Target Details
UniProt ACP18089
Gene SymbolADRA2B
Protein NameAlpha-2B adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 566
  • Clinical molecules 47
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (566)
InChIKey pChEMBL Type Targets Clinical
VWIAFKHHBIYXKV 10.8 IC50 3
MWIKFEVHBBAXIQ 10.8 IC50 3
SWDBYQPERYMOIS 10.5 IC50 3
FIERHAFMRVRMDV 9.9 Ki 4
YRDASYXEOGTMQU 9.9 IC50 3
BKRGVLQUQGGVSM 9.9 Ki 18
ARHWJJBPLJIHQP 9.7 Ki 4
JKDBLHWERQWYKF 9.7 Kd 3
JKDBLHWERQWYKF 9.7 Kd 3
WYFCRYMMLDTJAM 9.7 Ki 4
BJNQZYVNKAVYSF 9.6 Ki 6
GKDBTHSYQZTDAJ 9.6 IC50 13
XGXYGEYUGTVZAR 9.6 Ki 6
WCIDBLYFACGZGW 9.6 IC50 3
PRXCUMHAHRIDJF 9.5 Ki 4
JOAHPSVPXZTVEP 9.3 Ki 19
VSWBSWWIRNCQIJ 9.3 Ki 23
BKRGVLQUQGGVSM 9.3 Ki 26 Yes
WVDIRTLHBANRPM 9.2 IC50 3
VDSXZDLUEYFJGH 9.2 Ki 4
HOKCXDCTKLQEJE 9.1 Ki 3
JRDUBBHIPPPSLP 9.1 Ki 3
DLWKVBPPVYZEML 9.0 Ki 4
GZFYZEHGCPEJAC 9.0 IC50 4
ZFZUYTCCHMWWTD 9.0 Ki 9
JWXMKFUDAOLJCY 8.9 Ki 4
OSJJYEUEJRVVOD 8.9 IC50 17 Yes
OSJZLDGTMVBIRV 8.9 Ki 6
AKZOIEBLVQLVTR 8.9 IC50 3
XSOUHEXVEOQRKJ 8.9 Ki 14
QZUXRMOPAGPTIY 8.9 Ki 4
BRKWIMBSEICBCU 8.9 IC50 4
FPQNWBCHCMEAKI 8.8 IC50 4
HSRPTPAPMBHRRJ 8.8 IC50 5
PUJAGVRPJZNJPF 8.8 IC50 4
AKBJKOBHDJQWMB 8.8 Ki 4
HQGWKNGAKBPTBX 8.8 Ki 3
LWSVCEUUPRLOSZ 8.8 Ki 3
JVGBTTIJPBFLTE 8.8 Ki 16
FLAHEXULHVZYHT 8.8 Ki 3
UDURNHDRCUMUOV 8.8 IC50 4
RVRPAIWBGBVSKB 8.8 Ki 3
JRMVEEDZCPVFFK 8.7 IC50 3
HPNSJGWCFMHOJX 8.7 IC50 4
MUUSOYWTPTTZII 8.7 Ki 3
UJYGDMFEEDNVBF 8.7 IC50 12
FXNNPMSELIMMHU 8.7 Ki 4
RTXNZOCMRSFEID 8.7 IC50 4
WLWNODXEXGTHDO 8.7 IC50 4
HSWPZIDYAHLZDD 8.7 Ki 3
2D structure