Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDOHHPHBVZUFJE
|
9.5 | pIC50 | 2 | Yes | |
NOJQAHBGMABANB
|
9.5 | pIC50 | 3 | Yes | |
ORYVQNZEUSJYKM
|
9.5 | pIC50 | 4 | Yes | |
SNVIUSFXXHRDCP
|
9.5 | pIC50 | 3 | Yes | |
SXNATFXZAWSPSE
|
9.5 | pIC50 | 4 | Yes | |
UITYJROEGAFMRK
|
9.5 | pIC50 | 2 | Yes | |
UZOOIPXOYYJULJ
|
9.5 | pIC50 | 4 | Yes | |
VGFUTXNYAMRULN
|
9.5 | pIC50 | 4 | Yes | |
YMECUEKBIBTNRW
|
9.5 | pIC50 | 7 | Yes | |
CGNLKIUQLVMBMO
|
9.5 | pIC50 | 4 | Yes | |
XMACBUOIMKGMRP
|
9.5 | pIC50 | 4 | Yes | |
ZPPXQVFYCAJAFB
|
9.5 | pIC50 | 4 | Yes | |
RIUHJWNFKOJLRS
|
9.4 | pIC50 | 4 | Yes | |
NJFCQEZGMMGGKH
|
9.4 | pIC50 | 2 | Yes | |
IIACRCGMVDHOTQ
|
9.4 | pIC50 | 5 | Yes | |
PNGNVUOPWWBBSY
|
9.4 | pIC50 | 4 | Yes | |
AUBNMBTYWOGQSO
|
9.4 | pIC50 | 4 | Yes | |
BQJRUJTZSGYBEZ
|
9.4 | pIC50 | 13 | Yes | |
CHXGEQWNFRZIOC
|
9.4 | pIC50 | 3 | Yes | |
COJFASLRENZFLP
|
9.4 | pIC50 | 4 | Yes | |
JCPGSSZRKQLWNX
|
9.4 | pIC50 | 4 | Yes | |
KRKRBIVNILCKBI
|
9.4 | pIC50 | 4 | Yes | |
PYWHZNIQLVXCCU
|
9.4 | pIC50 | 4 | Yes | |
QFWCWQVDLDGJME
|
9.4 | pIC50 | 4 | Yes | |
QUUNMICPMYIHFS
|
9.4 | IC50 | 16 | — | |
RHJPBGWFGOAEID
|
9.4 | pIC50 | 8 | Yes | |
UOZGUWHPVZIRDP
|
9.4 | pIC50 | 4 | Yes | |
VMDUABMKBUKKPG
|
9.4 | IC50 | 16 | — | |
WLGDFYOOSGHIPS
|
9.4 | pIC50 | 4 | Yes | |
XBLYYDDTTORRLT
|
9.4 | pIC50 | 4 | Yes | |
XGALLCVXEZPNRQ
|
9.4 | pIC50 | 39 | Yes | |
XMOVBRJIOBDWGP
|
9.4 | pIC50 | 3 | Yes | |
ZFDWXHMWRIPYFL
|
9.4 | pIC50 | 4 | Yes | |
CLYUNXJFERDYMU
|
9.4 | pIC50 | 4 | Yes | |
CVYGUAJDEHYTCH
|
9.4 | pIC50 | 2 | Yes | |
AFAUDWQMESQGPR
|
9.4 | pIC50 | 4 | Yes | |
DVJGXMUWYFGXAS
|
9.4 | pIC50 | 4 | Yes | |
QJSMFUTULGSHNQ
|
9.4 | pIC50 | 4 | Yes | |
BWHGYXORZLZUIK
|
9.3 | pIC50 | 2 | Yes | |
HMWBDNPYGWPLRR
|
9.3 | pIC50 | 2 | Yes | |
MCXANZUXLRCMDM
|
9.3 | pIC50 | 2 | Yes | |
NWUCBGDFEQGJTP
|
9.3 | pIC50 | 2 | Yes | |
PXEXUKNUARXICD
|
9.3 | pIC50 | 2 | Yes | |
XKENJWNGLCKOBP
|
9.3 | IC50 | 16 | — | |
YMUNHDVCHMLVMN
|
9.3 | pIC50 | 4 | Yes | |
TUWAJCMXXFZLOS
|
9.3 | pIC50 | 4 | Yes | |
XIESSJVMWNJCGZ
|
9.3 | pIC50 | 4 | Yes | |
LXRGAVBXYQAUEY
|
9.3 | pIC50 | 4 | Yes | |
KYKWZUMHVAPNQH
|
9.3 | pIC50 | 4 | Yes | |
NJUMMJUUDUYSKB
|
9.3 | IC50 | 16 | — |