Target Details
| UniProt AC | P18505 |
|---|---|
| Gene Symbol | GABRB1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 5,316
- Clinical molecules 4981
- Avg pChEMBL 7.5
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (5,316)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGIBDQRYOFBMTC
|
12.0 | pIC50 | 6 | Yes | |
TXUZVZSFRXZGTL
|
10.8 | pIC50 | 7 | Yes | |
DUYNJNWVGIWJRI
|
10.8 | pIC50 | 4 | Yes | |
OEKMGABCSLYWOP
|
10.8 | pIC50 | 4 | Yes | |
RGLYKWWBQGJZGM
|
10.7 | pIC50 | 8 | Yes | |
DUYNJNWVGIWJRI
|
10.6 | pIC50 | 4 | Yes | |
QCTHZNDHZKAUOH
|
10.3 | pIC50 | 4 | Yes | |
SMYDPKRFVHAWET
|
10.2 | pIC50 | 4 | Yes | |
IQWWKHVNEDNTHC
|
10.2 | pIC50 | 4 | Yes | |
FBYRIOLLVVNZKA
|
10.0 | pIC50 | 2 | Yes | |
GXESHMAMLJKROZ
|
10.0 | pIC50 | 4 | Yes | |
CHSQDJYRTBPAPX
|
9.9 | pIC50 | 4 | Yes | |
NGADMKRMBVYAPF
|
9.8 | pIC50 | 2 | Yes | |
DTGDVCGLMWPOPE
|
9.8 | pIC50 | 4 | Yes | |
MUSZSITXXJNLPD
|
9.8 | pIC50 | 2 | Yes | |
MZFKWSFOAVBLQM
|
9.8 | IC50 | 16 | — | |
ZPECPOOQJUIDLY
|
9.8 | pIC50 | 4 | Yes | |
XIESSJVMWNJCGZ
|
9.8 | pIC50 | 4 | Yes | |
IAVUPMFITXYVAF
|
9.7 | pIC50 | 17 | Yes | |
MEFAURHMHWBYCD
|
9.7 | pIC50 | 4 | Yes | |
GZUITABIAKMVPG
|
9.7 | pIC50 | 22 | Yes | |
HJEXWDTYGATKLK
|
9.7 | pIC50 | 3 | Yes | |
KHBWKBINDOFBGN
|
9.7 | pIC50 | 7 | Yes | |
NHMZOHFSSLVUJN
|
9.7 | pIC50 | 4 | Yes | |
QWKKYJLAUWFPDB
|
9.7 | pIC50 | 13 | Yes | |
SSQLMQBZAPRIRS
|
9.7 | pIC50 | 4 | Yes | |
UOZGUWHPVZIRDP
|
9.7 | pIC50 | 4 | Yes | |
UQVQBJWQKAPUBT
|
9.7 | pIC50 | 4 | Yes | |
VEBGFZDIXSWIAZ
|
9.7 | pIC50 | 4 | Yes | |
WFPXOWCKXUEKCA
|
9.7 | IC50 | 16 | — | |
YPJXERWSOZSIOO
|
9.7 | pIC50 | 4 | Yes | |
FAZWUAVXVGSQEM
|
9.7 | pIC50 | 4 | Yes | |
VWUXBMIQPBEWFH
|
9.7 | pIC50 | 8 | Yes | |
JBFBGJWUIICAFO
|
9.7 | pIC50 | 4 | Yes | |
LHZOGDYGAMOXIH
|
9.6 | pIC50 | 2 | Yes | |
OGRZJPRETQPCLH
|
9.6 | pIC50 | 3 | Yes | |
VWBZVMZFOBZQTD
|
9.6 | pIC50 | 2 | Yes | |
KVKWRJDNIJTMGN
|
9.6 | IC50 | 16 | — | |
KNKMMFVVMHOSMW
|
9.6 | pIC50 | 4 | Yes | |
STDKUMSDTHTDBM
|
9.6 | pIC50 | 4 | Yes | |
WQYYZNGOTUCWQX
|
9.6 | Ki | 5 | — | |
XSIHFOOFJWBVHK
|
9.6 | pIC50 | 4 | Yes | |
RHQLNMNKTIOREN
|
9.6 | pIC50 | 4 | Yes | |
WDHIYKZHKBKYCY
|
9.6 | pIC50 | 4 | Yes | |
RCVOOQFPOXBKPQ
|
9.5 | pIC50 | 4 | Yes | |
DUTQYXPXGOBWIZ
|
9.5 | pIC50 | 4 | Yes | |
FVMJBLJQHQYJPU
|
9.5 | pIC50 | 3 | Yes | |
HCXSUZWCTCKJCT
|
9.5 | pIC50 | 4 | Yes | |
HHHDJHHNEURCNV
|
9.5 | pIC50 | 13 | Yes | |
HOLJYLOVIHBQHO
|
9.5 | pIC50 | 12 | Yes |