Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NMJILYFXNANMKC
|
8.0 | IC50 | 3 | — | |
SAJGQCIKURPXJS
|
8.0 | IC50 | 2 | — | |
VDSFUPFAWFPWHF
|
8.0 | IC50 | 4 | Yes | |
XHBVYDAKJHETMP
|
8.0 | IC50 | 24 | Yes | |
QEUXOHWRZLJLKW
|
8.0 | IC50 | 2 | — | |
SPMVMDHWKHCIDT
|
8.0 | IC50 | 5 | — | |
WSHIGLALBLRQGR
|
8.0 | IC50 | 2 | — | |
QKIHSGVZMXIBJB
|
7.9 | IC50 | 2 | — | |
ZYOXZBUWXWSWBB
|
7.9 | IC50 | 2 | — | |
FALXZGBOUDIVJB
|
7.9 | IC50 | 2 | — | |
JKDOLJKPWNOURO
|
7.9 | IC50 | 3 | — | |
JZGWDENJLOXKLZ
|
7.9 | IC50 | 4 | — | |
NEQZWEXWOFPKOT
|
7.9 | IC50 | 9 | Yes | |
ONIQOQHATWINJY
|
7.9 | IC50 | 25 | — | |
GXYDEHHVGKZABR
|
7.9 | IC50 | 2 | — | |
JIVWUFIEWHRAPG
|
7.9 | IC50 | 2 | — | |
ACNCCUVYXQGPKZ
|
7.9 | Ki | 31 | — | |
JSDGKSMNPHJDFK
|
7.9 | Ki | 35 | — | |
NWAUBAGBGOPJLF
|
7.9 | Ki | 51 | Yes | |
BNQPYLKCEUFMIL
|
7.9 | IC50 | 2 | — | |
FNHKPVJBJVTLMP
|
7.9 | IC50 | 29 | — | |
FWBUUGDBUKHCQX
|
7.9 | IC50 | 3 | — | |
JYJKNIHQZXCKPB
|
7.9 | IC50 | 2 | — | |
SJAAIJHENJPXTP
|
7.9 | IC50 | 2 | — | |
VPBYZLCHOKSGRX
|
7.9 | IC50 | 4 | — | |
IAYMHFSZYNWIEK
|
7.9 | IC50 | 2 | — | |
LJWDDKOCLWIIHJ
|
7.9 | IC50 | 2 | — | |
OYGVKPPKBAPROS
|
7.9 | IC50 | 2 | — | |
SOXNNGFGYDFPDL
|
7.9 | IC50 | 3 | — | |
ARXCFPVKEORMCL
|
7.8 | IC50 | 2 | — | |
CUIHSIWYWATEQL
|
7.8 | IC50 | 61 | Yes | |
DKNUPRMJNUQNHR
|
7.8 | Kd | 33 | — | |
NDIUYMHNCUTVGE
|
7.8 | Ki | 25 | — | |
QBRQTJMZEYORSP
|
7.8 | Kd | 12 | — | |
UKSRSPVTFVLKRY
|
7.8 | IC50 | 4 | Yes | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
BWWXVHUBUHUAHC
|
7.8 | IC50 | 2 | — | |
DBWLZXDWSDEPMX
|
7.8 | IC50 | 2 | — | |
HUQYQFBIFGUUQQ
|
7.8 | IC50 | 2 | Yes | |
IKVZCSGUEDRZOZ
|
7.8 | IC50 | 2 | — | |
TWOLOZGQZKJZKJ
|
7.8 | IC50 | 7 | Yes | |
YHVHYWYQEFELOW
|
7.8 | IC50 | 44 | — | |
FGZIONRFHVNRJB
|
7.8 | IC50 | 3 | — | |
HDFUJTPEMGTANU
|
7.8 | IC50 | 2 | — | |
KOHNRDPXFDZZJF
|
7.8 | Ki | 31 | — | |
LIRCRNNNGSPSBY
|
7.8 | IC50 | 2 | — | |
MLIFNJABMANKEU
|
7.8 | IC50 | 9 | Yes | |
MTCHQDWUHQADSY
|
7.8 | Ki | 29 | — | |
NHHQJBCNYHBUSI
|
7.8 | Kd | 220 | — | |
PATGADWTCHRVOQ
|
7.8 | IC50 | 9 | Yes |