Target Details
| UniProt AC | P17948 |
|---|---|
| Gene Symbol | FLT1 |
| Protein Name | Vascular endothelial growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 1,237
- Clinical molecules 189
- Avg pChEMBL 7.18
KEGG Pathways (10)
Active Molecules (1,237)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FOONBYIHFUMRSX
|
10.3 | Ki | 12 | — | |
SJMFZIGFOIPNPE
|
10.2 | Ki | 10 | — | |
HQPNLIKXAPLWBQ
|
10.1 | Ki | 12 | Yes | |
JPTQVDRPKXSDDN
|
10.0 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
10.0 | IC50 | 43 | — | |
ZQQVWTACALNOAJ
|
10.0 | Ki | 11 | — | |
QDOBTYVGPGFRCM
|
9.9 | Ki | 11 | — | |
BDPBZUHWAVABDM
|
9.8 | Ki | 11 | — | |
DMTDZFGYURLLKX
|
9.8 | Ki | 13 | Yes | |
DBXOMQJZSQLQED
|
9.7 | Ki | 12 | — | |
MCCCQFAOMZMZKE
|
9.7 | Ki | 52 | — | |
DKSNLQYRZJKYOC
|
9.6 | Ki | 51 | — | |
DLPARMNJOHFOLU
|
9.6 | Ki | 14 | Yes | |
MHCPAORAYMTGCZ
|
9.6 | Ki | 37 | — | |
QAKMQVCMEPKBHL
|
9.6 | Ki | 11 | — | |
KROLCVQARUUHNV
|
9.5 | Ki | 12 | — | |
RKLGMDOZEOTQEM
|
9.5 | Ki | 12 | — | |
ULHGAQSVFPOUDY
|
9.5 | Ki | 43 | — | |
BHSOPYVVEZFHDB
|
9.4 | Ki | 25 | Yes | |
SFPWNTQWFFNJIH
|
9.4 | Ki | 48 | — | |
UOOZSMNSBYVUGZ
|
9.4 | Ki | 32 | — | |
UTQPKPHUIMHAAN
|
9.4 | Ki | 22 | — | |
XBYVOPRDASFDMY
|
9.4 | Ki | 42 | — | |
XJSFDMGICAWQFS
|
9.4 | Ki | 60 | — | |
GWMATETWMAQOFL
|
9.3 | Ki | 36 | — | |
RBXYGQNZRVPDNB
|
9.3 | Ki | 34 | — | |
WUBFAXNVDMCVIO
|
9.3 | IC50 | 12 | Yes | |
XHORJSJFHVABEA
|
9.3 | Ki | 49 | — | |
XOOAAYRIVATZNM
|
9.3 | Ki | 55 | — | |
YACXOXQTGJXYNX
|
9.3 | Ki | 11 | — | |
KNACLJBHKVSTDL
|
9.2 | Ki | 40 | — | |
NSKFXNDKPCVDIN
|
9.2 | Ki | 12 | — | |
NWMPVMMGSHXANZ
|
9.2 | Ki | 58 | — | |
QONPPIZSNSSCSK
|
9.2 | Ki | 45 | Yes | |
SPMHGQZFMNZCBV
|
9.2 | Ki | 30 | Yes | |
UXQLMVSZSYZFID
|
9.2 | Ki | 12 | — | |
XKZINYYXWJEYEL
|
9.2 | Ki | 37 | — | |
VKBFHTIUXUCYRQ
|
9.2 | Ki | 66 | — | |
WEMHHXYZAJVSME
|
9.1 | IC50 | 3 | — | |
ZFFOQWCQWWHTIS
|
9.1 | IC50 | 3 | — | |
LGHBDVLAHHANMX
|
9.1 | Ki | 53 | — | |
MQRDVGBWWVWMEN
|
9.1 | Ki | 47 | — | |
NRGYZNJPCGRCLV
|
9.1 | Ki | 52 | — | |
UUVMNPKFPGJBNX
|
9.1 | Ki | 10 | — | |
XCHWBXBDZRJVDP
|
9.1 | Ki | 51 | — | |
MEBWIBLSBZGQSC
|
9.1 | IC50 | 3 | — | |
XPVAPOBXNPDLHJ
|
9.1 | IC50 | 3 | — | |
CQGCMAIBZGXOAJ
|
9.0 | IC50 | 3 | — | |
BIKYDWLMTPRSQL
|
9.0 | Ki | 50 | — | |
FGSVLADZCDNNOC
|
9.0 | Ki | 11 | — |