Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJHIKUXWIQORDE
|
8.5 | IC50 | 2 | — | |
CNIWCJQSFDYIDI
|
8.5 | IC50 | 3 | — | |
CSGDFNSJHVTVHD
|
8.5 | IC50 | 2 | Yes | |
FPTZKIGUSULXNI
|
8.5 | IC50 | 2 | — | |
GITNDHUJOBXSCE
|
8.5 | IC50 | 4 | — | |
HZIZEKOMOILAJT
|
8.5 | IC50 | 6 | Yes | |
MEAHQSFATRAJHG
|
8.5 | IC50 | 2 | — | |
QGRWLEOULVUBBC
|
8.5 | IC50 | 2 | Yes | |
QMTUQSYQTDJUEC
|
8.5 | IC50 | 2 | — | |
ZMZOKLZTXMCMNW
|
8.5 | IC50 | 4 | — | |
IWBIEKJAAQYGMI
|
8.5 | IC50 | 3 | — | |
LKWJIINNTXDWNN
|
8.5 | IC50 | 3 | — | |
AYJBHLUSGLQYDG
|
8.5 | Ki | 16 | — | |
KKYPRNBBPBRJQX
|
8.5 | Ki | 40 | — | |
KUNZDWIFPOMUOX
|
8.5 | Ki | 36 | — | |
LCGSWTFWYNYUKS
|
8.5 | Ki | 26 | — | |
RAPYFGJGASETOS
|
8.5 | Ki | 11 | — | |
XWFXAJNJXGILIN
|
8.5 | IC50 | 3 | — | |
DZFZXPPHBWCXPQ
|
8.5 | IC50 | 12 | — | |
NMMQJLYMIJYIAK
|
8.5 | IC50 | 3 | — | |
RFHIMTLASCGOTR
|
8.4 | IC50 | 3 | — | |
HSKISFLIRPOYCF
|
8.4 | IC50 | 5 | — | |
QAGLJDWYCCJEHH
|
8.4 | IC50 | 7 | Yes | |
OSZVHJYNXBUVAH
|
8.4 | IC50 | 12 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
BDTDDTOUVUTYCH
|
8.4 | IC50 | 2 | — | |
BRKGRQVBHFZISR
|
8.4 | IC50 | 7 | Yes | |
DDSTUHINLNZIIZ
|
8.4 | IC50 | 2 | Yes | |
FTHVRWNSFRDQNV
|
8.4 | IC50 | 2 | — | |
GALVWTFFXPRMQM
|
8.4 | Ki | 20 | — | |
GNOLTAIPEDJTSV
|
8.4 | IC50 | 2 | — | |
HRZOUBQYVUXBNS
|
8.4 | Ki | 38 | — | |
JRKYKAKARRYSSS
|
8.4 | IC50 | 14 | Yes | |
LNTWWMOOPMLARL
|
8.4 | IC50 | 2 | — | |
MDSJWBBQCSEPDO
|
8.4 | IC50 | 2 | — | |
MULNSLQVKKUPJN
|
8.4 | Ki | 41 | — | |
MVLNKEXGMMGTDC
|
8.4 | IC50 | 2 | — | |
NBYJQDZZRITHTA
|
8.4 | IC50 | 2 | — | |
PDLBTPKSQYCOOT
|
8.4 | IC50 | 2 | — | |
PJSBFZAYJQMORO
|
8.4 | Ki | 11 | — | |
RQIXEOXMOHDTLC
|
8.4 | IC50 | 2 | — | |
SEVCBWKJSOLMNQ
|
8.4 | Ki | 38 | — | |
UCSSQROSBFPVKH
|
8.4 | IC50 | 7 | Yes | |
UYTRUCYRZKTLND
|
8.4 | IC50 | 2 | Yes | |
VTLQAHPWBDJOFR
|
8.4 | IC50 | 2 | — | |
ZAARMHXLYCHRAK
|
8.4 | Ki | 20 | — | |
GUUYUIDTJAWAHO
|
8.4 | IC50 | 4 | — | |
ADLPKFFMGIJZIM
|
8.4 | IC50 | 44 | — | |
DELFTXSEBVUJAK
|
8.4 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
8.3 | Kd | 151 | — |