Target Details
| UniProt AC | P18074 |
|---|---|
| Gene Symbol | ERCC2 |
| Protein Name | General transcription and DNA repair factor IIH helicase subunit XPD |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF06733 (DEAD_2) PF06777 (HBB) PF13307 (Helicase_C_2) |
Summary
- Multi-target molecules 10
- Clinical molecules 3
- Avg pChEMBL 6.81
KEGG Pathways (2)
Associated Diseases (4)
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYCPARAPKDAOEN
|
8.7 | Kd | 73 | — | |
HUXYBQXJVXOMKX
|
8.0 | Kd | 28 | — | |
XKFTZKGMDDZMJI
|
6.9 | Kd | 64 | Yes | |
ZCCPLJOKGAACRT
|
6.8 | Kd | 599 | — | |
WKDACQVEJIVHMZ
|
6.6 | Kd | 46 | — | |
VXBAJLGYBMTJCY
|
6.5 | Kd | 34 | Yes | |
XLSYZSRXVVCHLS
|
6.3 | Kd | 48 | — | |
PIMQWRZWLQKKBJ
|
6.2 | Kd | 36 | — | |
BIIVYFLTOXDAOV
|
6.0 | Kd | 82 | Yes | |
ALKJNCZNEOTEMP
|
6.0 | Kd | 55 | — |