Target Details
UniProt ACP18505
Gene SymbolGABRB1
Protein NameGamma-aminobutyric acid receptor subunit beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 5,316
  • Clinical molecules 4981
  • Avg pChEMBL 7.5
Top Co-occurrence Targets
Active Molecules (5,316)
InChIKey pChEMBL Type Targets Clinical
TXWIVULJNOBLNT 8.2 pIC50 3 Yes
UKESULUDTYESMF 8.2 pIC50 3 Yes
URXCUZTXDKQVAL 8.2 pIC50 3 Yes
UWIGEYBKDHPGMV 8.2 pIC50 3 Yes
VVEGAMWEUUKVKL 8.2 pIC50 3 Yes
XHYVDZQPVPOUOG 8.2 pIC50 4 Yes
XLMNAJDPYXDADN 8.2 pIC50 3 Yes
XLMNAJDPYXDADN 8.2 pIC50 3 Yes
XVDJASFHUIQILX 8.2 pIC50 3 Yes
YLMDSHIOZFJIOC 8.2 pIC50 3 Yes
YUSWMAULDXZHPY 8.2 Ki 20
ZOCBCFXUQAYMNS 8.2 pIC50 4 Yes
ZRRVSALMQDOQAX 8.2 Ki 16
DHYYASBDCUAKNN 8.2 pIC50 4 Yes
KXJZCUXKVOHUTN 8.2 pIC50 5 Yes
LZSCCTRKINGQLX 8.2 pIC50 4 Yes
PTTQRLLAHZHAEV 8.2 pIC50 6 Yes
BDISWVKOOATATE 8.2 Ki 16
BJNQKVADRDIKFO 8.2 pIC50 6 Yes
GFNNBHLJANVSQV 8.2 pIC50 7 Yes
GUWYKWYVOAMUBX 8.2 pIC50 4 Yes
IPPCIRPZZWGBBN 8.2 pIC50 4 Yes
LNKZOOJJSXVZGP 8.2 pIC50 4 Yes
AYXPBYVGQSZELF 8.2 pIC50 3 Yes
MVLCAJYSCDCLPF 8.2 pIC50 4 Yes
WDFBMSONXFYEHT 8.2 pIC50 5 Yes
YTUPVOSKWNUXRI 8.2 pIC50 6 Yes
ZNPGUOAVCPGMFY 8.2 pIC50 4 Yes
ZZTHGPFXLVWJQY 8.2 pIC50 4 Yes
APPAUNZXIPSWAS 8.2 pIC50 7 Yes
IXHKQKNNYNMMIN 8.2 pIC50 3 Yes
KIHQVERTLRHJED 8.2 pIC50 3 Yes
ONVKFNZGEFTWQD 8.2 pIC50 4 Yes
QQGSJJXMDWGELG 8.2 pIC50 4 Yes
UVMOSTGNAOREDN 8.2 pIC50 5 Yes
UZHATVNWKBVHPB 8.2 pIC50 3 Yes
DFOLGWDCROPMCI 8.2 pIC50 6 Yes
DTWDCDSAKWSSGY 8.2 pIC50 7 Yes
HAGLWOQGYGIGRZ 8.2 pIC50 4 Yes
QGAJDSWCAJPCOD 8.2 pIC50 4 Yes
RKHXSEWVQGJCRM 8.2 pIC50 3 Yes
RUCGACIRHPJZEV 8.2 pIC50 3 Yes
RZSYRRUMXADKCN 8.2 pIC50 5 Yes
STPPVJHFCUPUSB 8.2 pIC50 3 Yes
TXDBKBXULDSLMV 8.2 pIC50 6 Yes
VJYZIBSNSBDTJT 8.2 pIC50 3 Yes
VLTLYBSKNONSPK 8.2 pIC50 5 Yes
YMCNZULRQVDFCL 8.2 pIC50 4 Yes
YUOOYQDBXTWPKL 8.2 Ki 16
BVMWXWLCRAKYDJ 8.2 pIC50 5 Yes
2D structure