Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTCHSFYIOSVBQO
|
8.1 | IC50 | 5 | — | |
WYVKIJXOPFCHFD
|
8.1 | IC50 | 4 | — | |
RUUXOWOHEJZKAR
|
8.1 | IC50 | 3 | — | |
XJZOWTKPNHFBKX
|
8.1 | IC50 | 2 | — | |
HOWZBTKZCUTFCU
|
8.0 | IC50 | 2 | — | |
HSACVEKFGJAKFH
|
8.0 | IC50 | 3 | — | |
LDHLQPMIUKAPSY
|
8.0 | IC50 | 4 | — | |
LDHLQPMIUKAPSY
|
8.0 | IC50 | 5 | — | |
PQYGSGMXFJNDPV
|
8.0 | IC50 | 3 | — | |
AJDOOWNOWOSWPT
|
8.0 | IC50 | 3 | — | |
CGDCNLRQFMWABO
|
8.0 | IC50 | 3 | — | |
DTNKZZXZAPCYPT
|
8.0 | IC50 | 3 | — | |
IIJWLNNXJHIKND
|
8.0 | IC50 | 3 | — | |
JESHEQMKKYQWKH
|
8.0 | IC50 | 4 | — | |
QEDWYURCTRDSED
|
8.0 | IC50 | 2 | — | |
VFHGPYIYENLDFG
|
8.0 | IC50 | 2 | — | |
YINCHOOHNDSILR
|
8.0 | IC50 | 4 | — | |
IAMUMIBDQILHMZ
|
8.0 | IC50 | 4 | — | |
JJUSNAIQJYMGPK
|
8.0 | IC50 | 3 | — | |
NKIPTRIPXHQDGW
|
8.0 | IC50 | 6 | — | |
VUDQMHAFTAQNOM
|
8.0 | IC50 | 4 | — | |
FCBBWFAJOJDUFL
|
7.9 | IC50 | 2 | — | |
FZBGGWKHCWPGOF
|
7.9 | IC50 | 5 | — | |
HGWMSQIIHVZYGE
|
7.9 | IC50 | 2 | — | |
SRAAZWOKIPPIDS
|
7.9 | IC50 | 6 | — | |
KNVMGBKMZYKHLR
|
7.9 | IC50 | 5 | — | |
KNVMGBKMZYKHLR
|
7.9 | IC50 | 4 | — | |
CFCPTSHVAOVLJR
|
7.9 | IC50 | 3 | — | |
SFCKQTNFUJZSFW
|
7.9 | IC50 | 2 | — | |
KXNBOEKASHEVEY
|
7.8 | IC50 | 2 | — | |
WVGKDHMQHAQBNH
|
7.8 | IC50 | 3 | — | |
NEBGAKBOVCHODI
|
7.8 | IC50 | 3 | — | |
GJIKWVOEJHFSSK
|
7.8 | IC50 | 2 | — | |
AVGHGSKYPBYCGD
|
7.8 | IC50 | 2 | — | |
DRMIWPCMCBXOEN
|
7.8 | IC50 | 6 | — | |
HTVBJLAHDXBYNO
|
7.8 | IC50 | 4 | — | |
VYLBOUQMYNRGBR
|
7.8 | IC50 | 3 | — | |
ZYPBXFINEXHXPV
|
7.8 | IC50 | 4 | — | |
JTOSMCOFPADVGU
|
7.8 | IC50 | 4 | — | |
AJVBWPQQXWRZHQ
|
7.8 | IC50 | 3 | — | |
DKGATRXTJTUOON
|
7.8 | IC50 | 3 | — | |
JRVUMBDCNCWNEP
|
7.8 | IC50 | 3 | — | |
GRLGGJHKWVARHL
|
7.8 | IC50 | 2 | — | |
ZMWIYVLLRRYJEL
|
7.8 | IC50 | 3 | — | |
XKXMEMPIHRKAQX
|
7.7 | IC50 | 5 | — | |
CGSLGBRMSMBNMX
|
7.7 | IC50 | 6 | — | |
GGDGXCWXJDMCHZ
|
7.7 | IC50 | 2 | — | |
HQFQHOPPJBTIBG
|
7.7 | IC50 | 4 | — | |
ITGKMDQIQJNXCY
|
7.7 | IC50 | 3 | — | |
MFVBSMYEXLRRIU
|
7.7 | IC50 | 5 | — |