Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IOCHAGJKMZSJCF
|
8.4 | pIC50 | 3 | Yes | |
IQSIOBJHBCJWRX
|
8.4 | pIC50 | 4 | Yes | |
JDAULUKGZUDSNK
|
8.4 | pIC50 | 3 | Yes | |
JGJPGWCZPKIATB
|
8.4 | pIC50 | 4 | Yes | |
JTYYMOMTGZSRFM
|
8.4 | IC50 | 16 | — | |
KCQUSTRLBHEXNM
|
8.4 | pIC50 | 3 | Yes | |
LMXUGQJMQSMLIQ
|
8.4 | Ki | 17 | — | |
LOLPPWBBNUVNQZ
|
8.4 | pIC50 | 97 | Yes | |
LTOXHEYDPJRTGT
|
8.4 | pIC50 | 3 | Yes | |
MRGJPQCXQRRGHN
|
8.4 | pIC50 | 3 | Yes | |
MVJGBJOMTDVGRA
|
8.4 | pIC50 | 3 | Yes | |
NOOBQTYVTDBXTL
|
8.4 | pIC50 | 12 | Yes | |
ONSKSKMJNHEONW
|
8.4 | pIC50 | 3 | Yes | |
OQJYJENHHOZHPV
|
8.4 | pIC50 | 4 | Yes | |
PITUMGJELDUJEZ
|
8.4 | pIC50 | 3 | Yes | |
PVSWUJNBHHDSMN
|
8.4 | pIC50 | 5 | Yes | |
QLJSQRVXMOGBQC
|
8.4 | pIC50 | 3 | Yes | |
QOPZRTKUPLJDOO
|
8.4 | pIC50 | 3 | Yes | |
QYZVZGPAIPNEDN
|
8.4 | pIC50 | 4 | Yes | |
RCMWOTCXCCDSQD
|
8.4 | pIC50 | 3 | Yes | |
RYZHAZRYCADWGS
|
8.4 | pIC50 | 3 | Yes | |
RYZHAZRYCADWGS
|
8.4 | pIC50 | 3 | Yes | |
SSAWUSNORQCOED
|
8.4 | pIC50 | 3 | Yes | |
UDAQLYMFTARBIE
|
8.4 | pIC50 | 4 | Yes | |
UFTKNTUWDMJOIX
|
8.4 | IC50 | 16 | — | |
UNFQCVGQBRBWHG
|
8.4 | pIC50 | 4 | Yes | |
UULFOYXSWNADTF
|
8.4 | IC50 | 16 | — | |
VQVMRAKFGMGHHR
|
8.4 | pIC50 | 4 | Yes | |
WCSKQUVECCMYCW
|
8.4 | pIC50 | 3 | Yes | |
XQANRQYTWBLZNV
|
8.4 | pIC50 | 3 | Yes | |
YSLYGNKZBSKTIF
|
8.4 | pIC50 | 4 | Yes | |
ZDUQAOBGFYJNTD
|
8.4 | pIC50 | 3 | Yes | |
ZGQCWNCUDXFCQJ
|
8.4 | pIC50 | 3 | Yes | |
ZIQFYVPVJZEOFS
|
8.4 | pIC50 | 9 | Yes | |
ZRXRKAYJXHMMIU
|
8.4 | pIC50 | 3 | Yes | |
IBRPSHUYWHRYQA
|
8.4 | pIC50 | 4 | Yes | |
JLALBSSBYZKONR
|
8.4 | pIC50 | 4 | Yes | |
PBCZSGKMGDDXIJ
|
8.4 | pIC50 | 68 | Yes | |
RRDYXHHANIMNOJ
|
8.4 | pIC50 | 4 | Yes | |
SHANKUTWRXLKIV
|
8.4 | pIC50 | 4 | Yes | |
UGWRDFFACAHWMU
|
8.4 | pIC50 | 4 | Yes | |
VPTXVOFVTSHNSY
|
8.4 | pIC50 | 4 | Yes | |
YQYRRRVQWIMSFP
|
8.4 | Ki | 5 | — | |
DOWMHKGEUBGVCN
|
8.4 | pIC50 | 4 | Yes | |
DQDHQICCPRPMJN
|
8.4 | pIC50 | 3 | Yes | |
GSWRTFGMHRKLKT
|
8.4 | pIC50 | 14 | Yes | |
LRXFNZWLYRPLKR
|
8.4 | pIC50 | 3 | Yes | |
MKNXZRAKHYWDOS
|
8.4 | IC50 | 16 | — | |
XQUJTESAXUTXNH
|
8.4 | Ki | 16 | — | |
ZBRROTSBDAODQD
|
8.4 | pIC50 | 7 | Yes |