Target Details
| UniProt AC | P18031 |
|---|---|
| Gene Symbol | PTPN1 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 511
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (4)
Active Molecules (511)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYZCGGRZINLQBL
|
9.5 | IC50 | 8 | — | |
FKAWLXNLHHIHLA
|
9.3 | IC50 | 6 | — | |
KJYRSQLWJMEJNM
|
9.2 | IC50 | 2 | — | |
RFCWHQNNCOJYTR
|
9.2 | IC50 | 2 | — | |
KCHARSDIPZLYSD
|
9.0 | Ki | 2 | — | |
VILXHPHHLYDHSF
|
9.0 | IC50 | 2 | — | |
IXBQSRWSVIBXNC
|
8.9 | IC50 | 3 | — | |
DVFCRTGTEXUFIN
|
8.9 | IC50 | 2 | — | |
CUHZHOXGTHDNHJ
|
8.7 | Ki | 2 | — | |
FGSXDTAUWKYQDX
|
8.7 | Ki | 2 | — | |
FKOYIUYWMSVYKN
|
8.6 | Ki | 3 | — | |
DVFLCZRDIYUKAC
|
8.6 | IC50 | 2 | — | |
GACMVJUHSZEQKS
|
8.6 | IC50 | 2 | — | |
HRRVYDRPXPDYLV
|
8.6 | IC50 | 2 | — | |
IKXDLGHKPZYRQO
|
8.6 | IC50 | 2 | — | |
JJAKOVJYRJPWCA
|
8.6 | IC50 | 2 | — | |
JWMMMHPUESCKGP
|
8.6 | IC50 | 2 | — | |
LGTHMILFSZSRTC
|
8.6 | IC50 | 2 | — | |
QCQBPGLPSWQNRF
|
8.6 | IC50 | 2 | — | |
WAFGROQSQYZAFP
|
8.6 | IC50 | 2 | — | |
XONPLQMOBSLFAU
|
8.6 | IC50 | 2 | — | |
RHAMUMTWKSKBAD
|
8.6 | IC50 | 2 | — | |
CKONQMSCSZANCB
|
8.6 | IC50 | 2 | — | |
OVVNHIFLGPWASE
|
8.6 | IC50 | 2 | — | |
RQCOGPUQNNWPRV
|
8.5 | IC50 | 2 | — | |
DGVSSAPOBXDLAY
|
8.5 | Ki | 2 | — | |
DIRCLNUEXQQLRT
|
8.5 | IC50 | 2 | — | |
SUBZYMCEXNHIGE
|
8.5 | Ki | 2 | — | |
TUOKAOKHDHDMSS
|
8.5 | Ki | 2 | — | |
ZKLIYMLNDGMWPU
|
8.5 | IC50 | 2 | — | |
CVWLNWLJBZNMAZ
|
8.5 | IC50 | 2 | — | |
QNDVLZJODHBUFM
|
8.5 | IC50 | 7 | — | |
TYUZPPWVKQRZTK
|
8.5 | IC50 | 2 | — | |
NBHAOUUNAYVYOB
|
8.4 | IC50 | 2 | — | |
DSQQCWKGLUBDBP
|
8.4 | IC50 | 2 | — | |
SFVWMZDZTMHYBM
|
8.4 | IC50 | 2 | — | |
BBINWNMZKGHSMF
|
8.4 | Ki | 2 | — | |
FEPAAIQAIYOLJA
|
8.4 | Ki | 2 | — | |
KREWQXMKBWYIBM
|
8.4 | Ki | 2 | — | |
UBRICIIBZMGNGX
|
8.4 | IC50 | 2 | — | |
XZBONGJVYMLTQL
|
8.4 | IC50 | 2 | — | |
BMDONGLAMUYAQD
|
8.3 | IC50 | 2 | — | |
OQKUXLQNMZJIEY
|
8.3 | IC50 | 2 | — | |
OADLYFBQFFZCCM
|
8.3 | IC50 | 2 | — | |
UVMSRZSQDQTMKV
|
8.3 | Ki | 2 | — | |
ABRZBKRUFDGIHD
|
8.3 | IC50 | 2 | — | |
DELVPFVMXYCLMW
|
8.3 | IC50 | 2 | — | |
PWNDGSNZJKMHJB
|
8.3 | IC50 | 2 | — | |
QMJPTLBHDYKKJF
|
8.3 | IC50 | 2 | — | |
XFJJNGDTJHVAME
|
8.3 | Ki | 2 | — |