Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UTZFAVQAWTWOKK
|
7.5 | IC50 | 5 | — | |
IONVXRPWTRMITM
|
7.4 | Ki | 6 | — | |
LWAMOKCDAHOWOM
|
7.4 | IC50 | 3 | — | |
CPTVWYCNJGYSDW
|
7.4 | IC50 | 3 | — | |
QNIMLRHYPMIYSE
|
7.4 | IC50 | 7 | Yes | |
QXCNZYXAYYZRIY
|
7.4 | IC50 | 2 | Yes | |
SFCSGFUQASTWES
|
7.4 | IC50 | 3 | — | |
UQHQUPSFNPQLNI
|
7.4 | IC50 | 8 | Yes | |
VJRMARZDCXLFER
|
7.4 | IC50 | 3 | — | |
KIXJPVWFCZCXOL
|
7.4 | IC50 | 4 | Yes | |
KMXYTUMWDQTWTG
|
7.4 | IC50 | 3 | — | |
QKKIWEILHCXECO
|
7.4 | IC50 | 24 | — | |
AUNHGNQTPLHIRO
|
7.4 | IC50 | 2 | — | |
DOKIBWCVABZHOH
|
7.4 | IC50 | 3 | — | |
HEPDAJRNJBNJAE
|
7.4 | IC50 | 15 | Yes | |
IFPPYSWJNWHOLQ
|
7.4 | Ki | 52 | Yes | |
JTRNNNVASYCTLO
|
7.4 | Ki | 14 | — | |
MFMXAWQGPQXDRJ
|
7.4 | Ki | 27 | — | |
NHFDRBXTEDBWCZ
|
7.4 | Ki | 41 | — | |
NKEUPUJTVALZIK
|
7.4 | Ki | 28 | — | |
PIQCTGMSNWUMAF
|
7.4 | IC50 | 137 | Yes | |
RTDSHUGNRVXRHN
|
7.4 | Ki | 51 | — | |
UTBZTQCKLUFYTQ
|
7.4 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
7.4 | Ki | 56 | — | |
ZKHDDJKHTPLPOQ
|
7.4 | Ki | 62 | — | |
ZOTXBRHWIDKKFO
|
7.4 | IC50 | 4 | Yes | |
CVWXJKQAOSCOAB
|
7.4 | Kd | 35 | — | |
DEEQWPIMFASFIP
|
7.4 | IC50 | 7 | Yes | |
LQAMNACDVZLTDL
|
7.4 | IC50 | 5 | — | |
QTBWCSQGBMPECM
|
7.4 | IC50 | 21 | Yes | |
QUTYYJGQIXIMSJ
|
7.4 | Ki | 6 | — | |
LHKUVOGMYOGQMG
|
7.4 | Ki | 6 | — | |
TUGBVZCJQUNZOM
|
7.4 | IC50 | 2 | — | |
WUWDLXZGHZSWQZ
|
7.4 | IC50 | 11 | Yes | |
YMKCMNJQFGEWCA
|
7.4 | IC50 | 8 | Yes | |
HOZCIXWJOIJVFG
|
7.4 | IC50 | 2 | — | |
NEJMZWVLFRWQSG
|
7.4 | IC50 | 3 | — | |
RBOQJYWZBIOHKR
|
7.4 | IC50 | 2 | Yes | |
LTJCRCKPWKQPOV
|
7.3 | Ki | 6 | — | |
ONSZEUCTVQJHOZ
|
7.3 | IC50 | 9 | — | |
RHEKRIVAMQDVLV
|
7.3 | IC50 | 3 | — | |
HESUKNSDMPJYHF
|
7.3 | Ki | 6 | — | |
SHKVYTQIJOOEMA
|
7.3 | IC50 | 6 | — | |
XYGDYCMPYIUPHS
|
7.3 | IC50 | 4 | Yes | |
GZOYOEIHAGHGFM
|
7.3 | IC50 | 6 | — | |
JAYZLGOACZERIJ
|
7.3 | IC50 | 7 | Yes | |
PYUIBNGQBBAKFO
|
7.3 | IC50 | 7 | Yes | |
BLYDOULCQABGHT
|
7.3 | Ki | 6 | — | |
CGDLXUGHZUDIDJ
|
7.3 | IC50 | 3 | — | |
GFMYTWVSAZEZRD
|
7.3 | IC50 | 2 | Yes |