Target Details
| UniProt AC | P18031 |
|---|---|
| Gene Symbol | PTPN1 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 511
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (4)
Active Molecules (511)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPHDXLHQZXGWHE
|
8.3 | IC50 | 2 | — | |
IGSRHSLPIMXATI
|
8.3 | IC50 | 2 | — | |
FYFGJSXDYQEBFJ
|
8.3 | IC50 | 2 | — | |
LAPGBIJFPPUGBM
|
8.3 | IC50 | 2 | — | |
JIIVYTJYOIJGBD
|
8.2 | IC50 | 2 | — | |
GBIIFVOJJXWYBK
|
8.2 | IC50 | 2 | — | |
IKMFYRRINXPKDQ
|
8.2 | IC50 | 2 | — | |
JYCQYNKZQPFRCV
|
8.2 | Ki | 2 | — | |
MQBLQNQFNLXLNE
|
8.2 | Ki | 2 | — | |
OLYDIQWQGAMQGY
|
8.2 | IC50 | 2 | — | |
NWWQGUAIJYKFLA
|
8.2 | IC50 | 2 | — | |
KEABENMPBSNYQR
|
8.2 | IC50 | 2 | — | |
QVSQVEINPYJMCF
|
8.2 | IC50 | 2 | — | |
SPPVIUWVPRGMHP
|
8.1 | IC50 | 2 | — | |
CHFWGYBRJKTHFL
|
8.1 | IC50 | 2 | — | |
NNBJKHVKXGWCKK
|
8.1 | IC50 | 2 | — | |
YBKOSQQXDYYDHT
|
8.1 | IC50 | 2 | — | |
GSWOTWPVTQSOFC
|
8.1 | IC50 | 2 | — | |
JPBWVFAXRYZXCR
|
8.1 | IC50 | 2 | — | |
YVEATRODDMUDLE
|
8.1 | IC50 | 2 | — | |
AYECJSPYFYCUEG
|
8.1 | IC50 | 2 | — | |
VVTVWJUCTYBBSN
|
8.1 | IC50 | 2 | — | |
FFMOCESMSKZHKT
|
8.1 | IC50 | 2 | — | |
NCPIGKQSZGEVJJ
|
8.1 | IC50 | 2 | — | |
SSOMGKXRFNKWLO
|
8.1 | IC50 | 2 | — | |
AIZHRJSCLDQRHW
|
8.0 | IC50 | 2 | — | |
IWYBGWRQXUJTOC
|
8.0 | IC50 | 2 | — | |
AIZHRJSCLDQRHW
|
8.0 | IC50 | 2 | — | |
MZUGWQGUEOQWFO
|
8.0 | IC50 | 2 | — | |
TYMUGKGQQMRQDI
|
8.0 | Ki | 2 | — | |
VTRFCUCEJIBDSE
|
8.0 | IC50 | 2 | — | |
ARNPBLSVPATIMI
|
8.0 | IC50 | 2 | — | |
KTEHTCIZIKZYJM
|
8.0 | IC50 | 2 | — | |
NUILBBMSKPQAHH
|
8.0 | IC50 | 2 | — | |
SOKOIOOIIJFRGN
|
8.0 | IC50 | 2 | — | |
JHSDETVLWLSJCK
|
7.9 | IC50 | 2 | — | |
JSQTVHLIHASFFJ
|
7.9 | IC50 | 2 | — | |
KZIABLBMUCEAFR
|
7.9 | IC50 | 2 | — | |
VFRGJCJXWUENFG
|
7.9 | IC50 | 2 | — | |
OVNWLVRODPOTMR
|
7.9 | IC50 | 2 | — | |
SZXQFEXBARNEFM
|
7.9 | IC50 | 2 | — | |
IUUJUPQTFPPAGO
|
7.9 | IC50 | 2 | — | |
DIUZJDCNEHZMBR
|
7.9 | IC50 | 2 | — | |
LWTPNPORLJJUTF
|
7.9 | IC50 | 2 | — | |
BTAGTGWPDROBMG
|
7.9 | IC50 | 2 | — | |
ZBWXOSLAWDYQKD
|
7.9 | IC50 | 2 | — | |
CWADQFRFGSOBTO
|
7.8 | IC50 | 2 | — | |
QEENZXFTRSDPEF
|
7.8 | Ki | 2 | — | |
VLRCQXLUVXXERA
|
7.8 | IC50 | 2 | — | |
VAIQRJONRRRIIM
|
7.8 | IC50 | 2 | — |