Target Details
| UniProt AC | P18031 |
|---|---|
| Gene Symbol | PTPN1 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 511
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (4)
Active Molecules (511)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YGZGHANEFYTVGR
|
7.5 | IC50 | 2 | — | |
LFXAIDSJTUOQFR
|
7.5 | IC50 | 2 | — | |
LWVWNRJXLRQLPR
|
7.5 | IC50 | 2 | — | |
WVJWIEWUQYYLAY
|
7.5 | IC50 | 2 | — | |
CLRSCKINFSDJJY
|
7.5 | IC50 | 2 | — | |
UPDKUSVMZDXEOA
|
7.5 | IC50 | 2 | — | |
OGMLETJFLKSCML
|
7.5 | IC50 | 2 | — | |
OSQARHVGUZHHGT
|
7.5 | Ki | 2 | — | |
ASKBTOFTHQFAII
|
7.5 | IC50 | 2 | — | |
LGGCTIPSFMQVAC
|
7.5 | IC50 | 2 | — | |
NFYJBAFWWYMJRQ
|
7.5 | IC50 | 2 | — | |
DQQDAWIRIOIFBQ
|
7.5 | IC50 | 2 | — | |
FBFPKPPWVZPZDO
|
7.5 | IC50 | 2 | — | |
WSWRGQALHBTKAP
|
7.5 | IC50 | 2 | — | |
YLMTWYKRXNHYEX
|
7.5 | IC50 | 2 | — | |
ZCFDJLHEIXJWMR
|
7.5 | IC50 | 2 | — | |
NZTPDNHCASNUAT
|
7.5 | IC50 | 2 | — | |
ULSPKAJVYCBONR
|
7.4 | IC50 | 2 | — | |
YEAQQCBAQBWTDA
|
7.4 | IC50 | 2 | — | |
ACQKGLSIWFAMLA
|
7.4 | IC50 | 2 | — | |
NDSPEMBEVBIGPD
|
7.4 | IC50 | 2 | — | |
CWDWNOPXQHKDTA
|
7.4 | Ki | 2 | — | |
HAXBERRGQGXJNU
|
7.4 | IC50 | 2 | — | |
SYIZDBIAKCCYKI
|
7.4 | IC50 | 2 | — | |
UTZGYWMRZLQRNA
|
7.4 | IC50 | 2 | — | |
GWWTUJWRRCTCSI
|
7.4 | IC50 | 2 | — | |
GWWTUJWRRCTCSI
|
7.4 | IC50 | 2 | — | |
USHZWXCUJLENMD
|
7.4 | IC50 | 2 | — | |
APNZSLHVCOVLLC
|
7.4 | IC50 | 2 | — | |
GHQSTVDLTPVSRM
|
7.4 | IC50 | 2 | — | |
QOPBMVGFMRLORF
|
7.4 | Ki | 2 | — | |
NNVPHKXQFKGLHD
|
7.4 | IC50 | 2 | — | |
VGFNWVTYIUOBOR
|
7.4 | IC50 | 2 | — | |
HMUGMCSGKHKDGY
|
7.4 | Ki | 2 | — | |
MEACXYRFUVMDEQ
|
7.4 | IC50 | 2 | — | |
OMGQUFBPDFOYKP
|
7.4 | IC50 | 2 | — | |
AYYVCIVIOZHWEO
|
7.4 | IC50 | 2 | — | |
FBMYMFVFOFLWSL
|
7.4 | IC50 | 2 | — | |
NEXGDYGIWBZQBB
|
7.4 | IC50 | 2 | — | |
IQWGAAHPACZIDQ
|
7.4 | IC50 | 2 | — | |
KRBSOPWOZRXRRQ
|
7.4 | IC50 | 2 | — | |
UMPCSHCFHPFPLH
|
7.3 | IC50 | 2 | — | |
ALTWGIIQPLQAAM
|
7.3 | IC50 | 2 | — | |
LSGOVYNHVSXFFJ
|
7.3 | IC50 | 4 | — | |
PFZHAEHAZWEORU
|
7.3 | IC50 | 2 | — | |
LGLBYUGWPCGOBG
|
7.3 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.3 | Kd | 1075 | — | |
PKTGUMBRDSBGAA
|
7.3 | IC50 | 2 | — | |
IPNJQCVHNPGYOX
|
7.3 | IC50 | 2 | — | |
JNCPSODLWJEFQC
|
7.3 | IC50 | 5 | — |