | Yes | |
DODQJNMQWMSYGS
|
9.3 | pIC50 | 4 | Yes | |
FOUMLJPHHOLTNI
|
9.3 | pIC50 | 4 | Yes | |
FYEARXADVSSUQS
|
9.3 | pIC50 | 4 | Yes | |
GAZIJXXDYOWMAS
|
9.3 | pIC50 | 3 | Yes | |
GWRGVEOEXIBMJH
|
9.3 | pIC50 | 4 | Yes | |
HBPRHKLSAUIZHE
|
9.3 | pIC50 | 3 | Yes | |
HRVAZKKEGJGZOW
|
9.3 | pIC50 | 3 | Yes | |
IUHKSTINHDUYRO
|
9.3 | IC50 | 16 | — | |
MBHOBWXKVAOSNF
|
9.3 | pIC50 | 3 | Yes | |
OVEYKEUBLRTYDZ
|
9.3 | pIC50 | 3 | Yes | |
PJDIJYZHMSPAKC
|
9.3 | pIC50 | 4 | Yes | |
SAJDFWWOBZTXQE
|
9.3 | pIC50 | 3 | Yes | |
SFUGTTJDFJMSGN
|
9.3 | pIC50 | 2 | Yes | |
TYKGMSWZEALPBQ
|
9.3 | pIC50 | 4 | Yes | |
ULKYBVFYFLCZOX
|
9.3 | pIC50 | 4 | Yes | |
UNUQONUFWDAEON
|
9.3 | pIC50 | 3 | Yes | |
UZOOIPXOYYJULJ
|
9.3 | pIC50 | 4 | Yes | |
VJVAWKPXJCDEQG
|
9.3 | IC50 | 16 | — | |
VTXPJLWYFJDDQR
|
9.3 | pIC50 | 4 | Yes | |
WLGDFYOOSGHIPS
|
9.3 | pIC50 | 4 | Yes | |
WRXDVVALWQGPMW
|
9.3 | IC50 | 16 | — | |
XUTZDXHKQDPUMA
|
9.3 | pIC50 | 4 | Yes | |
YAGJNFGKXDDDJI
|
9.3 | pIC50 | 3 | Yes | |
YGIGTTQRWLXDFG
|
9.3 | pIC50 | 4 | Yes | |
ZRKMLXOVZYKUKU
|
9.3 | pIC50 | 3 | Yes | |
ZTMDXFVSRFQNLX
|
9.3 | pIC50 | 4 | Yes | |
ZZLLLCNRSQXFHU
|
9.3 | pIC50 | 4 | Yes | |
GPFRMIHXGMVMGF
|
9.3 | pIC50 | 4 | Yes | |
IKZMTNSYXDOFJH
|
9.3 | pIC50 | 4 | Yes | |
VFJFQJKZWLXQQX
|
9.3 | pIC50 | 4 | Yes | |
CWBFECUIDZXHBY
|
9.2 | pIC50 | 3 | Yes | |
BKCXBMXTXLGZCV
|
9.2 | pIC50 | 3 | Yes | |
BKCXBMXTXLGZCV
|
9.2 | pIC50 | 3 | Yes | |
BLJPKQXXDFIIFR
|
9.2 | IC50 | 16 | — | |
CYGCWJCVIJAEOL
|
9.2 | pIC50 | 7 | Yes | |
DWSHVVSVJWDKEK
|
9.2 | pIC50 | 3 | Yes | |
FAGYSQSLIMHWHR
|
9.2 | pIC50 | 4 | Yes | |
HHUWJVYTBKEMON
|
9.2 | pIC50 | 5 | Yes | |
HIMQJMWVIJRMHV
|
9.2 | pIC50 | 4 | Yes | |
IBIQLEWQPHHHEE
|
9.2 | pIC50 | 4 | Yes | |
JAVIIUAYGNOEAR
|
9.2 | pIC50 | 4 | Yes |