Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQBIOEFDDDEARX
|
8.6 | pIC50 | 4 | Yes | |
ZOCSXAVNDGMNBV
|
8.6 | IC50 | 16 | — | |
DEFIOUDVRMACDV
|
8.6 | pIC50 | 4 | Yes | |
FCIILWHQWNLPJU
|
8.6 | pIC50 | 4 | Yes | |
HHVMWRVANSDUKF
|
8.6 | pIC50 | 4 | Yes | |
HMRMTWUTVVIJSI
|
8.6 | pIC50 | 4 | Yes | |
HOUIRAFTHIMUSN
|
8.6 | pIC50 | 7 | Yes | |
JGIGPQNAVZRGNQ
|
8.6 | pIC50 | 4 | Yes | |
JWJOTENAMICLJG
|
8.6 | pIC50 | 4 | Yes | |
KCOSTVZZMPPIOT
|
8.6 | pIC50 | 3 | Yes | |
MRGUGRIOWDDLNC
|
8.6 | pIC50 | 4 | Yes | |
PNISVVXQFRITLW
|
8.6 | pIC50 | 3 | Yes | |
ZRHZEPFBMCFVEY
|
8.6 | pIC50 | 4 | Yes | |
COOZRRUJSWPFHC
|
8.6 | pIC50 | 3 | Yes | |
DXLDXLIYYQFLKD
|
8.6 | pIC50 | 4 | Yes | |
IDSZLHFEKAUIOL
|
8.6 | pIC50 | 7 | Yes | |
IZGMIMKTZXSTLH
|
8.6 | pIC50 | 4 | Yes | |
LBHMZZJMZZTTAJ
|
8.6 | pIC50 | 4 | Yes | |
MOQPSDNFBMURQO
|
8.6 | pIC50 | 4 | Yes | |
NIYUBSMBQZFXKI
|
8.6 | pIC50 | 5 | Yes | |
QIGGJMQSVPHSJB
|
8.6 | pIC50 | 16 | Yes | |
QMDVSLSBTALLFL
|
8.6 | pIC50 | 4 | Yes | |
QYUUNIHMDGHUKF
|
8.6 | pIC50 | 4 | Yes | |
VUQWRXYPRNBJPA
|
8.6 | pIC50 | 4 | Yes | |
YHEHVRSGKUYDON
|
8.6 | pIC50 | 4 | Yes | |
DHZJVHCWDITFSE
|
8.6 | pIC50 | 4 | Yes | |
LNBPRSYIRUMTPD
|
8.6 | pIC50 | 3 | Yes | |
OEVSLFVSLIUCMB
|
8.6 | pIC50 | 4 | Yes | |
UQRWUYACRDDBAE
|
8.6 | pIC50 | 4 | Yes | |
WJSKTFAFISQDLB
|
8.6 | pIC50 | 4 | Yes | |
XCDFAEWNVRKGJA
|
8.6 | pIC50 | 4 | Yes | |
ZXWAFSSPWCHAJT
|
8.6 | pIC50 | 10 | Yes | |
HLXZJWIQXIKPRD
|
8.6 | pIC50 | 4 | Yes | |
KTSURNWKXITSNO
|
8.6 | pIC50 | 5 | Yes | |
MASOXJRADXYGSF
|
8.6 | pIC50 | 4 | Yes | |
MEBNSJCLFXPYII
|
8.6 | pIC50 | 3 | Yes | |
NSSOSHDCWCMNDM
|
8.6 | pIC50 | 4 | Yes | |
XTQWBGVHINEJTO
|
8.6 | pIC50 | 4 | Yes | |
CHIFCDOIPRCHCF
|
8.6 | IC50 | 16 | — | |
CHQPOBHNDRMXFK
|
8.6 | Ki | 18 | — | |
FRBSOYMIYWABCH
|
8.6 | pIC50 | 2 | Yes | |
NVVASLWKXTZLJN
|
8.6 | pIC50 | 3 | Yes | |
RLXHHKSCSSXJLX
|
8.6 | pIC50 | 3 | Yes | |
SIJIWSROAVIHBN
|
8.6 | pIC50 | 4 | Yes | |
TWZNCTCQAGRUGQ
|
8.6 | pIC50 | 4 | Yes | |
VFNJKWBUAUKQIJ
|
8.6 | pIC50 | 3 | Yes | |
VLJUOFGVEJAFFK
|
8.6 | pIC50 | 4 | Yes | |
DWLVUAOJOFAURW
|
8.5 | pIC50 | 3 | Yes | |
JSGFVHXKEVDABH
|
8.5 | pIC50 | 4 | Yes | |
PFXDRFNBOIJAJH
|
8.5 | pIC50 | 3 | Yes |