Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UYLKMCAJPYTSGJ
|
7.4 | IC50 | 4 | — | |
UYLKMCAJPYTSGJ
|
7.4 | IC50 | 3 | — | |
LXRNNOYGXXYOIM
|
7.4 | IC50 | 5 | — | |
FPMATBDSZPMWSV
|
7.4 | IC50 | 2 | — | |
VYIBTYZRYKIMKX
|
7.4 | IC50 | 3 | — | |
FOIPXCGYGBYXAS
|
7.3 | IC50 | 5 | — | |
OUYHRBRXZUOZRC
|
7.3 | IC50 | 4 | — | |
NNZBVLNVFSQLGP
|
7.3 | IC50 | 3 | — | |
HCUONOGSJKCNGD
|
7.3 | IC50 | 5 | — | |
SGFBXTDHLSCRBX
|
7.3 | IC50 | 4 | — | |
BSLQJJPIELRITP
|
7.3 | IC50 | 7 | — | |
LEBUVLVDRAIZDW
|
7.3 | IC50 | 5 | — | |
NIVBRIPUAQCFIE
|
7.3 | IC50 | 6 | — | |
NTOCWOHJTCYCPV
|
7.3 | IC50 | 4 | — | |
OISGDSNHYNQFQH
|
7.3 | IC50 | 2 | — | |
RLSMGFIEFQMTPO
|
7.3 | IC50 | 5 | — | |
HAWHNGUKUZPYEE
|
7.2 | IC50 | 4 | — | |
JUCATPBOBDBSCE
|
7.2 | IC50 | 4 | — | |
KALOYQBAVHVFJS
|
7.2 | IC50 | 5 | — | |
KEXLTXLRSNUTNU
|
7.2 | IC50 | 2 | — | |
SBUMUHUTBKYAPS
|
7.2 | IC50 | 4 | — | |
YYYKEWBUGLVEQB
|
7.2 | IC50 | 3 | — | |
YDHAGPCZRFQPOI
|
7.2 | IC50 | 6 | — | |
CJMISCRXEFTMEV
|
7.2 | IC50 | 6 | — | |
HCCLOZIGOHDHLA
|
7.2 | IC50 | 5 | — | |
IUQPRHFUTQDNBT
|
7.2 | IC50 | 5 | — | |
KRLSGXAAVBXUNS
|
7.2 | IC50 | 5 | — | |
ROFCWWUBJHHVGZ
|
7.2 | IC50 | 6 | — | |
UNCCZOQBJPENMD
|
7.2 | IC50 | 5 | — | |
UQVXTUIZRQSMCZ
|
7.2 | IC50 | 5 | — | |
NMFMDJLYTCYODM
|
7.2 | IC50 | 5 | — | |
HISPCWBBRIZTIO
|
7.2 | IC50 | 4 | — | |
AXIJMLLLPVCDAY
|
7.2 | IC50 | 2 | — | |
NUPIGKKRXBENIY
|
7.2 | IC50 | 2 | — | |
CGVRSJVSZRAVEI
|
7.1 | IC50 | 4 | — | |
UVOUWFPJSKSTMI
|
7.1 | IC50 | 2 | — | |
WEXQBLSMARBRMG
|
7.1 | IC50 | 6 | — | |
HSQHKAOCNXUSQN
|
7.1 | IC50 | 3 | — | |
NWNHXYNBSWSDHY
|
7.1 | IC50 | 2 | — | |
POHCCPZJODTAKF
|
7.1 | IC50 | 3 | — | |
AFBPNQXAQLFHKE
|
7.1 | IC50 | 2 | — | |
DCQCDEPHHWZADO
|
7.1 | IC50 | 4 | — | |
FLABGAZLPSNUBD
|
7.1 | IC50 | 3 | — | |
HKDUWRRLEDNORE
|
7.1 | IC50 | 6 | — | |
JWYJAXVOVLDVAL
|
7.1 | IC50 | 6 | — | |
RLABYQGJZRFBJA
|
7.1 | IC50 | 3 | — | |
SBBQXRAHGMRHHD
|
7.1 | IC50 | 5 | — | |
YSBLTULPICYNEV
|
7.1 | IC50 | 2 | — | |
YWTMANCVOUNUAR
|
7.1 | IC50 | 4 | — | |
ZTISQJYIMPGHCK
|
7.1 | IC50 | 5 | — |