Target Details
| UniProt AC | P18433 |
|---|---|
| Gene Symbol | PTPRA |
| Protein Name | Receptor-type tyrosine-protein phosphatase alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 6.61
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKOYIUYWMSVYKN
|
7.6 | Ki | 3 | — | |
IQYFRRLUZSIOTL
|
7.2 | Ki | 3 | — | |
HMUGMCSGKHKDGY
|
7.1 | Ki | 2 | — | |
CZHXFEWAZCRHGB
|
6.9 | Ki | 2 | — | |
FSRCMOQVSVRBJH
|
6.8 | Ki | 2 | — | |
QOPBMVGFMRLORF
|
6.6 | Ki | 2 | — | |
JYWLVKREVMTEJA
|
6.4 | Ki | 3 | — | |
JTJBRKLISQICDU
|
6.3 | Ki | 3 | — | |
MATPDXBXMLXXPY
|
6.1 | Ki | 2 | — | |
MOSWXYTWKAJKPK
|
6.1 | Ki | 2 | — | |
NXIFQDCSZVPVLT
|
6.0 | Ki | 2 | — | |
SUACYXRSGYYBGT
|
6.0 | IC50 | 2 | — |