Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTHSJRSUDUUQFI
|
8.1 | IC50 | 3 | — | |
IFFBOVLYGJAFKB
|
8.1 | IC50 | 5 | — | |
UVZNMKLHIOHOBN
|
8.1 | IC50 | 3 | — | |
DSBPVMDUESDKNK
|
8.1 | IC50 | 9 | Yes | |
MHZIGJBWNNGGBZ
|
8.1 | IC50 | 3 | — | |
MPVGZUGXCQEXTM
|
8.1 | IC50 | 61 | Yes | |
FGPIVIJULBNRBX
|
8.1 | IC50 | 4 | — | |
AEXAYHMFAIXNSU
|
8.1 | IC50 | 2 | Yes | |
APUCFXHENVUXCY
|
8.1 | Ki | 15 | — | |
BOBGABAXWFYHQX
|
8.1 | Ki | 9 | — | |
CSJKWUOGGSICJS
|
8.1 | IC50 | 2 | — | |
NVQDLTVJFMBRNP
|
8.1 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
8.1 | Ki | 33 | — | |
RSUMIXOOUBJDRH
|
8.1 | IC50 | 2 | — | |
SBPVMWFTFWQYKB
|
8.1 | IC50 | 2 | — | |
WPXVVAWAHQHJPF
|
8.1 | IC50 | 41 | — | |
YCZNRSBAKIVMMQ
|
8.1 | IC50 | 2 | — | |
BMFHAIYLTOVZTR
|
8.1 | IC50 | 2 | — | |
BYDMGYUSZLFTLB
|
8.1 | IC50 | 2 | — | |
KNDPXYAMINMLED
|
8.1 | IC50 | 11 | — | |
BRFOGQVFBWDQGX
|
8.1 | IC50 | 6 | — | |
ZAJKUNDNLWGYKD
|
8.1 | IC50 | 3 | — | |
KEDANNMRCOENMZ
|
8.1 | IC50 | 7 | — | |
PHXJVRSECIGDHY
|
8.1 | IC50 | 59 | — | |
DNBSBOYLZWOFKX
|
8.1 | IC50 | 2 | — | |
DVMIIUOULRDNLG
|
8.1 | IC50 | 3 | — | |
QCARBCGPQHFPOS
|
8.1 | IC50 | 2 | — | |
UQRZISCZHYAQAL
|
8.1 | IC50 | 2 | — | |
ZFHLKLQIDSNDHN
|
8.1 | IC50 | 3 | — | |
KBLQLKPQLQTCDT
|
8.0 | IC50 | 3 | — | |
KOFXELGVKHKUJR
|
8.0 | IC50 | 3 | — | |
UFRGYRZAPMGFPZ
|
8.0 | IC50 | 2 | — | |
IHJBFEQZLKXMGF
|
8.0 | IC50 | 3 | — | |
BWLBVHWCNZAPOW
|
8.0 | IC50 | 4 | — | |
GCYXEGSPUDSZJY
|
8.0 | Ki | 82 | — | |
IHGRRQDGJVUJSZ
|
8.0 | IC50 | 2 | — | |
JGEBLDKNWBUGRZ
|
8.0 | IC50 | 20 | Yes | |
KTQYQHLIMZOBSM
|
8.0 | Ki | 12 | — | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
LRYKPJMJKRDDIX
|
8.0 | IC50 | 3 | Yes | |
PUPCRRRSBUYJAD
|
8.0 | Ki | 44 | Yes | |
PYXQMJSGJIJHJT
|
8.0 | Ki | 28 | — | |
QKPLUKMJEKRAJD
|
8.0 | IC50 | 30 | Yes | |
RIUZPIBUSOHUKF
|
8.0 | Ki | 23 | — | |
RYYNGWLOYLRZLK
|
8.0 | Ki | 104 | — | |
YUZDAIVFOGPJIS
|
8.0 | IC50 | 2 | Yes | |
ZXLFIHLBHMLHFJ
|
8.0 | Ki | 31 | — | |
JPMRQZPGRKLGGS
|
8.0 | IC50 | 2 | — | |
FAIYNQQPUQQMIC
|
8.0 | IC50 | 3 | — | |
JEUQHZZAJFLFGO
|
8.0 | IC50 | 4 | — |