Target Details
| UniProt AC | P17752 |
|---|---|
| Gene Symbol | TPH1 |
| Protein Name | Tryptophan 5-hydroxylase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00351 (Biopterin_H) |
Summary
- Multi-target molecules 77
- Clinical molecules 0
- Avg pChEMBL 6.58
KEGG Pathways (4)
Top Co-occurrence Targets
- TPH2 77 shared
Active Molecules (77)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PNHHLSZYXLYIJJ
|
6.4 | IC50 | 2 | — | |
VAZSMDMETIFIBH
|
6.4 | IC50 | 2 | — | |
XFMJUABYLXDYGS
|
6.4 | IC50 | 2 | — | |
KRRLVHYAVVYHJV
|
6.4 | IC50 | 2 | — | |
RDEPTIRSFNDUOK
|
6.3 | IC50 | 2 | — | |
GVYDINLTFQEVNV
|
6.3 | IC50 | 2 | — | |
VLFJNBWPDSYJKV
|
6.3 | IC50 | 2 | — | |
QMMNAVKAIUPSEK
|
6.3 | IC50 | 2 | — | |
DYALZIDUQZQWAO
|
6.2 | IC50 | 2 | — | |
XBAIZUUPWRHPSF
|
6.2 | IC50 | 2 | — | |
LFTLBIABLIVZFE
|
6.2 | IC50 | 2 | — | |
CNVVLEOEWMATCW
|
6.1 | IC50 | 2 | — | |
GOHNCSPZIXYWEG
|
6.1 | IC50 | 2 | — | |
VBYFKIYMVQBKPN
|
6.1 | IC50 | 2 | — | |
IQIGWZLZUMNRAB
|
6.1 | IC50 | 2 | — | |
KTMJKDQZZJLZQQ
|
6.1 | IC50 | 2 | — | |
MDSQOJYHHZBZKA
|
6.1 | IC50 | 2 | — | |
NCLGDOBQAWBXRA
|
6.1 | IC50 | 2 | — | |
XNMUICFMGGQSMZ
|
6.1 | IC50 | 2 | — | |
NFUIGWIHITWNAY
|
6.1 | IC50 | 2 | — | |
JSUKDSWMYLASNP
|
6.1 | IC50 | 2 | — | |
CPISMKNBAXDQEB
|
6.1 | IC50 | 2 | — | |
GLUWCNQLKSIYKQ
|
6.1 | IC50 | 2 | — | |
OQKHEXPFNSCIHH
|
6.1 | IC50 | 2 | — | |
BYPGBGBRKVMXKG
|
6.0 | IC50 | 2 | — | |
MEZRLGNWKWWNDN
|
6.0 | IC50 | 2 | — | |
FFSQYZANLRAXHZ
|
6.0 | IC50 | 2 | — |