Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SZJIXBKHTOPEKG
|
8.2 | pIC50 | 6 | Yes | |
XWSXOSVPGQCPDX
|
8.2 | pIC50 | 4 | Yes | |
ZZRJPSUBAGGGKW
|
8.2 | pIC50 | 4 | Yes | |
HXXGIDLDLCJJDB
|
8.2 | pIC50 | 4 | Yes | |
KTYJLJQTVQUQCU
|
8.2 | pIC50 | 3 | Yes | |
MFDXIQNXGJGENZ
|
8.2 | pIC50 | 4 | Yes | |
AIBKIFHSQQYXLG
|
8.2 | pIC50 | 4 | Yes | |
AQULIWLSIITFDZ
|
8.2 | pIC50 | 3 | Yes | |
BTLWEEGNXUJKKB
|
8.2 | IC50 | 16 | — | |
CLNZVLYLUNHHJW
|
8.2 | pIC50 | 6 | Yes | |
CWWNTMKCOPSSCO
|
8.2 | pIC50 | 3 | Yes | |
DPAMLAKLEWYMGF
|
8.2 | pIC50 | 3 | Yes | |
DYFALINGOOHZSX
|
8.2 | pIC50 | 4 | Yes | |
FCHMBSURKDQMKR
|
8.2 | pIC50 | 3 | Yes | |
FDIUAXKVVLMXEX
|
8.2 | pIC50 | 4 | Yes | |
GCQZFVAHUZIDRP
|
8.2 | pIC50 | 4 | Yes | |
HRABVSOIJXZING
|
8.2 | pIC50 | 3 | Yes | |
HZYKIFUDWNXIGV
|
8.2 | pIC50 | 3 | Yes | |
JBIMYQPMDQEGTO
|
8.2 | pIC50 | 4 | Yes | |
JSCKSAAAUCSGDM
|
8.2 | pIC50 | 4 | Yes | |
KIVQXKXZISOGBE
|
8.2 | Ki | 17 | — | |
KJBZSRKWLOOUML
|
8.2 | pIC50 | 4 | Yes | |
KSTBRFAYWXRXEX
|
8.2 | pIC50 | 2 | Yes | |
KTKGBEYRKDMODK
|
8.2 | pIC50 | 5 | Yes | |
KYOHBMZTYDOMED
|
8.2 | pIC50 | 3 | Yes | |
LDKNESVHONOUJK
|
8.2 | pIC50 | 3 | Yes | |
MLPLUGYJGCEXRH
|
8.2 | pIC50 | 3 | Yes | |
MMOGWZPLKFNWRO
|
8.2 | pIC50 | 3 | Yes | |
MVLSXWFLBKVSDR
|
8.2 | pIC50 | 5 | Yes | |
NKIYALPHXLYICR
|
8.2 | IC50 | 16 | — | |
NLFHVYVHJAOOCP
|
8.2 | pIC50 | 4 | Yes | |
NRVQBQRMJRRVGL
|
8.2 | pIC50 | 4 | Yes | |
ODCTUBPUHXFKPX
|
8.2 | pIC50 | 3 | Yes | |
ODCTUBPUHXFKPX
|
8.2 | pIC50 | 3 | Yes | |
OJIHLNZBFOHKCT
|
8.2 | pIC50 | 3 | Yes | |
ONXVIWURXZZGRP
|
8.2 | pIC50 | 5 | Yes | |
OQSPFWYBYACCQS
|
8.2 | pIC50 | 2 | Yes | |
OYAOKYMFRYPRMN
|
8.2 | pIC50 | 3 | Yes | |
PCSLANZLBGQJII
|
8.2 | pIC50 | 3 | Yes | |
PCWJJXZGAQSUKE
|
8.2 | pIC50 | 4 | Yes | |
PMFBLJXNSAHZSG
|
8.2 | pIC50 | 3 | Yes | |
QADHLRWLCPCEKT
|
8.2 | pIC50 | 5 | Yes | |
QAYAKBOPHPQBCX
|
8.2 | pIC50 | 3 | Yes | |
QIPCVTBKOSBJFB
|
8.2 | pIC50 | 4 | Yes | |
QQWUGDVOUVUTOY
|
8.2 | pIC50 | 231 | Yes | |
QSCXUBQIKQZMSG
|
8.2 | pIC50 | 3 | Yes | |
RSGBEHCRTCQOMK
|
8.2 | pIC50 | 3 | Yes | |
RZZMXYDKPZINQM
|
8.2 | pIC50 | 4 | Yes | |
SNNNDCMXZYWCCI
|
8.2 | pIC50 | 4 | Yes | |
TWHYYPIAGPPMKW
|
8.2 | pIC50 | 3 | Yes |