Target Details
UniProt ACP18089
Gene SymbolADRA2B
Protein NameAlpha-2B adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 566
  • Clinical molecules 47
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (566)
InChIKey pChEMBL Type Targets Clinical
SIYLLGKDQZGJHK 6.4 IC50 13
BNXNWRSVYQHTOH 6.3 Ki 12
BVWLLEDYRCHASI 6.3 Ki 3
GPVHKTUBAXLWKX 6.3 Ki 3
GZKLJWGUPQBVJQ 6.3 Ki 24 Yes
IAIZHDGEGFGNMO 6.3 Ki 3
SVJMLYUFVDMUHP 6.3 Ki 26
BTDBEHJEPKRBOL 6.3 Kd 3
CKLWXPRLRVVKLX 6.3 Ki 3
LNEPOXFFQSENCJ 6.3 Ki 33 Yes
LOGUSYSMQQMCJG 6.3 Ki 3
YVSAGYHRJDVYHG 6.3 Ki 3
AHCOOGMIZVMEKD 6.3 Ki 6
FBCSWIXKXHSYBN 6.3 Ki 18
MJJALKDDGIKVBE 6.3 IC50 30 Yes
OGOLMGZJNRNULQ 6.3 Ki 4
OTXMFMMMNBKXQC 6.3 Ki 4
ZMDCNVSZNFXVKI 6.3 Ki 3
CXQUOFVDYCOSEZ 6.3 Ki 10 Yes
QQBCCUCHUBUQEQ 6.3 Ki 6
UREJDUPKGMFJRU 6.3 Ki 17
XWUSTWDFKOHGNW 6.3 Ki 6
YQTAOHSPORUWMC 6.3 Ki 5
ARFIQGOUMZSQLT 6.3 IC50 3
DCSUBABJRXZOMT 6.3 Ki 24
JXZZEXZZKAWDSP 6.3 Ki 5
LROGAFKJTOPROQ 6.3 Ki 3
RFWZESUMWJKKRN 6.3 Ki 5
RLMGUPUESXPDFJ 6.3 Ki 5 Yes
YAORIDZYZDUZCM 6.3 Ki 5
CKZOGIXOGHVXNW 6.3 Ki 3
MDMPKBVNLDREMU 6.3 Ki 3
NFKNRFTZWQGNTI 6.3 Ki 4
OITKDPXYSUWTOJ 6.3 Ki 3
KJTFLBJQHBFQAF 6.3 Ki 5
QVTLLPCYIGXVLX 6.3 Ki 3
XBWFPEVESQMIBM 6.3 Ki 3
IOIMNYMJVKCZNT 6.2 Ki 3
JFIOVJDNOJYLKP 6.2 Ki 12 Yes
KLPWJLBORRMFGK 6.2 Ki 8
MNMDMCKHXVHLAW 6.2 Ki 3
QYCJTZDZQXSXSC 6.2 Ki 3
BTYBILKFYYEYRM 6.2 Ki 6
GJSIQLZDGMIVKC 6.2 Ki 2
HXJKWPGVENNMCC 6.2 Ki 5
ISZKYBBFFMQCLL 6.2 Ki 6
KFMXRGXNQZECTP 6.2 Ki 9
XTIBNNVUTCNMBE 6.2 IC50 3
YSPOTMDNGADFCJ 6.2 Ki 6
MGJOAQODMQCCGV 6.2 Ki 3
2D structure