Target Details
| UniProt AC | P18031 |
|---|---|
| Gene Symbol | PTPN1 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 511
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (4)
Active Molecules (511)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WCNVLBVQNHYTKC
|
6.6 | IC50 | 2 | — | |
GRDVSGMHNMMXOE
|
6.5 | IC50 | 2 | — | |
KIICICZHTFLRLA
|
6.5 | IC50 | 2 | — | |
BBDCFVIVCWDRRA
|
6.5 | IC50 | 3 | — | |
OGQLYNGGVJABGS
|
6.5 | IC50 | 2 | — | |
SWVKHXPKNLYPNG
|
6.5 | IC50 | 2 | — | |
ZIBMATWHOAGNTR
|
6.5 | Ki | 2 | — | |
UMIIBUJRMKQTQV
|
6.5 | IC50 | 2 | — | |
ZMFYDQLSNJQHRP
|
6.5 | IC50 | 2 | — | |
CUFAXDWQDQQKFF
|
6.5 | IC50 | 2 | — | |
SAXBGANSQIEGOH
|
6.5 | IC50 | 2 | — | |
QVGRIONJTRDTAM
|
6.5 | IC50 | 2 | — | |
VKNUYCHZQCHJFX
|
6.5 | IC50 | 2 | — | |
LJADUJGFRNMNRC
|
6.5 | IC50 | 2 | — | |
DAZSGUOJKRVDFC
|
6.5 | IC50 | 2 | — | |
FIWRNZMEMMAYAC
|
6.5 | IC50 | 2 | — | |
DZTSPUIXGGCGGS
|
6.5 | IC50 | 2 | — | |
HEZDUVOOOSBRGR
|
6.5 | IC50 | 3 | — | |
PSDPTXNLJQPTIU
|
6.4 | IC50 | 2 | — | |
MOSWXYTWKAJKPK
|
6.4 | Ki | 2 | — | |
UEELPALQXUYKFT
|
6.4 | Ki | 2 | — | |
FONCZICQWCUXEB
|
6.4 | IC50 | 2 | — | |
BBPBZPASZSZJRI
|
6.4 | IC50 | 3 | — | |
BOOMNQMMZXXWGF
|
6.4 | IC50 | 2 | — | |
MFXHVHAGJSIZDY
|
6.4 | IC50 | 2 | — | |
SXLQVLBGTXXABW
|
6.4 | IC50 | 2 | — | |
WIMBRSZNUZJCNR
|
6.4 | IC50 | 2 | — | |
CQHDXEWKDCKMHF
|
6.4 | IC50 | 6 | — | |
IPYSLWNCHIOLRH
|
6.4 | IC50 | 2 | — | |
MPSINWMATOYLCR
|
6.4 | IC50 | 2 | — | |
RQLOUXBWHZRSNQ
|
6.4 | IC50 | 2 | — | |
LCYZNUOBTSKXLT
|
6.4 | IC50 | 2 | — | |
PKLOTZYRQCNNNX
|
6.4 | Ki | 2 | — | |
ULVYQKPUAYJYAI
|
6.4 | IC50 | 2 | — | |
FSNNWMONNMKYTQ
|
6.4 | Ki | 2 | — | |
IBIICFQQAQDOQU
|
6.4 | IC50 | 3 | — | |
SIYOCNTTXYFSHJ
|
6.4 | IC50 | 2 | — | |
JXENTZRLDBYGPD
|
6.3 | IC50 | 2 | — | |
OQIPKIWETZMTHT
|
6.3 | IC50 | 2 | — | |
ZWNRYIDJCJHYOQ
|
6.3 | IC50 | 2 | — | |
GEZHEQNLKAOMCA
|
6.3 | Ki | 6 | — | |
XRNNZLZAOGRJIB
|
6.3 | IC50 | 2 | — | |
ADWUPJWQDFWASY
|
6.3 | IC50 | 2 | — | |
NYXUMJHUNMSZOC
|
6.3 | IC50 | 2 | — | |
VDEMVVHUPJWQFD
|
6.3 | IC50 | 2 | — | |
VIIXHWYAUWYXPH
|
6.3 | IC50 | 2 | — | |
GKLPVCJRSVXISG
|
6.3 | Ki | 2 | — | |
GRUUQSKAGOPWSG
|
6.3 | IC50 | 2 | — | |
IKQRBVJYSDCFNA
|
6.3 | IC50 | 2 | — | |
NNLBBBPQOLHKLK
|
6.3 | IC50 | 2 | — |