Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CECSFCKUXJBSMW
|
8.2 | pIC50 | 2 | Yes | |
CECSFCKUXJBSMW
|
8.2 | pIC50 | 2 | Yes | |
FFUQBLRMMDTIAJ
|
8.2 | pIC50 | 4 | Yes | |
GUBQQMYDBCRCTJ
|
8.2 | pIC50 | 4 | Yes | |
IOCQUYQFGCLDTM
|
8.2 | pIC50 | 6 | Yes | |
MTYJWRJHWYZYOK
|
8.2 | pIC50 | 4 | Yes | |
QLSJUBOKAWBLMY
|
8.2 | pIC50 | 5 | Yes | |
RSBCSHUOPBBKNZ
|
8.2 | pIC50 | 3 | Yes | |
SPEYBQKWONGMOH
|
8.2 | pIC50 | 5 | Yes | |
UJXRTXMHXLXLOL
|
8.2 | pIC50 | 4 | Yes | |
ACGLVUUHVAFLSL
|
8.2 | pIC50 | 4 | Yes | |
ACOCIZXLRWIONJ
|
8.2 | pIC50 | 4 | Yes | |
AGZFZUWEZRMIFV
|
8.2 | pIC50 | 3 | Yes | |
AMYPZOHWWHXUFZ
|
8.2 | pIC50 | 3 | Yes | |
AVXVDGLQCDKAHR
|
8.2 | pIC50 | 2 | Yes | |
BSNWTBJRGJXKOF
|
8.2 | pIC50 | 3 | Yes | |
CZOYTUWENNKTEB
|
8.2 | pIC50 | 5 | Yes | |
DNJKYTRZNPUEST
|
8.2 | pIC50 | 3 | Yes | |
DUGZDTXPMNFUOR
|
8.2 | pIC50 | 3 | Yes | |
FDHBUMXEERWSFK
|
8.2 | pIC50 | 3 | Yes | |
FPIUXIZJGYSEDC
|
8.2 | pIC50 | 4 | Yes | |
GKSHXHOOVHLDDC
|
8.2 | pIC50 | 3 | Yes | |
GLNSILZLFCRAHR
|
8.2 | pIC50 | 3 | Yes | |
GYKVWKUDZTYCIL
|
8.2 | pIC50 | 4 | Yes | |
IQXRPQJFASFEKZ
|
8.2 | pIC50 | 3 | Yes | |
JRBRWFNCUIDSLH
|
8.2 | pIC50 | 3 | Yes | |
KMZODUVSKUKAQG
|
8.2 | pIC50 | 5 | Yes | |
KPJDVEHDTNHFPM
|
8.2 | pIC50 | 3 | Yes | |
KQBPCTUKTLMUPL
|
8.2 | pIC50 | 4 | Yes | |
KUBGHMJBEUKTTN
|
8.2 | pIC50 | 3 | Yes | |
LGKMEHLZMDCMTK
|
8.2 | pIC50 | 2 | Yes | |
LTJDGKNETMQCBO
|
8.2 | pIC50 | 3 | Yes | |
LVTDYTBCBYJNAP
|
8.2 | pIC50 | 5 | Yes | |
MEGWHNJGIHFDSO
|
8.2 | pIC50 | 4 | Yes | |
NZRRGHGVIJAYDH
|
8.2 | pIC50 | 3 | Yes | |
OGXPLQPIIFXSCV
|
8.2 | pIC50 | 3 | Yes | |
OTQXKRRISJPTFS
|
8.2 | IC50 | 16 | — | |
PBKRGGSLHOYZBI
|
8.2 | pIC50 | 4 | Yes | |
PECXPDOXZCZHML
|
8.2 | pIC50 | 5 | Yes | |
QTRNBRCYOZEWCV
|
8.2 | pIC50 | 4 | Yes | |
RDSADKNUIYUYDN
|
8.2 | pIC50 | 3 | Yes | |
UHNNGPQIKLRTPI
|
8.2 | pIC50 | 3 | Yes | |
UMNYCEDKFPPMLV
|
8.2 | pIC50 | 3 | Yes | |
UMYBZVYPQATGDV
|
8.2 | pIC50 | 3 | Yes | |
UPQRKLKIHQKKRP
|
8.2 | pIC50 | 2 | Yes | |
VPRDEFURXBNFEY
|
8.2 | pIC50 | 5 | Yes | |
VQATUPWMFYRKSD
|
8.2 | pIC50 | 4 | Yes | |
VWJONQJOSJAUSS
|
8.2 | pIC50 | 3 | Yes | |
WMCJJXHYPNOCMT
|
8.2 | IC50 | 16 | — | |
XDZNGWTVLSNZFM
|
8.2 | pIC50 | 3 | Yes |