Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXWIVULJNOBLNT
|
8.2 | pIC50 | 3 | Yes | |
UKESULUDTYESMF
|
8.2 | pIC50 | 3 | Yes | |
URXCUZTXDKQVAL
|
8.2 | pIC50 | 3 | Yes | |
UWIGEYBKDHPGMV
|
8.2 | pIC50 | 3 | Yes | |
VVEGAMWEUUKVKL
|
8.2 | pIC50 | 3 | Yes | |
XHYVDZQPVPOUOG
|
8.2 | pIC50 | 4 | Yes | |
XLMNAJDPYXDADN
|
8.2 | pIC50 | 3 | Yes | |
XLMNAJDPYXDADN
|
8.2 | pIC50 | 3 | Yes | |
XVDJASFHUIQILX
|
8.2 | pIC50 | 3 | Yes | |
YLMDSHIOZFJIOC
|
8.2 | pIC50 | 3 | Yes | |
YUSWMAULDXZHPY
|
8.2 | Ki | 20 | — | |
ZOCBCFXUQAYMNS
|
8.2 | pIC50 | 4 | Yes | |
ZRRVSALMQDOQAX
|
8.2 | Ki | 16 | — | |
DHYYASBDCUAKNN
|
8.2 | pIC50 | 4 | Yes | |
KXJZCUXKVOHUTN
|
8.2 | pIC50 | 5 | Yes | |
LZSCCTRKINGQLX
|
8.2 | pIC50 | 4 | Yes | |
PTTQRLLAHZHAEV
|
8.2 | pIC50 | 6 | Yes | |
BDISWVKOOATATE
|
8.2 | Ki | 16 | — | |
BJNQKVADRDIKFO
|
8.2 | pIC50 | 6 | Yes | |
GFNNBHLJANVSQV
|
8.2 | pIC50 | 7 | Yes | |
GUWYKWYVOAMUBX
|
8.2 | pIC50 | 4 | Yes | |
IPPCIRPZZWGBBN
|
8.2 | pIC50 | 4 | Yes | |
LNKZOOJJSXVZGP
|
8.2 | pIC50 | 4 | Yes | |
AYXPBYVGQSZELF
|
8.2 | pIC50 | 3 | Yes | |
MVLCAJYSCDCLPF
|
8.2 | pIC50 | 4 | Yes | |
WDFBMSONXFYEHT
|
8.2 | pIC50 | 5 | Yes | |
YTUPVOSKWNUXRI
|
8.2 | pIC50 | 6 | Yes | |
ZNPGUOAVCPGMFY
|
8.2 | pIC50 | 4 | Yes | |
ZZTHGPFXLVWJQY
|
8.2 | pIC50 | 4 | Yes | |
APPAUNZXIPSWAS
|
8.2 | pIC50 | 7 | Yes | |
IXHKQKNNYNMMIN
|
8.2 | pIC50 | 3 | Yes | |
KIHQVERTLRHJED
|
8.2 | pIC50 | 3 | Yes | |
ONVKFNZGEFTWQD
|
8.2 | pIC50 | 4 | Yes | |
QQGSJJXMDWGELG
|
8.2 | pIC50 | 4 | Yes | |
UVMOSTGNAOREDN
|
8.2 | pIC50 | 5 | Yes | |
UZHATVNWKBVHPB
|
8.2 | pIC50 | 3 | Yes | |
DFOLGWDCROPMCI
|
8.2 | pIC50 | 6 | Yes | |
DTWDCDSAKWSSGY
|
8.2 | pIC50 | 7 | Yes | |
HAGLWOQGYGIGRZ
|
8.2 | pIC50 | 4 | Yes | |
QGAJDSWCAJPCOD
|
8.2 | pIC50 | 4 | Yes | |
RKHXSEWVQGJCRM
|
8.2 | pIC50 | 3 | Yes | |
RUCGACIRHPJZEV
|
8.2 | pIC50 | 3 | Yes | |
RZSYRRUMXADKCN
|
8.2 | pIC50 | 5 | Yes | |
STPPVJHFCUPUSB
|
8.2 | pIC50 | 3 | Yes | |
TXDBKBXULDSLMV
|
8.2 | pIC50 | 6 | Yes | |
VJYZIBSNSBDTJT
|
8.2 | pIC50 | 3 | Yes | |
VLTLYBSKNONSPK
|
8.2 | pIC50 | 5 | Yes | |
YMCNZULRQVDFCL
|
8.2 | pIC50 | 4 | Yes | |
YUOOYQDBXTWPKL
|
8.2 | Ki | 16 | — | |
BVMWXWLCRAKYDJ
|
8.2 | pIC50 | 5 | Yes |