Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJZXDUKUMALHNP
|
7.6 | Ki | 10 | — | |
IXIJKXSIADDKHR
|
7.6 | IC50 | 12 | — | |
KHOVFNRAIYTEPO
|
7.6 | Ki | 5 | — | |
KJTNEZSZMBPREH
|
7.6 | IC50 | 2 | — | |
KNCMFVBGBJGBGI
|
7.6 | IC50 | 7 | Yes | |
MVJMMLFMPWITEJ
|
7.6 | Ki | 110 | — | |
OWRXHGAFWZFFCW
|
7.6 | Ki | 113 | — | |
QDCNUYNTRDKBDB
|
7.6 | IC50 | 3 | — | |
RKKIDHHGKNGTQI
|
7.6 | Ki | 28 | — | |
RTYJMUXLFRYRBU
|
7.6 | Ki | 35 | — | |
SIABKVPDKZOJCK
|
7.6 | IC50 | 5 | Yes | |
TXHOCWWJSGCZLC
|
7.6 | Ki | 18 | — | |
PSWWUMTWJRPKLC
|
7.6 | IC50 | 3 | — | |
ZJFCBQXPTQSTCZ
|
7.6 | IC50 | 8 | — | |
FAYFMVHYNQOQRQ
|
7.6 | IC50 | 7 | Yes | |
HWZNBJUXOVHGSL
|
7.6 | Ki | 6 | — | |
IFUCZPASJWTYRU
|
7.5 | IC50 | 5 | — | |
JBJZIAHKSVQDAN
|
7.5 | IC50 | 5 | Yes | |
NHFDRBXTEDBWCZ
|
7.5 | IC50 | 12 | Yes | |
OSHPNNCEUZTANR
|
7.5 | IC50 | 4 | Yes | |
SQUBJXXBYMPOFW
|
7.5 | IC50 | 6 | Yes | |
VFUZEFVLUHADNS
|
7.5 | IC50 | 4 | Yes | |
CXMKJARIDJFGGI
|
7.5 | IC50 | 3 | — | |
IQCIFDSCWKQXJA
|
7.5 | IC50 | 4 | — | |
DEXMHPPNXPZZKY
|
7.5 | IC50 | 3 | — | |
KWVDRTIIZKGPOQ
|
7.5 | Ki | 6 | — | |
AYBLFKIMJMUPEC
|
7.5 | Ki | 6 | — | |
LDACHLNBCOVNBL
|
7.5 | IC50 | 8 | — | |
MYMOMVBHZSIFSG
|
7.5 | IC50 | 2 | — | |
UXTWDPHPOWZONL
|
7.5 | IC50 | 2 | Yes | |
XHXOJKOXEKXDSQ
|
7.5 | IC50 | 5 | Yes | |
KULLGNXUHQGZIB
|
7.5 | IC50 | 3 | — | |
MLDQJTXFUGDVEO
|
7.5 | Kd | 85 | Yes | |
VHIADSOUXPEWOM
|
7.5 | Ki | 6 | — | |
FDVSOQRNTAPCHB
|
7.5 | Ki | 40 | — | |
JLFPGEKGHMUMDY
|
7.5 | Ki | 6 | — | |
JMVVTEATJVVTPU
|
7.5 | Ki | 6 | — | |
SKZQZGSPYYHTQG
|
7.5 | IC50 | 3 | — | |
TVUWQDLBEOZVOU
|
7.5 | Ki | 41 | — | |
BALLNEJQLSTPIO
|
7.5 | IC50 | 3 | — | |
SLZDAHQKZCFNCA
|
7.5 | IC50 | 3 | — | |
XYJONLOLMGUYBZ
|
7.5 | IC50 | 6 | — | |
KUYVWUAGELSGSE
|
7.5 | IC50 | 2 | — | |
QTIHZRQNFPNCHT
|
7.5 | IC50 | 4 | — | |
XZXHXSATPCNXJR
|
7.5 | IC50 | 165 | Yes | |
BYSPSKYBWHPEJW
|
7.5 | IC50 | 6 | — | |
JLXBHBVYBGZIEY
|
7.5 | IC50 | 7 | Yes | |
PSNSRJNHZPJVJH
|
7.5 | IC50 | 18 | — | |
PWDPLHOKCYLVIC
|
7.5 | IC50 | 5 | — | |
SQQOETQMUXTTJU
|
7.5 | IC50 | 3 | — |