Target Details
UniProt ACP18505
Gene SymbolGABRB1
Protein NameGamma-aminobutyric acid receptor subunit beta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 5,316
  • Clinical molecules 4981
  • Avg pChEMBL 7.5
Top Co-occurrence Targets
Active Molecules (5,316)
InChIKey pChEMBL Type Targets Clinical
WWMGAPRXPIKGFI 8.5 pIC50 4 Yes
XOISNQGKACZMII 8.5 pIC50 3 Yes
CKIDATLRUHCUAK 8.5 pIC50 3 Yes
DNOMWUYUDHLCAY 8.5 pIC50 4 Yes
NBTXJDAHLMMIGY 8.5 pIC50 4 Yes
NTSDFQBCKBKNJW 8.5 pIC50 4 Yes
PLZOWXHKTJJSQR 8.5 pIC50 3 Yes
VAYMOEILCNGWNC 8.5 pIC50 4 Yes
YMMHAHMATMOTRF 8.5 pIC50 4 Yes
ZFZLLLFBWBJQJN 8.5 pIC50 2 Yes
RFSFIDGEFVXSQM 8.4 pIC50 12 Yes
CBUXLBQVPVOWAL 8.4 pIC50 3 Yes
HBMCAYMASSWIBL 8.4 pIC50 3 Yes
IAOYQLOKTBWIQA 8.4 pIC50 3 Yes
JHVBNAPBDHLDMW 8.4 pIC50 5 Yes
MVBVNOZDVRVMNH 8.4 IC50 16
PESQNLUMBCKJOK 8.4 pIC50 4 Yes
PMNXCGMIMVLCRP 8.4 pIC50 2 Yes
SFNUIOHIVSABQR 8.4 pIC50 3 Yes
WOAYEAZNVGHCDU 8.4 pIC50 6 Yes
XSWVYGHDSDATRA 8.4 pIC50 4 Yes
BDKWTFFBJKKPEK 8.4 pIC50 4 Yes
BRMVQUBTTGWVNX 8.4 pIC50 4 Yes
CDRJTNGWNAODES 8.4 pIC50 3 Yes
SNPIZVSBDKYJEJ 8.4 pIC50 2 Yes
VCETZICKGRMEAH 8.4 pIC50 4 Yes
CNAUCDPBQHEQHN 8.4 pIC50 3 Yes
CRPUDAVZTZIKMJ 8.4 pIC50 7 Yes
HMDBQCJZLHHNQM 8.4 pIC50 4 Yes
OBIWZXNLWSUNOP 8.4 pIC50 4 Yes
QNHUAOAFGVCXEA 8.4 pIC50 4 Yes
UCJGJABZCDBEDK 8.4 pIC50 4 Yes
YMMHAHMATMOTRF 8.4 pIC50 4 Yes
YPZSGGRHSBFMRE 8.4 pIC50 4 Yes
NHJGGBOIASKXGY 8.4 pIC50 4 Yes
ZMYUKKKHJVNBAM 8.4 pIC50 5 Yes
AAXOJAXCFROOJI 8.4 pIC50 3 Yes
ACUNYYFYYWOKOD 8.4 IC50 16
AXPGZURVLRWNBR 8.4 Ki 16
BAOYJOYLDRTITD 8.4 pIC50 3 Yes
BLPILBAOBRFNLK 8.4 pIC50 4 Yes
BZVWONIGXAYZIT 8.4 IC50 16
CDWXZILKRXSANI 8.4 IC50 16
DYSDYZCGZCYPCT 8.4 IC50 16
FNICBGZPBTURDA 8.4 pIC50 4 Yes
HHMSOLCNQSSGIC 8.4 pIC50 3 Yes
HZPYQCSGTTZVLW 8.4 pIC50 4 Yes
ICVMJXJRTYOTJH 8.4 pIC50 3 Yes
IMTGUGLNCFNYNG 8.4 pIC50 3 Yes
IMTGUGLNCFNYNG 8.4 pIC50 3 Yes
2D structure