Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GSXRCPJTNIGKSZ
|
9.0 | Ki | 43 | — | |
HKZKELVPGXJIMW
|
9.0 | Ki | 41 | — | |
QXIOZIFTPMAING
|
9.0 | IC50 | 17 | — | |
RPDVCUCXMGWTFA
|
9.0 | Ki | 10 | — | |
SMWFHLHWOOWYAP
|
9.0 | IC50 | 4 | Yes | |
SXKJHBJVKCAXFA
|
9.0 | IC50 | 3 | — | |
ZGDSBEUMPIMXBM
|
9.0 | Ki | 42 | — | |
QEXZHTIPIXJKTN
|
9.0 | IC50 | 3 | — | |
PIBOSMWVYTUUIX
|
9.0 | IC50 | 3 | — | |
STINDBVFOPRZHE
|
9.0 | IC50 | 8 | Yes | |
FQYLJBVSYHZWLT
|
8.9 | Ki | 35 | Yes | |
LVECPYVAIBNSRV
|
8.9 | Ki | 33 | — | |
QJIVDCJIPGAKQZ
|
8.9 | Ki | 25 | — | |
KGSRYTUWXUESJK
|
8.9 | IC50 | 7 | — | |
HPTVZCOLBBFDMI
|
8.8 | IC50 | 3 | — | |
TTZSNFLLYPYKIL
|
8.8 | IC50 | 7 | — | |
BRTHUECZMVKNMQ
|
8.8 | IC50 | 7 | — | |
CQBBMNXXVMOFCA
|
8.8 | Ki | 39 | — | |
GMYYMEOGFRKSFS
|
8.8 | Ki | 29 | — | |
OWFXKTOLFUQPDJ
|
8.8 | Ki | 36 | — | |
RWEHAHIEUDLKGT
|
8.8 | Ki | 33 | — | |
UXMNYFJHEBEDJS
|
8.8 | Ki | 19 | Yes | |
YDWMUCKJUNLURC
|
8.8 | Ki | 24 | — | |
WINHZLLDWRZWRT
|
8.7 | Kd | 201 | Yes | |
WJZSUSVUKVZGLF
|
8.7 | IC50 | 7 | Yes | |
UGEJLCNSVIVALC
|
8.7 | IC50 | 41 | — | |
CFIBXVQLBVNOHW
|
8.7 | Ki | 64 | — | |
CNTCGRJDUJEUDG
|
8.7 | Ki | 37 | — | |
DZSUJUOJJJCWGG
|
8.7 | IC50 | 55 | Yes | |
JPKSISIJPSXDLA
|
8.7 | IC50 | 10 | Yes | |
MZEOWSVWCPCLAR
|
8.7 | IC50 | 2 | Yes | |
PSRIIUUKNWOHQJ
|
8.7 | IC50 | 2 | — | |
PTUJZMRANLZUJP
|
8.7 | IC50 | 2 | — | |
RAHBGWKEPAQNFF
|
8.7 | IC50 | 26 | — | |
WSBZFFNSBMBYQA
|
8.7 | IC50 | 9 | — | |
YEPNVBNYCRGZRX
|
8.7 | Ki | 26 | — | |
VKBFHTIUXUCYRQ
|
8.7 | IC50 | 8 | — | |
AMRDEKYBJXNLRC
|
8.7 | IC50 | 3 | — | |
OSPKANQURMXUIE
|
8.7 | IC50 | 7 | Yes | |
PLKAJXMYXBXIGX
|
8.7 | IC50 | 7 | Yes | |
WPHKIQPVPYJNAX
|
8.7 | IC50 | 81 | — | |
NKKLZQAIJJQHIF
|
8.7 | IC50 | 3 | — | |
GDEJPGKNPRJNGE
|
8.6 | Ki | 6 | — | |
PTVPBWWDGZSEAF
|
8.6 | Ki | 63 | — | |
VCFDMLBPASGZTP
|
8.6 | Ki | 38 | — | |
VZRLBUJXKJBRFA
|
8.6 | IC50 | 3 | — | |
MZZIULFUXGVMGF
|
8.5 | IC50 | 3 | — | |
PMCATQTXBPQRSD
|
8.5 | IC50 | 3 | — | |
AQYYPSFZMCKSEL
|
8.5 | IC50 | 4 | Yes | |
CIAUVJBQJHPXQG
|
8.5 | IC50 | 2 | — |