Target Details
| UniProt AC | P18031 |
|---|---|
| Gene Symbol | PTPN1 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 511
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (4)
Active Molecules (511)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FSRCMOQVSVRBJH
|
6.8 | Ki | 2 | — | |
FSRCMOQVSVRBJH
|
6.8 | Ki | 2 | — | |
NZHOJYVDRHNLLO
|
6.8 | Ki | 2 | — | |
OACZRTSAVJISLU
|
6.8 | IC50 | 2 | — | |
CXIBSEYTPRXOHP
|
6.8 | IC50 | 2 | — | |
DIGCHRPBTQFUGF
|
6.8 | IC50 | 2 | — | |
RKSWLQKLKPOCSU
|
6.8 | IC50 | 2 | — | |
MZJXRTPTOYLFDN
|
6.8 | IC50 | 2 | — | |
SIUKGJQBSLZIDB
|
6.8 | IC50 | 3 | — | |
IRTOFMLHAJDDRZ
|
6.7 | IC50 | 2 | — | |
KHMNVQHMQBBZIT
|
6.7 | IC50 | 2 | — | |
WGCMBTDMQOGRIE
|
6.7 | IC50 | 2 | — | |
XAXRETYEKMHBIX
|
6.7 | IC50 | 2 | — | |
LVGFRMIIXODOEQ
|
6.7 | IC50 | 4 | — | |
UILYPHAKDBTKQV
|
6.7 | IC50 | 2 | — | |
XJPMAFHARDVTJH
|
6.7 | IC50 | 2 | — | |
BCWHINKEOIUUJT
|
6.7 | IC50 | 3 | — | |
SYBFWGDOOCHMMZ
|
6.7 | IC50 | 2 | — | |
APPXYONGBIXGRO
|
6.7 | Ki | 2 | — | |
FHNSBIYBHXTXGH
|
6.7 | IC50 | 2 | — | |
HTUSEAHGOKFFRF
|
6.7 | Ki | 2 | — | |
ZHOJVBCBTIUSRX
|
6.7 | IC50 | 2 | — | |
SFPAQPMKUYAZGZ
|
6.7 | IC50 | 3 | — | |
GHZZKDIRNWVGOA
|
6.7 | IC50 | 2 | — | |
JDNCJZHDKRCMPJ
|
6.7 | IC50 | 2 | — | |
SKKOLYYKBOHFIL
|
6.7 | IC50 | 2 | — | |
UTZIAOQRNXJCSV
|
6.7 | IC50 | 2 | — | |
XKVWTVIOHRIVIZ
|
6.7 | IC50 | 4 | — | |
BEWNGQMBEVZWOA
|
6.7 | IC50 | 4 | — | |
VDKSZWXBGUWQAQ
|
6.7 | IC50 | 2 | — | |
VOJWGGTZIBFRLD
|
6.7 | IC50 | 2 | — | |
FCTSDHPUCRRBOK
|
6.6 | IC50 | 2 | — | |
PNRIWQJDPMCJMC
|
6.6 | IC50 | 2 | — | |
FUXZGPPEJFSVLE
|
6.6 | IC50 | 2 | — | |
DFUUFMXIWXRVSC
|
6.6 | Kd | 2 | — | |
MHIWHHOLYWCPAQ
|
6.6 | Kd | 2 | — | |
QAWXEOBACQVHDL
|
6.6 | IC50 | 2 | — | |
WHKVCJHBYDWODM
|
6.6 | IC50 | 2 | — | |
BPNNNYROBOUMKH
|
6.6 | IC50 | 2 | — | |
SLDHXYALWLMHEO
|
6.6 | IC50 | 2 | — | |
ATKLXHUMKYDIQA
|
6.6 | IC50 | 2 | — | |
PONPMHNRESGPEZ
|
6.6 | IC50 | 2 | — | |
RCYZJMHAZBYKMI
|
6.6 | IC50 | 2 | — | |
RRGYQZSBDNWDJM
|
6.6 | Ki | 2 | — | |
OFEGIUHAMIWNEU
|
6.6 | Ki | 2 | — | |
VCHUVBOJPRHHGT
|
6.6 | IC50 | 2 | — | |
CKXJADBCEBWSHG
|
6.6 | IC50 | 2 | — | |
BEZNLIPMYCSTDS
|
6.6 | IC50 | 2 | — | |
BEZNLIPMYCSTDS
|
6.6 | IC50 | 2 | — | |
LNJOONXJASRMBV
|
6.6 | IC50 | 2 | — |