Target Details
| UniProt AC | P17706 |
|---|---|
| Gene Symbol | PTPN2 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 199
- Clinical molecules 0
- Avg pChEMBL 6.97
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (199)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KJYRSQLWJMEJNM
|
9.2 | IC50 | 2 | — | |
VILXHPHHLYDHSF
|
9.0 | IC50 | 2 | — | |
DVFCRTGTEXUFIN
|
8.7 | IC50 | 2 | — | |
CUHZHOXGTHDNHJ
|
8.7 | Ki | 2 | — | |
FGSXDTAUWKYQDX
|
8.7 | Ki | 2 | — | |
JYCQYNKZQPFRCV
|
8.7 | Ki | 2 | — | |
KCHARSDIPZLYSD
|
8.7 | Ki | 2 | — | |
XUXBACQLMYJEOX
|
8.7 | IC50 | 2 | — | |
DIRCLNUEXQQLRT
|
8.5 | IC50 | 2 | — | |
OVVNHIFLGPWASE
|
8.4 | IC50 | 2 | — | |
SLWJGFJPTJPJCI
|
8.4 | IC50 | 2 | — | |
XFJJNGDTJHVAME
|
8.4 | Ki | 2 | — | |
DZZMIHDOJVEPRL
|
8.4 | Ki | 2 | — | |
FEPAAIQAIYOLJA
|
8.3 | Ki | 2 | — | |
SUBZYMCEXNHIGE
|
8.3 | Ki | 2 | — | |
TUOKAOKHDHDMSS
|
8.3 | Ki | 2 | — | |
BBINWNMZKGHSMF
|
8.2 | Ki | 2 | — | |
KREWQXMKBWYIBM
|
8.2 | Ki | 2 | — | |
OADLYFBQFFZCCM
|
8.2 | IC50 | 2 | — | |
BTAGTGWPDROBMG
|
8.1 | IC50 | 2 | — | |
MQBLQNQFNLXLNE
|
8.1 | Ki | 2 | — | |
DGVSSAPOBXDLAY
|
8.1 | Ki | 2 | — | |
TYMUGKGQQMRQDI
|
8.1 | Ki | 2 | — | |
CVWLNWLJBZNMAZ
|
8.0 | IC50 | 2 | — | |
CWDWNOPXQHKDTA
|
8.0 | Ki | 2 | — | |
IQWGAAHPACZIDQ
|
8.0 | IC50 | 2 | — | |
VTRFCUCEJIBDSE
|
8.0 | IC50 | 2 | — | |
WNNXXNZHCLRWMD
|
8.0 | IC50 | 2 | — | |
ZQCMFHAFPWWDAP
|
8.0 | IC50 | 2 | — | |
YVEATRODDMUDLE
|
8.0 | IC50 | 2 | — | |
QEENZXFTRSDPEF
|
7.9 | Ki | 2 | — | |
HZALVWNZBKXRAP
|
7.9 | IC50 | 2 | — | |
ALTWGIIQPLQAAM
|
7.8 | IC50 | 2 | — | |
LSGOVYNHVSXFFJ
|
7.8 | IC50 | 4 | — | |
CLRSCKINFSDJJY
|
7.8 | IC50 | 2 | — | |
NFYJBAFWWYMJRQ
|
7.8 | IC50 | 2 | — | |
GBIIFVOJJXWYBK
|
7.8 | IC50 | 2 | — | |
LUQYNJZVPGUNOW
|
7.7 | IC50 | 2 | — | |
QKSXFCNKUJJHHX
|
7.7 | IC50 | 2 | — | |
GHQSTVDLTPVSRM
|
7.7 | IC50 | 2 | — | |
IKMFYRRINXPKDQ
|
7.7 | IC50 | 2 | — | |
SZXQFEXBARNEFM
|
7.7 | IC50 | 2 | — | |
UVMSRZSQDQTMKV
|
7.7 | Ki | 2 | — | |
KTEHTCIZIKZYJM
|
7.7 | IC50 | 2 | — | |
AYYVCIVIOZHWEO
|
7.6 | IC50 | 2 | — | |
UTZGYWMRZLQRNA
|
7.6 | IC50 | 2 | — | |
FBFPKPPWVZPZDO
|
7.6 | IC50 | 2 | — | |
KKLWOJSLYYMENS
|
7.6 | IC50 | 2 | — | |
RLNXXAOIKBYYIZ
|
7.6 | IC50 | 2 | — | |
FKOYIUYWMSVYKN
|
7.6 | Ki | 3 | — |