Target Details
UniProt ACP18505
Gene SymbolGABRB1
Protein NameGamma-aminobutyric acid receptor subunit beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 5,316
  • Clinical molecules 4981
  • Avg pChEMBL 7.5
Top Co-occurrence Targets
Active Molecules (5,316)
InChIKey pChEMBL Type Targets Clinical
NDOHHPHBVZUFJE 9.5 pIC50 2 Yes
NOJQAHBGMABANB 9.5 pIC50 3 Yes
ORYVQNZEUSJYKM 9.5 pIC50 4 Yes
SNVIUSFXXHRDCP 9.5 pIC50 3 Yes
SXNATFXZAWSPSE 9.5 pIC50 4 Yes
UITYJROEGAFMRK 9.5 pIC50 2 Yes
UZOOIPXOYYJULJ 9.5 pIC50 4 Yes
VGFUTXNYAMRULN 9.5 pIC50 4 Yes
YMECUEKBIBTNRW 9.5 pIC50 7 Yes
CGNLKIUQLVMBMO 9.5 pIC50 4 Yes
XMACBUOIMKGMRP 9.5 pIC50 4 Yes
ZPPXQVFYCAJAFB 9.5 pIC50 4 Yes
RIUHJWNFKOJLRS 9.4 pIC50 4 Yes
NJFCQEZGMMGGKH 9.4 pIC50 2 Yes
IIACRCGMVDHOTQ 9.4 pIC50 5 Yes
PNGNVUOPWWBBSY 9.4 pIC50 4 Yes
AUBNMBTYWOGQSO 9.4 pIC50 4 Yes
BQJRUJTZSGYBEZ 9.4 pIC50 13 Yes
CHXGEQWNFRZIOC 9.4 pIC50 3 Yes
COJFASLRENZFLP 9.4 pIC50 4 Yes
JCPGSSZRKQLWNX 9.4 pIC50 4 Yes
KRKRBIVNILCKBI 9.4 pIC50 4 Yes
PYWHZNIQLVXCCU 9.4 pIC50 4 Yes
QFWCWQVDLDGJME 9.4 pIC50 4 Yes
QUUNMICPMYIHFS 9.4 IC50 16
RHJPBGWFGOAEID 9.4 pIC50 8 Yes
UOZGUWHPVZIRDP 9.4 pIC50 4 Yes
VMDUABMKBUKKPG 9.4 IC50 16
WLGDFYOOSGHIPS 9.4 pIC50 4 Yes
XBLYYDDTTORRLT 9.4 pIC50 4 Yes
XGALLCVXEZPNRQ 9.4 pIC50 39 Yes
XMOVBRJIOBDWGP 9.4 pIC50 3 Yes
ZFDWXHMWRIPYFL 9.4 pIC50 4 Yes
CLYUNXJFERDYMU 9.4 pIC50 4 Yes
CVYGUAJDEHYTCH 9.4 pIC50 2 Yes
AFAUDWQMESQGPR 9.4 pIC50 4 Yes
DVJGXMUWYFGXAS 9.4 pIC50 4 Yes
QJSMFUTULGSHNQ 9.4 pIC50 4 Yes
BWHGYXORZLZUIK 9.3 pIC50 2 Yes
HMWBDNPYGWPLRR 9.3 pIC50 2 Yes
MCXANZUXLRCMDM 9.3 pIC50 2 Yes
NWUCBGDFEQGJTP 9.3 pIC50 2 Yes
PXEXUKNUARXICD 9.3 pIC50 2 Yes
XKENJWNGLCKOBP 9.3 IC50 16
YMUNHDVCHMLVMN 9.3 pIC50 4 Yes
TUWAJCMXXFZLOS 9.3 pIC50 4 Yes
XIESSJVMWNJCGZ 9.3 pIC50 4 Yes
LXRGAVBXYQAUEY 9.3 pIC50 4 Yes
KYKWZUMHVAPNQH 9.3 pIC50 4 Yes
NJUMMJUUDUYSKB 9.3 IC50 16
2D structure