Target Details
| UniProt AC | P18084 |
|---|---|
| Gene Symbol | ITGB5 |
| Protein Name | Integrin beta-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF18372 (I-EGF_1) PF08725 (Integrin_b_cyt) PF07965 (Integrin_B_tail) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 402
- Clinical molecules 0
- Avg pChEMBL 7.8
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Efferocytosis
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
Active Molecules (402)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OOGFIRRTGDWFJR
|
9.0 | IC50 | 2 | — | |
YYQUWEHEBOMRPH
|
9.0 | IC50 | 3 | — | |
BDFMVIGZRRIXCL
|
9.0 | IC50 | 5 | — | |
WWUJBWRZVJNABY
|
9.0 | IC50 | 3 | — | |
CTCHISHHHJCIRE
|
9.0 | IC50 | 2 | — | |
DIMDWQUSJSWNOO
|
9.0 | IC50 | 5 | — | |
MYSBVCKSODARFZ
|
9.0 | IC50 | 3 | — | |
NXKFHFCWTSGLDC
|
9.0 | IC50 | 4 | — | |
QLBXWVBTUGYSGI
|
9.0 | IC50 | 8 | — | |
WUEJDPFGPRMOTL
|
9.0 | IC50 | 2 | — | |
XWMGBLCMRLASDS
|
9.0 | IC50 | 8 | — | |
YEGQGRLKVPOBBE
|
9.0 | IC50 | 3 | — | |
YVGFDNFQFUSINK
|
9.0 | IC50 | 3 | — | |
JTQSBYUBJLIDAK
|
9.0 | IC50 | 5 | — | |
NIGWPUUZRHIDKJ
|
9.0 | IC50 | 3 | — | |
YGOKSIVHHLSPET
|
8.9 | IC50 | 4 | — | |
YTKGKCKBCJZBIX
|
8.9 | IC50 | 4 | — | |
PZAMXSCMHJPGFV
|
8.8 | IC50 | 3 | — | |
YULSCDVUYRTZCA
|
8.8 | IC50 | 2 | — | |
ZQAQMOMRTYIDJU
|
8.8 | IC50 | 4 | — | |
HIKCELHIZSKMGI
|
8.8 | IC50 | 5 | — | |
PRTDUHZCDXSBIZ
|
8.8 | IC50 | 5 | — | |
KRAZOLZZRSRPAE
|
8.7 | IC50 | 4 | — | |
CTOPQASYIWIPDN
|
8.7 | IC50 | 3 | — | |
CXHCNOMGODVIKB
|
8.7 | IC50 | 7 | — | |
ILKRHUYCJMCBRQ
|
8.7 | IC50 | 8 | — | |
PJAIDMVOZWYNMM
|
8.7 | IC50 | 2 | — | |
SXPOKSLVUGPVBG
|
8.7 | IC50 | 3 | — | |
CTHYLBXDQVAGEJ
|
8.7 | IC50 | 5 | — | |
LJKWPNDKPDWWIA
|
8.7 | IC50 | 4 | — | |
BPBHTITUTUZWBT
|
8.7 | IC50 | 3 | — | |
BZPNVJGCQPADST
|
8.7 | IC50 | 3 | — | |
KAVRMLREXXGTPY
|
8.7 | IC50 | 3 | — | |
MRXQBHPWVQTUKZ
|
8.7 | IC50 | 3 | — | |
TZTYGQORWRHJNU
|
8.7 | IC50 | 2 | — | |
PFYZSIGLKDYGAG
|
8.6 | IC50 | 4 | — | |
DTLIDYQJLOBQPK
|
8.6 | Ki | 3 | — | |
IPLLAQOFEDGGKD
|
8.6 | IC50 | 4 | — | |
UQEWVVUNGPKKKR
|
8.6 | IC50 | 6 | — | |
HODBWQCCKYDYPY
|
8.6 | Ki | 3 | — | |
QXAYHAXWXRCLTG
|
8.6 | IC50 | 4 | — | |
GTSHXMCHGDUGRQ
|
8.5 | IC50 | 4 | — | |
IKALVLPAIVXDBO
|
8.5 | IC50 | 3 | — | |
FCUCMIIVLCLREX
|
8.5 | IC50 | 3 | — | |
MWLPKZBBCRIXMO
|
8.5 | IC50 | 4 | — | |
NQIOUHXNYUMMLV
|
8.5 | IC50 | 4 | — | |
NYIZCWIYRUTEKV
|
8.5 | IC50 | 5 | — | |
ZWPCJINLOLYZBQ
|
8.5 | IC50 | 4 | — | |
AKOSSGWXDCGWFL
|
8.5 | IC50 | 4 | — | |
IFUROQAKNZUNFY
|
8.5 | IC50 | 5 | — |