Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLEMEZZZALNBAS
|
7.8 | IC50 | 2 | — | |
QHWJRQVVIZMMLO
|
7.8 | IC50 | 2 | — | |
QLVYHQCCXVCBRH
|
7.8 | IC50 | 2 | — | |
AZOXWOCICFEBCQ
|
7.8 | IC50 | 11 | — | |
BPXQYAXTDCQZHB
|
7.8 | IC50 | 7 | Yes | |
ULUUNYJTTJIXHY
|
7.8 | IC50 | 2 | — | |
ABDZDGAYOUCIOR
|
7.8 | IC50 | 4 | — | |
GVEYCTQROBIZHZ
|
7.8 | IC50 | 5 | — | |
VOYMOBPSYVKQGF
|
7.8 | IC50 | 3 | — | |
UNERFOYGRRSDAU
|
7.7 | IC50 | 2 | — | |
VLXIXYDIKYYMAQ
|
7.7 | IC50 | 7 | — | |
YRXBBYUECWYNNN
|
7.7 | IC50 | 2 | — | |
AAVVJYRIFZWOQJ
|
7.7 | IC50 | 3 | — | |
HIFPXVLZYKQXID
|
7.7 | IC50 | 3 | — | |
NZBQAOCZTUIYGZ
|
7.7 | IC50 | 3 | — | |
DMQYDVBIPXAAJA
|
7.7 | IC50 | 4 | — | |
FLEAYYMORDPWAJ
|
7.7 | Ki | 90 | — | |
FTDWSWREBGYXDZ
|
7.7 | IC50 | 10 | — | |
HCAUEIOBSYOQPN
|
7.7 | IC50 | 5 | Yes | |
IBHVLWYGIJLFTH
|
7.7 | IC50 | 2 | — | |
MSHIDVJWNMVTDI
|
7.7 | IC50 | 3 | — | |
QLJWNTHEJPFKDE
|
7.7 | IC50 | 2 | — | |
SDBOIBYRBWPIEL
|
7.7 | Ki | 31 | — | |
SUSFJVCPEPRLCX
|
7.7 | IC50 | 6 | Yes | |
UDVJBRYBBSVDDS
|
7.7 | IC50 | 14 | — | |
WUWDLXZGHZSWQZ
|
7.7 | Ki | 41 | — | |
YADAQXVHBLKOIU
|
7.7 | IC50 | 4 | — | |
HMKZBWZSRGIVPM
|
7.7 | IC50 | 2 | — | |
QNDAYXSCYXLLNB
|
7.7 | IC50 | 3 | — | |
ADFZKKWKESWUFY
|
7.7 | IC50 | 8 | — | |
HZJFSGCBXSPJTM
|
7.7 | IC50 | 2 | Yes | |
IPBGKKBBYNOXCG
|
7.7 | IC50 | 10 | — | |
IXKNBAGOTATIPL
|
7.7 | IC50 | 2 | — | |
MHHCPQUFBADOGH
|
7.7 | IC50 | 3 | — | |
WOSKHXYHFSIKNG
|
7.7 | IC50 | 24 | — | |
YUAOWJBCURIMGN
|
7.7 | IC50 | 3 | — | |
HUBJRBJFRJHZIG
|
7.7 | IC50 | 3 | — | |
AMQUNUQXLQUCGJ
|
7.6 | IC50 | 3 | — | |
DSRUNANRDDLTEB
|
7.6 | IC50 | 9 | — | |
GUDCGYXTFRTWMP
|
7.6 | IC50 | 3 | — | |
PVNVVSOCNKJUKM
|
7.6 | IC50 | 3 | — | |
UXWPGZNWYZLVFJ
|
7.6 | IC50 | 3 | — | |
VAARYSWULJUGST
|
7.6 | Kd | 119 | Yes | |
SWNPCLQLHUWVAZ
|
7.6 | IC50 | 9 | Yes | |
UFWXSGVSQZKZTR
|
7.6 | IC50 | 4 | — | |
UGWUUDYHNSCFBW
|
7.6 | IC50 | 2 | — | |
YZRLWPBYTMKRQR
|
7.6 | IC50 | 11 | — | |
BLQYVHBZHAISJM
|
7.6 | Ki | 54 | — | |
CKVWQORGCCEYHS
|
7.6 | Ki | 50 | — | |
CYPOOUITBHWAKE
|
7.6 | IC50 | 4 | — |