Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HAWQJVUHZAYNCF
|
8.3 | IC50 | 5 | — | |
AGYRJOAGMDIFKL
|
8.3 | Ki | 17 | — | |
CXBBWVXSZINRCS
|
8.3 | Ki | 41 | — | |
CXMPCGNEOYUNQP
|
8.3 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
HOGCJPPMBAIRFC
|
8.3 | IC50 | 2 | — | |
JCKSFAJUCQVQOF
|
8.3 | IC50 | 2 | — | |
LYHXSDWIWVVZPB
|
8.3 | IC50 | 6 | Yes | |
MADCXGNPDBWPLM
|
8.3 | Ki | 25 | — | |
NFKMFNBKEOQNPZ
|
8.3 | Ki | 43 | — | |
NRZYTPAJGVTKIM
|
8.3 | Ki | 38 | — | |
QXRJBJVCBQSLTA
|
8.3 | Ki | 29 | — | |
QYULUQACUCDZHT
|
8.3 | IC50 | 2 | — | |
SILANKVZJSUJHJ
|
8.3 | IC50 | 9 | — | |
SJSZXGFLISXGGM
|
8.3 | IC50 | 2 | — | |
SJXKDSURXYKBQG
|
8.3 | IC50 | 2 | — | |
UCHQCSDTPQKAKL
|
8.3 | IC50 | 9 | Yes | |
UWDBNTXEKYRMSG
|
8.3 | Ki | 26 | — | |
XXJWYDDUDKYVKI
|
8.3 | IC50 | 52 | — | |
SUXYGJZMCWKJJI
|
8.3 | IC50 | 26 | Yes | |
ZDMGPVTVMCERRZ
|
8.3 | IC50 | 3 | — | |
FYLZILJOKOVUAW
|
8.3 | IC50 | 3 | — | |
MPCFFXIIMLGUSM
|
8.3 | IC50 | 2 | — | |
AISWQGLURAAAKE
|
8.2 | IC50 | 7 | — | |
OIANGKGOYKDGQV
|
8.2 | Kd | 10 | — | |
AGFATOYGCIURQX
|
8.2 | IC50 | 2 | — | |
IUNORHVEZRZFIC
|
8.2 | IC50 | 2 | — | |
OPPRLSONSGULSP
|
8.2 | IC50 | 7 | Yes | |
SNYMIRFSGCNEHH
|
8.2 | IC50 | 2 | Yes | |
TYSQFVMRVYDAEQ
|
8.2 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.2 | Ki | 31 | — | |
SPMVMDHWKHCIDT
|
8.2 | IC50 | 30 | — | |
XLFYOIVELARSKP
|
8.2 | Ki | 33 | — | |
XNEPVLVYFUGJLF
|
8.2 | Ki | 27 | — | |
XYXLUJQBBIBJFV
|
8.2 | Ki | 36 | — | |
UYWCBKUMESQOKL
|
8.2 | IC50 | 5 | — | |
CXQHYVUVSFXTMY
|
8.2 | IC50 | 154 | — | |
GUOKMFDFLUGBPS
|
8.2 | IC50 | 7 | Yes | |
PFPXVMRFOYULPT
|
8.2 | IC50 | 7 | Yes | |
CBVLEYGWBRVGRZ
|
8.2 | IC50 | 2 | — | |
CCUYECGXGAFGTM
|
8.2 | IC50 | 2 | — | |
CUDVHEFYRIWYQD
|
8.2 | IC50 | 11 | — | |
DFTANXXGINSIBO
|
8.2 | IC50 | 2 | — | |
GEGCXGMFUYJULA
|
8.2 | IC50 | 30 | Yes | |
HHPVWJJNJSJOLQ
|
8.2 | IC50 | 3 | — | |
LSVIBAPJYUUVJJ
|
8.2 | IC50 | 4 | — | |
ONHZXYNGPZWHBN
|
8.2 | IC50 | 3 | — | |
OZMHYBXYOWXNJV
|
8.2 | IC50 | 2 | — | |
XHCPCYVQXFHJAU
|
8.2 | IC50 | 12 | — | |
XZJHYNMIHBWFCD
|
8.2 | IC50 | 3 | — |