Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBYHIUUMRHTEFF
|
8.7 | pIC50 | 4 | Yes | |
UQDOACBQOXYBML
|
8.7 | pIC50 | 4 | Yes | |
VSKDFCJBACLKIC
|
8.7 | pIC50 | 4 | Yes | |
VTGCXQMCXKWQQC
|
8.7 | pIC50 | 4 | Yes | |
VUNIFGGEGAVCOL
|
8.7 | pIC50 | 3 | Yes | |
WIXIWLDQHOAOLL
|
8.7 | pIC50 | 3 | Yes | |
WKGYLLVUZFUDMJ
|
8.7 | pIC50 | 4 | Yes | |
WSTRMUBDMCVGEG
|
8.7 | pIC50 | 3 | Yes | |
WVZXXBYXJNDMGS
|
8.7 | pIC50 | 5 | Yes | |
XIIPLMMVMAKDTM
|
8.7 | pIC50 | 4 | Yes | |
XKHSVUSPZVNCOT
|
8.7 | pIC50 | 3 | Yes | |
XRYIGRCTVWSVLX
|
8.7 | pIC50 | 3 | Yes | |
ZIZPSSXZSNIUPK
|
8.7 | pIC50 | 3 | Yes | |
ZZIALNLLNHEQPJ
|
8.7 | pIC50 | 8 | Yes | |
BCIVLSCOJWTHHI
|
8.7 | pIC50 | 3 | Yes | |
BTFPBKCBDXRECY
|
8.7 | pIC50 | 7 | Yes | |
IIOQCHDSPPQIPA
|
8.7 | pIC50 | 3 | Yes | |
NICMQGUSJRULBD
|
8.7 | pIC50 | 4 | Yes | |
NRJDKQAGGSKGKV
|
8.7 | pIC50 | 4 | Yes | |
OAVGBZOFDPFGPJ
|
8.7 | pIC50 | 42 | Yes | |
PRSCKUYRGQJIGJ
|
8.7 | pIC50 | 4 | Yes | |
SJIOLEJMBXAEAX
|
8.7 | pIC50 | 4 | Yes | |
UUCSGILLVJJEAR
|
8.7 | pIC50 | 2 | Yes | |
WIPFLAIFCHZLJT
|
8.7 | pIC50 | 4 | Yes | |
DNZYOZKYEXTOPJ
|
8.7 | pIC50 | 16 | Yes | |
GGEKOZPXKBYLNK
|
8.7 | pIC50 | 4 | Yes | |
JZLFYMHIISZQCZ
|
8.7 | pIC50 | 12 | Yes | |
NMXUKCANMSBQDR
|
8.7 | pIC50 | 4 | Yes | |
OXSZPKWHXPJDKU
|
8.7 | pIC50 | 3 | Yes | |
PIEBWUHNLFOEHS
|
8.7 | pIC50 | 2 | Yes | |
QQYOOMZAIWLSOT
|
8.7 | pIC50 | 4 | Yes | |
QTEUJQNPMLXVLL
|
8.7 | IC50 | 16 | — | |
SBOATZBNXFFCER
|
8.7 | pIC50 | 4 | Yes | |
YVWMSUSLLTXXJV
|
8.7 | pIC50 | 4 | Yes | |
ODWSOTDOGQCHBR
|
8.7 | pIC50 | 3 | Yes | |
UKHFPVCOXBJPIN
|
8.7 | IC50 | 17 | — | |
VAARYSWULJUGST
|
8.7 | pIC50 | 119 | Yes | |
AOWCVRXIHIHAPN
|
8.6 | pIC50 | 4 | Yes | |
AUZLISXBMGKYGA
|
8.6 | pIC50 | 4 | Yes | |
CMLISELCGZYWIN
|
8.6 | pIC50 | 4 | Yes | |
FOAPLJPPCBMVSP
|
8.6 | pIC50 | 4 | Yes | |
GMDCWQKESXVLDQ
|
8.6 | pIC50 | 5 | Yes | |
HKOBHPSQGCLOAD
|
8.6 | pIC50 | 4 | Yes | |
HSQPVXYXQYREJB
|
8.6 | pIC50 | 2 | Yes | |
IVJIWGTXXHDRCU
|
8.6 | pIC50 | 4 | Yes | |
OGCUOHKSMKRIOU
|
8.6 | pIC50 | 4 | Yes | |
TXYRLWYXGWLWIJ
|
8.6 | pIC50 | 4 | Yes | |
UDUPSRWUDACGIS
|
8.6 | pIC50 | 13 | Yes | |
UXVJUMKPIQCRPX
|
8.6 | pIC50 | 4 | Yes | |
VIDLZOFQQMUWMT
|
8.6 | pIC50 | 4 | Yes |