Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VLRGJZDVGRNUEG
|
8.5 | pIC50 | 3 | Yes | |
ZEGZELDRYWOPRH
|
8.5 | pIC50 | 5 | Yes | |
ZHYYNYNDPMTVTM
|
8.5 | pIC50 | 3 | Yes | |
ZSOQJLDYHKQACD
|
8.5 | pIC50 | 4 | Yes | |
FGXXHFWGZTYOIF
|
8.5 | pIC50 | 4 | Yes | |
ABEINLXYVVBZFJ
|
8.5 | pIC50 | 3 | Yes | |
AGMWSULMQRTJAC
|
8.5 | pIC50 | 3 | Yes | |
AQLSMJNYPXRRTF
|
8.5 | pIC50 | 2 | Yes | |
AUURCJRXNDZHEQ
|
8.5 | pIC50 | 4 | Yes | |
BEXPELAOVIOQHQ
|
8.5 | pIC50 | 3 | Yes | |
BFGNFBFKLUVDAE
|
8.5 | pIC50 | 3 | Yes | |
BIHDKIAANBTOQT
|
8.5 | pIC50 | 3 | Yes | |
BMZKCTYVBYFWRQ
|
8.5 | pIC50 | 3 | Yes | |
DCQUEYKYABNNDA
|
8.5 | pIC50 | 5 | Yes | |
DGOSXPMLHQFJNM
|
8.5 | pIC50 | 3 | Yes | |
DJZWACVLMZUPTI
|
8.5 | pIC50 | 3 | Yes | |
DSODZSDBFKQUST
|
8.5 | pIC50 | 4 | Yes | |
FLDXQSCXJKEXJF
|
8.5 | pIC50 | 4 | Yes | |
FLYNZEXUURBXAW
|
8.5 | pIC50 | 6 | Yes | |
FMHTWDQAFBPUBC
|
8.5 | pIC50 | 3 | Yes | |
GGHZQYDERZQJFP
|
8.5 | pIC50 | 4 | Yes | |
GMFHJKFOVOFXCU
|
8.5 | pIC50 | 3 | Yes | |
GNWBLLYJQXKPIP
|
8.5 | pIC50 | 4 | Yes | |
GXCDFQARGZTHCW
|
8.5 | pIC50 | 4 | Yes | |
HBVCBMSBBJBRRW
|
8.5 | pIC50 | 4 | Yes | |
HCRKCZRJWPKOAR
|
8.5 | pIC50 | 18 | Yes | |
HMQTZLWTWCWYRU
|
8.5 | pIC50 | 4 | Yes | |
HSLBNURTOUIFTB
|
8.5 | pIC50 | 3 | Yes | |
HVBWXXIYKVDHBO
|
8.5 | pIC50 | 3 | Yes | |
IHRUNMOVLQBVOV
|
8.5 | pIC50 | 3 | Yes | |
ILJNEBRGMAWPTI
|
8.5 | pIC50 | 3 | Yes | |
IXHHOJONZMCEDC
|
8.5 | pIC50 | 3 | Yes | |
JSBXKENODQYJRW
|
8.5 | pIC50 | 3 | Yes | |
KJMALBRUCRDMTE
|
8.5 | pIC50 | 6 | Yes | |
KVKYGVOAHGNAKZ
|
8.5 | IC50 | 17 | — | |
LACIBZRFAYFTOV
|
8.5 | pIC50 | 4 | Yes | |
LDZKSFIAAKAVTR
|
8.5 | pIC50 | 3 | Yes | |
LENHHZQGSWCZJW
|
8.5 | Ki | 16 | — | |
LPAODQAWVMEXKR
|
8.5 | IC50 | 16 | — | |
LSXMKXXXTANXHO
|
8.5 | pIC50 | 3 | Yes | |
MSZBMHGVHMVLSL
|
8.5 | pIC50 | 3 | Yes | |
NEOUOHDNZDRDNJ
|
8.5 | IC50 | 16 | — | |
NQSAAPCTPUNSPD
|
8.5 | pIC50 | 4 | Yes | |
OFANLVRXZQQUMO
|
8.5 | pIC50 | 3 | Yes | |
OSICGNXFPBDFRO
|
8.5 | pIC50 | 3 | Yes | |
OUZWUKMCLIBBOG
|
8.5 | pIC50 | 17 | Yes | |
PEONKJNVFIKXTH
|
8.5 | pIC50 | 4 | Yes | |
PIRRYRRDDTYFPP
|
8.5 | pIC50 | 4 | Yes | |
QIZPCEVRKTWHIE
|
8.5 | IC50 | 16 | — | |
QKRCKJHTQMYVMG
|
8.5 | pIC50 | 3 | Yes |