Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LKLFMSIRSSIJBV
|
8.5 | IC50 | 3 | — | |
WMRZMQGCPFGLAL
|
8.5 | IC50 | 3 | — | |
ZHXUKLZFCFJOMF
|
8.5 | IC50 | 3 | — | |
UMSKKXXFLOGWFX
|
8.5 | IC50 | 4 | — | |
XHPZRPHYLGZLTO
|
8.5 | IC50 | 5 | — | |
FPMATBDSZPMWSV
|
8.5 | IC50 | 2 | — | |
VYIBTYZRYKIMKX
|
8.5 | IC50 | 3 | — | |
SLTMEZLQPRTTBL
|
8.5 | IC50 | 3 | — | |
VYTWTVISEPFYEI
|
8.5 | IC50 | 2 | — | |
QZTBJCSOVXRYCX
|
8.4 | IC50 | 6 | — | |
MXSJSHDIEDILST
|
8.4 | IC50 | 4 | — | |
WMAYUSHYHMSHFY
|
8.4 | IC50 | 6 | — | |
WMAYUSHYHMSHFY
|
8.4 | IC50 | 4 | — | |
FPSTULSQRYACMJ
|
8.4 | IC50 | 3 | — | |
FRVXYRMGRBRKHN
|
8.4 | IC50 | 3 | — | |
HODJKXWPFAAILA
|
8.4 | IC50 | 3 | — | |
KIYRVDKWZZHATH
|
8.4 | IC50 | 3 | — | |
KZYLTZUXEHTOHA
|
8.4 | IC50 | 3 | — | |
XNXMLWZMXHUKQT
|
8.4 | IC50 | 3 | — | |
DPFLAGDMGNKRSD
|
8.4 | IC50 | 4 | — | |
CFCPTSHVAOVLJR
|
8.3 | IC50 | 3 | — | |
LWHWQLNSWIQIMG
|
8.3 | IC50 | 4 | — | |
SFCKQTNFUJZSFW
|
8.3 | IC50 | 2 | — | |
NSLLXYFCBUUZFG
|
8.3 | IC50 | 2 | — | |
XKLDZRHFLSCFBG
|
8.3 | IC50 | 3 | — | |
ZDUUJAZQZQAJEO
|
8.3 | IC50 | 6 | — | |
GDRIGENBEFKVKD
|
8.3 | IC50 | 2 | — | |
YPBCOKBVZUVWMI
|
8.3 | IC50 | 3 | — | |
GARROJJZLJSGSW
|
8.3 | IC50 | 4 | — | |
DZUCEYPUEFNCRE
|
8.3 | IC50 | 3 | — | |
FYRPCZSQQACFLX
|
8.3 | IC50 | 2 | — | |
RCCYAIQAQJPLAH
|
8.2 | IC50 | 3 | — | |
HMKFSFPLRDCCAB
|
8.2 | IC50 | 3 | — | |
IUYOOUVOXKZZKL
|
8.2 | IC50 | 2 | — | |
NLUXMQVEMDAZTJ
|
8.2 | IC50 | 6 | — | |
UEJGLOZXWKIXSB
|
8.2 | IC50 | 2 | — | |
ANXTXJZVXQRTGD
|
8.2 | IC50 | 2 | — | |
QEWKBLVMROGVIO
|
8.2 | IC50 | 6 | — | |
VGFHUCRCHTYYLJ
|
8.2 | IC50 | 3 | — | |
XGMBDTKPGSGTQW
|
8.2 | IC50 | 4 | — | |
SLTMEZLQPRTTBL
|
8.2 | IC50 | 3 | — | |
VYTWTVISEPFYEI
|
8.2 | IC50 | 2 | — | |
ZPRQEMGTRXGZPE
|
8.1 | IC50 | 5 | — | |
ZPRQEMGTRXGZPE
|
8.1 | IC50 | 4 | — | |
IKBMFRHCMUKOBA
|
8.1 | IC50 | 3 | — | |
YHUQGENXDJHDMM
|
8.1 | IC50 | 2 | — | |
AMLYAMJWYAIXIA
|
8.1 | IC50 | 7 | — | |
KGLSWJYMOBWYKH
|
8.1 | IC50 | 2 | — | |
PRUDMEXVXGQSAD
|
8.1 | IC50 | 3 | — | |
YJXODXFHFQYURN
|
8.1 | IC50 | 6 | — |