Target Details
UniProt ACP18089
Gene SymbolADRA2B
Protein NameAlpha-2B adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 566
  • Clinical molecules 47
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (566)
InChIKey pChEMBL Type Targets Clinical
NREVCQNJBZJFTB 6.8 Ki 2
OGJGQVFWEPNYSB 6.8 Ki 11
FKKPXTRMLVLGJG 6.8 Ki 7 Yes
XMXHEBAFVSFQEX 6.8 Ki 17
ZEWQUBUPAILYHI 6.8 Ki 21
CDQCFGYTKJPHKT 6.8 Ki 3
CWWOITPDZXNTSJ 6.8 Ki 3
MDFFTELFADBPIZ 6.8 Ki 4
MPCNSEQVVHOHGO 6.8 Ki 3
INJOMKTZOLKMBF 6.8 IC50 6
XRJGWSMTLAFHBN 6.8 Ki 21
SQZSBSSOJVUBRM 6.8 Ki 3
AEDGYKKUCHJGJO 6.8 Ki 3
HDOZVRUNCMBHFH 6.8 Ki 26 Yes
VSEIJSADDBOANG 6.8 Ki 3
XBWUQSHGQYCHAA 6.8 Ki 3
JWAAXMLRAVOKBQ 6.7 Ki 3
UKOCGOXTVCIACM 6.7 Ki 13
YJDXDLLDGRBMIT 6.7 Ki 3
BTDBEHJEPKRBOL 6.7 Kd 3
RIMQFOFQYZBTDB 6.7 Ki 3
VRBKIVRKKCLPHA 6.7 Ki 22
WIQCERUTOBWUOL 6.7 Ki 3
ZKIAIYBUSXZPLP 6.7 Ki 29
MBPZQLMDDBIIGZ 6.7 IC50 3
QSLMDECMDJKHMQ 6.7 IC50 20
WVVSZNPYNCNODU 6.7 IC50 8
FPCCSQOGAWCVBH 6.7 Ki 16
GUTLHNWEBBMLCC 6.7 Ki 4
VUBWIAJSRQTELD 6.7 Kd 3
YVENIGOVHPMTDH 6.7 Ki 23
DHSSDEDRBUKTQY 6.7 Ki 6
JCCIEQKRVYXDHE 6.7 Ki 4
MWOOWQMUFWOYRV 6.7 Ki 4
PHWBOXQYWZNQIN 6.7 IC50 6
HAEPGZUGYMHCJE 6.7 Kd 3
KVWDHTXUZHCGIO 6.7 Ki 32 Yes
UXABARREKCJULM 6.7 IC50 3
LJLYHROZJUTILK 6.7 Ki 3
TYBWDPQQOPIKEB 6.7 Ki 3
ALTKABGEMCJWJH 6.7 Ki 15
FFCFXJXBXUOFIU 6.7 Ki 4
KADUIVAIJUZKJS 6.7 Ki 6
RONZAEMNMFQXRA 6.7 IC50 9 Yes
GWQQAPMSNKFDFF 6.6 Ki 3
JWPAYBAIIARWMG 6.6 Ki 19
MBUVEWMHONZEQD 6.6 Ki 17 Yes
YTBMWHRBVZXATF 6.6 Ki 3
GYQWYEJFOYQDMB 6.6 Ki 3
MHNSOBBJZCWUGS 6.6 Ki 17
2D structure