Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MPXAADAXXFWYMY
|
7.7 | IC50 | 7 | — | |
NIHKLJCATASIRV
|
7.7 | IC50 | 6 | — | |
QGLIEPQLAXSZRG
|
7.7 | IC50 | 3 | — | |
RKBFMHGYXWQNKU
|
7.7 | IC50 | 4 | — | |
RZAGOFCCJINLJO
|
7.7 | IC50 | 6 | — | |
ZHKXSTJFXIMBBI
|
7.7 | IC50 | 6 | — | |
ZILGGGDRKNJYPR
|
7.7 | IC50 | 3 | — | |
ZMXBIIQMSGOIRZ
|
7.7 | IC50 | 7 | — | |
POHCCPZJODTAKF
|
7.7 | IC50 | 3 | — | |
QTQQUVKCPJYESZ
|
7.7 | IC50 | 3 | — | |
CQDWPOURVPAZAM
|
7.6 | IC50 | 5 | — | |
HUEYQBNZGBYJGI
|
7.6 | IC50 | 2 | — | |
LHDRGDKBCVAGOV
|
7.6 | IC50 | 3 | — | |
RLABYQGJZRFBJA
|
7.6 | IC50 | 3 | — | |
YSBLTULPICYNEV
|
7.6 | IC50 | 2 | — | |
DHKPZDWVBJIRBP
|
7.6 | IC50 | 6 | — | |
GHWOXCUYNGDEQZ
|
7.6 | IC50 | 2 | — | |
QRTUGFDKIIABQN
|
7.6 | IC50 | 5 | — | |
RZAGOFCCJINLJO
|
7.6 | IC50 | 6 | — | |
NGJLAUMTWASOIM
|
7.6 | IC50 | 4 | — | |
VYTWTVISEPFYEI
|
7.6 | IC50 | 2 | — | |
BLJRESKVKZWVMU
|
7.6 | IC50 | 5 | — | |
NGJLAUMTWASOIM
|
7.6 | IC50 | 5 | — | |
SLTMEZLQPRTTBL
|
7.6 | IC50 | 3 | — | |
NGLDQEAARWHFFU
|
7.5 | IC50 | 3 | — | |
NGLDQEAARWHFFU
|
7.5 | IC50 | 4 | — | |
PMZAMOSBWUCNBG
|
7.5 | IC50 | 5 | — | |
XLANGJRVQABTFO
|
7.5 | IC50 | 5 | — | |
CFCPTSHVAOVLJR
|
7.5 | IC50 | 3 | — | |
SFCKQTNFUJZSFW
|
7.5 | IC50 | 2 | — | |
RURWNESJHWLUMA
|
7.5 | IC50 | 3 | — | |
XQHLFZJLRICIOE
|
7.5 | IC50 | 6 | — | |
MNMNKSRAIMNXQS
|
7.5 | IC50 | 4 | — | |
DGXVRVIKQDYUDK
|
7.5 | IC50 | 3 | — | |
UMZVBZDHGKJFGQ
|
7.5 | IC50 | 5 | — | |
JNEZPOFKGHMQAC
|
7.4 | IC50 | 3 | — | |
JRIGXBQWNCXPOG
|
7.4 | IC50 | 2 | — | |
RBSUHEPCSZKVSP
|
7.4 | IC50 | 4 | — | |
DPRPMOCPAJEXJM
|
7.4 | IC50 | 4 | — | |
GXNRMXKXTHPZDX
|
7.4 | IC50 | 5 | — | |
AICBXHQRXOXRSL
|
7.4 | IC50 | 3 | — | |
AVGZVNRRKZUYJJ
|
7.4 | IC50 | 6 | — | |
AYRVAWFOHYBCGQ
|
7.4 | IC50 | 4 | — | |
CCHDZAZXCIHJMH
|
7.4 | IC50 | 5 | — | |
HLYAJAMUFRQZFN
|
7.4 | IC50 | 2 | — | |
HUIWUMINMQIJSX
|
7.4 | IC50 | 4 | — | |
JXJGHJUDGYCRBL
|
7.4 | IC50 | 6 | — | |
KRLSGXAAVBXUNS
|
7.4 | IC50 | 5 | — | |
LJRNCZFZZOWSEH
|
7.4 | IC50 | 5 | — | |
RIJYZNGFJGMMPF
|
7.4 | IC50 | 4 | — |