Target Details
UniProt ACP18089
Gene SymbolADRA2B
Protein NameAlpha-2B adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 566
  • Clinical molecules 47
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (566)
InChIKey pChEMBL Type Targets Clinical
LJRFIWIVFLBBPS 7.4 Kd 6
JFKKLIJAJCMWRM 7.4 Ki 8
NUMRIDYCRYHYHT 7.4 Ki 3
WBGSURPVIDDDHF 7.4 Ki 3
YEPGXJIOCYXZAI 7.4 Ki 3
WYFPZXUWZCKNMJ 7.4 Ki 3
WZOMJNATDSYQHS 7.4 Ki 3
CQXADFVORZEARL 7.4 Ki 4
YYTGOWDNUUXBGS 7.4 Ki 5
GIJXKZJWITVLHI 7.4 IC50 16
RWDJYHMGMOOTRK 7.3 Ki 3
BYPMJBXPNZMNQD 7.3 Ki 18
PXPKAXRRJYZLDN 7.3 Ki 3
CJFOJUCLYBZSAN 7.3 Ki 3
OABROWXKGQFLDH 7.3 Ki 3
ODQWQRRAPPTVAG 7.3 IC50 20 Yes
PLDUPXSUYLZYBN 7.3 Ki 22
QOYHHIBFXOOADH 7.3 Ki 16
CETMNKCDAHCKRC 7.3 Ki 3
XHLHZPFSBCZVEA 7.3 Ki 3
QZUDBNBUXVUHMW 7.3 Ki 39 Yes
RATZLMXRALDSJW 7.3 Ki 4
IPSCUIDJZTXJJO 7.3 Ki 3
QNWVOPOAKHMIHV 7.3 Ki 3
UZRVBSAZMGMVTH 7.3 Ki 3
OHRDRIOXKSBXGK 7.2 Kd 6
SXCVVYUSUGUSMW 7.2 Ki 14
ZFDWAPWETDMDSZ 7.2 Ki 3
AJWTXSLKVJNYAB 7.2 Ki 3
IQDINXFLUAYBCC 7.2 Ki 3
MOJPEWKNYNURQQ 7.2 Ki 2
CVKQUGPVDVFRAT 7.2 Ki 4
OGHNVEJMJSYVRP 7.2 IC50 18
NTSMKZTVZAMTDB 7.2 Ki 8
FASDKYOPVNHBLU 7.2 Ki 9
GDLIGKIOYRNHDA 7.2 IC50 24 Yes
KSMAGQUYOIHWFS 7.2 Ki 4
MRSWPVWIMKYKPA 7.2 Ki 3
VDDKWLCHDOJXJM 7.2 Ki 3
VJQWCCBDYLTRPZ 7.2 Ki 3
CQXADFVORZEARL 7.2 Ki 4
IYLGKCYRBQLWIN 7.1 Ki 3
KORNTPPJEAJQIU 7.1 Ki 17
ZTBWRKAKTUWRSC 7.1 Ki 3
DFZXRUBHUWNVAN 7.1 Ki 3
WPNJAUFVNXKLIM 7.1 Ki 4
YMYZKGIHGMHZDL 7.1 Ki 5
VCKUSRYTPJJLNI 7.1 Ki 6
ZFYOCHWWKWULRT 7.1 Ki 3
GPPWMDRIVISCNC 7.1 Ki 3
2D structure