Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJWWIXPWIBPUOV
|
6.7 | IC50 | 2 | — | |
FRXCQHJSACJLPG
|
6.7 | IC50 | 4 | — | |
AFBPNQXAQLFHKE
|
6.7 | IC50 | 2 | — | |
FLABGAZLPSNUBD
|
6.7 | IC50 | 3 | — | |
PRUCOWVKLZWPSA
|
6.7 | IC50 | 3 | — | |
RNDRXNFFHJEMIZ
|
6.7 | IC50 | 3 | — | |
NZSZQHHTXGSVGH
|
6.7 | IC50 | 5 | — | |
PSZYZEZKPQGGPA
|
6.6 | IC50 | 6 | — | |
PJJWGMOYKFOUPO
|
6.6 | IC50 | 5 | — | |
WEYZFBLZVFBVAR
|
6.6 | IC50 | 5 | — | |
YJXODXFHFQYURN
|
6.6 | IC50 | 4 | — | |
XRIHUZYLIIDSBZ
|
6.6 | IC50 | 5 | — | |
QYOKHKZTOCBBQY
|
6.6 | IC50 | 5 | — | |
BSTGKAROMCRBDW
|
6.6 | IC50 | 3 | — | |
FVIAXINNEOEZCZ
|
6.5 | IC50 | 6 | — | |
WBNIBVOJNZUYKZ
|
6.5 | IC50 | 3 | — | |
KIOBNTPONYOMJE
|
6.5 | IC50 | 4 | — | |
NVHPXYIRNJFKTE
|
6.5 | IC50 | 6 | — | |
APIKKGOIHMESQS
|
6.5 | IC50 | 5 | — | |
PCEMPIMHMWVATP
|
6.5 | IC50 | 5 | — | |
YJLXHQJWGPXYIB
|
6.5 | IC50 | 5 | — | |
OURYZIAAXSSBIO
|
6.5 | IC50 | 5 | — | |
TVAOKDIBRVLPTB
|
6.5 | IC50 | 4 | — | |
GNNSUMADLWATJP
|
6.5 | IC50 | 5 | — | |
ZXXBSSKQLMNDPX
|
6.5 | IC50 | 4 | — | |
GWYITMXKBHRSJF
|
6.4 | IC50 | 5 | — | |
KGVFBFPXRYIQHI
|
6.4 | IC50 | 5 | — | |
PBBRGHSUTCYOJM
|
6.4 | IC50 | 5 | — | |
VHSMIAWMPAKQCQ
|
6.4 | IC50 | 2 | — | |
VNLGSUKLIVHSOW
|
6.4 | IC50 | 3 | — | |
XXGGOJFTDMPZAG
|
6.4 | IC50 | 3 | — | |
SIVAZRUSFYJFGM
|
6.4 | IC50 | 3 | — | |
AQAUYHNXROATLO
|
6.3 | IC50 | 4 | — | |
ADHOGOCWYMYMBV
|
6.3 | IC50 | 5 | — | |
BXOSGYRJKCYDLH
|
6.3 | IC50 | 5 | — | |
FFGKQSKYPTZWNF
|
6.3 | IC50 | 2 | — | |
OILZZIXLONGEMV
|
6.3 | IC50 | 3 | — | |
YRBHDRXOHRYTHS
|
6.3 | IC50 | 2 | — | |
YUBVJZGWIJZEGM
|
6.3 | IC50 | 5 | — | |
RNDRXNFFHJEMIZ
|
6.3 | IC50 | 3 | — | |
DPVUQQDISRAKFA
|
6.3 | IC50 | 2 | — | |
DPVUQQDISRAKFA
|
6.3 | IC50 | 3 | — | |
UZVROHMMUDQAOJ
|
6.3 | IC50 | 5 | — | |
ANHVXOMSUJRVTQ
|
6.2 | IC50 | 5 | — | |
FNDMWTXEBTVCPM
|
6.2 | IC50 | 4 | — | |
LOXDBHIFADBELN
|
6.2 | IC50 | 7 | — | |
SVFSXWWDSXBQLC
|
6.2 | IC50 | 2 | — | |
SVFSXWWDSXBQLC
|
6.2 | IC50 | 3 | — | |
CVFCIUNYJXEWIG
|
6.1 | IC50 | 5 | — | |
GFTVRPWYQDITLC
|
6.0 | IC50 | 5 | — |