Target Details
| UniProt AC | P17655 |
|---|---|
| Gene Symbol | CAPN2 |
| Protein Name | Calpain-2 catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2) |
Summary
- Multi-target molecules 114
- Clinical molecules 6
- Avg pChEMBL 7.11
KEGG Pathways (8)
Active Molecules (114)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IAIIFNKYOCEUDZ
|
6.5 | Ki | 2 | — | |
NGBKFLTYGSREKK
|
6.5 | IC50 | 6 | Yes | |
DJCVSFWGKYHMKH
|
6.4 | Ki | 2 | — | |
CAILNONEKASNSH
|
6.4 | IC50 | 4 | — | |
MDMSJUTXKFAZPC
|
6.3 | Ki | 2 | — | |
JGMRVBHBMAPFGQ
|
6.3 | Ki | 3 | — | |
LPIGFPBIPKWMAQ
|
6.2 | Ki | 2 | — | |
WKNXHKNTWIOTFP
|
6.2 | Ki | 2 | — | |
ASXVEBPEZMSPHB
|
6.2 | IC50 | 3 | — | |
LWZDBQBMLCPSSM
|
6.2 | Ki | 2 | — | |
YGHHDWRITNGHCH
|
6.2 | IC50 | 3 | — | |
TZYWCYJVHRLUCT
|
6.2 | Ki | 23 | — | |
OCIZFJKKIPDOAQ
|
6.2 | Ki | 2 | — | |
JKZCALXNJCQERK
|
6.1 | Ki | 3 | — |