Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WWMGAPRXPIKGFI
|
8.5 | pIC50 | 4 | Yes | |
XOISNQGKACZMII
|
8.5 | pIC50 | 3 | Yes | |
CKIDATLRUHCUAK
|
8.5 | pIC50 | 3 | Yes | |
DNOMWUYUDHLCAY
|
8.5 | pIC50 | 4 | Yes | |
NBTXJDAHLMMIGY
|
8.5 | pIC50 | 4 | Yes | |
NTSDFQBCKBKNJW
|
8.5 | pIC50 | 4 | Yes | |
PLZOWXHKTJJSQR
|
8.5 | pIC50 | 3 | Yes | |
VAYMOEILCNGWNC
|
8.5 | pIC50 | 4 | Yes | |
YMMHAHMATMOTRF
|
8.5 | pIC50 | 4 | Yes | |
ZFZLLLFBWBJQJN
|
8.5 | pIC50 | 2 | Yes | |
RFSFIDGEFVXSQM
|
8.4 | pIC50 | 12 | Yes | |
CBUXLBQVPVOWAL
|
8.4 | pIC50 | 3 | Yes | |
HBMCAYMASSWIBL
|
8.4 | pIC50 | 3 | Yes | |
IAOYQLOKTBWIQA
|
8.4 | pIC50 | 3 | Yes | |
JHVBNAPBDHLDMW
|
8.4 | pIC50 | 5 | Yes | |
MVBVNOZDVRVMNH
|
8.4 | IC50 | 16 | — | |
PESQNLUMBCKJOK
|
8.4 | pIC50 | 4 | Yes | |
PMNXCGMIMVLCRP
|
8.4 | pIC50 | 2 | Yes | |
SFNUIOHIVSABQR
|
8.4 | pIC50 | 3 | Yes | |
WOAYEAZNVGHCDU
|
8.4 | pIC50 | 6 | Yes | |
XSWVYGHDSDATRA
|
8.4 | pIC50 | 4 | Yes | |
BDKWTFFBJKKPEK
|
8.4 | pIC50 | 4 | Yes | |
BRMVQUBTTGWVNX
|
8.4 | pIC50 | 4 | Yes | |
CDRJTNGWNAODES
|
8.4 | pIC50 | 3 | Yes | |
SNPIZVSBDKYJEJ
|
8.4 | pIC50 | 2 | Yes | |
VCETZICKGRMEAH
|
8.4 | pIC50 | 4 | Yes | |
CNAUCDPBQHEQHN
|
8.4 | pIC50 | 3 | Yes | |
CRPUDAVZTZIKMJ
|
8.4 | pIC50 | 7 | Yes | |
HMDBQCJZLHHNQM
|
8.4 | pIC50 | 4 | Yes | |
OBIWZXNLWSUNOP
|
8.4 | pIC50 | 4 | Yes | |
QNHUAOAFGVCXEA
|
8.4 | pIC50 | 4 | Yes | |
UCJGJABZCDBEDK
|
8.4 | pIC50 | 4 | Yes | |
YMMHAHMATMOTRF
|
8.4 | pIC50 | 4 | Yes | |
YPZSGGRHSBFMRE
|
8.4 | pIC50 | 4 | Yes | |
NHJGGBOIASKXGY
|
8.4 | pIC50 | 4 | Yes | |
ZMYUKKKHJVNBAM
|
8.4 | pIC50 | 5 | Yes | |
AAXOJAXCFROOJI
|
8.4 | pIC50 | 3 | Yes | |
ACUNYYFYYWOKOD
|
8.4 | IC50 | 16 | — | |
AXPGZURVLRWNBR
|
8.4 | Ki | 16 | — | |
BAOYJOYLDRTITD
|
8.4 | pIC50 | 3 | Yes | |
BLPILBAOBRFNLK
|
8.4 | pIC50 | 4 | Yes | |
BZVWONIGXAYZIT
|
8.4 | IC50 | 16 | — | |
CDWXZILKRXSANI
|
8.4 | IC50 | 16 | — | |
DYSDYZCGZCYPCT
|
8.4 | IC50 | 16 | — | |
FNICBGZPBTURDA
|
8.4 | pIC50 | 4 | Yes | |
HHMSOLCNQSSGIC
|
8.4 | pIC50 | 3 | Yes | |
HZPYQCSGTTZVLW
|
8.4 | pIC50 | 4 | Yes | |
ICVMJXJRTYOTJH
|
8.4 | pIC50 | 3 | Yes | |
IMTGUGLNCFNYNG
|
8.4 | pIC50 | 3 | Yes | |
IMTGUGLNCFNYNG
|
8.4 | pIC50 | 3 | Yes |