Target Details
UniProt ACP18089
Gene SymbolADRA2B
Protein NameAlpha-2B adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 566
  • Clinical molecules 47
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (566)
InChIKey pChEMBL Type Targets Clinical
LQKQCQKZRUYZOI 8.6 Ki 4
FGTWZUQEDNXLLZ 8.6 IC50 4
GICQFAWDMCTLDM 8.6 IC50 4
XCGSFFUVFURLIX 8.6 IC50 17
ZYXHQIPQIKTEDI 8.6 IC50 4
FYLKUCQQWYKEOG 8.6 Ki 4
CARQBUHFBAORAB 8.5 Ki 3
WKXSXFYQPCWZOS 8.5 Ki 6
UCNOTTVNPRSTFW 8.4 Ki 8 Yes
LUZRJRNZXALNLM 8.4 Ki 20
WGLYZLZIIJTKAG 8.4 IC50 4
HNRZWHPQDGUUSO 8.4 IC50 4
IEJXVRYNEISIKR 8.3 Ki 6
HGEYJZMMUGWEOT 8.3 Ki 17
HSSBMQXDKGERBI 8.3 Ki 4
FAFGGANFZMERDR 8.3 Ki 3
VKABNRMTNPWHBD 8.3 Ki 3
DEQITUUQPICUMR 8.3 IC50 13
WDSZUSABLKNHCZ 8.2 Ki 3
WDSZUSABLKNHCZ 8.2 Ki 4
PMXMIIMHBWHSKN 8.2 Ki 19
IAHLXXAKFXOKST 8.2 Ki 3
IXRPDYSTGHYEBR 8.2 Ki 4
HAEPGZUGYMHCJE 8.2 Kd 3
JWYUBODPEUBFLH 8.2 Ki 11
KXSUAWAUCNFBQJ 8.2 Ki 3
MGQIWQQQIZXANT 8.2 Ki 3
WIKYUJGCLQQFNW 8.2 IC50 23 Yes
HAEPGZUGYMHCJE 8.2 Kd 3
ZMOPTLXEYOVARP 8.2 Ki 14 Yes
GUYATMODRNZQDL 8.1 Ki 6
NEQHKSNFFVEGHN 8.1 Ki 6
OSEADGVOKYGIER 8.1 Ki 3
JWYUBODPEUBFLH 8.1 Ki 3
WLQWOUULTDRZTQ 8.1 Ki 3
SJTUPIJPFNBFHK 8.1 Ki 3
MRBDMNSDAVCSSF 8.1 Ki 10
PGOVKWAJCVAZNG 8.1 Ki 3
UEZSUAXJWCMWEK 8.1 Kd 3
XXQLSAWUSXSJTK 8.1 Ki 6
IRIQHWJBJQBIEB 8.1 Ki 3
YWALOGYVALOLTL 8.1 Ki 3
ASHFKBMVCDTQQO 8.0 Ki 4
DAIRUBYTBODIKT 8.0 Ki 3
XYLJNLCSTIOKRM 8.0 Ki 4
KKLYBLFGKSXYJZ 8.0 IC50 4
MHPMXTGKTXJIDI 8.0 Ki 6
JMXRRARDLWHYJN 8.0 IC50 4
CUHVIMMYOGQXCV 7.9 Ki 6
FJABWASNVHOPLU 7.9 Ki 3
2D structure