Target Details
UniProt ACP17655
Gene SymbolCAPN2
Protein NameCalpain-2 catalytic subunit
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2)
Summary
  • Multi-target molecules 114
  • Clinical molecules 6
  • Avg pChEMBL 7.11
Top Co-occurrence Targets
Active Molecules (114)
InChIKey pChEMBL Type Targets Clinical
VTIAIZFLWATOKO 7.1 Ki 3
QFMKANIDVYDNPI 7.1 Ki 3
VZPAOLJPGFQEEK 7.1 Ki 3
BXUSCFDRWLTJIE 7.0 Ki 2
VMVOHHPQIAPYHG 7.0 IC50 4
BWKQXOPKLULOSF 7.0 Ki 2
GPBVKHGLFLZPRW 7.0 Ki 2
PVWAECRYPMJXPR 7.0 Ki 2
JNRHNGGTJOBXHL 7.0 IC50 3 Yes
WJFAAUIYJQVQJJ 7.0 IC50 3 Yes
NRYJQWJSMMVVFJ 7.0 Ki 2
QXMOZKBLCRFIAZ 7.0 Ki 2
YFQOCPUAXDVMOS 7.0 Ki 2
BFOUDLDYLQQVEB 6.9 Ki 2
PBXPKBVKBJPJNW 6.9 Ki 2
PCBGEKNWVUOWNB 6.9 Ki 2
PLVWMBFPIAQRHK 6.9 Ki 5
YYVPOIBILWMYMW 6.9 Ki 2
FUUFQEWEOLXXBO 6.8 Ki 2
NGBKFLTYGSREKK 6.8 IC50 4
SFOHMHDPSOPFJL 6.8 Ki 3
DQCYYWKVEFPNIO 6.8 Ki 3
FYNLJGLHDFSIRG 6.8 Ki 2
ITIYFQNKFLZJTC 6.8 Ki 2
ONIATLXCZWBRKB 6.8 Ki 2
SFZKIYLOJIJGLV 6.8 Ki 2
ODDXFSGPQQWPEO 6.8 Ki 2
WIWTZPBWDNQRGX 6.8 Ki 2
FOBRVMHYTDWMJG 6.7 Ki 2
PGOQBJBMASKTEL 6.7 IC50 3 Yes
QVDJMLQSYRSZKC 6.7 IC50 6 Yes
GMTPAJDXCPJPRB 6.7 Ki 2
ALWTVFUIPPAQBH 6.7 Ki 2
MRMDMJWTKTVMPI 6.7 Ki 2
RFLQJGASGWLMCH 6.7 Ki 3
WYYJIPJWAOEKRW 6.7 Ki 2
YVMYGKAQQWIQNK 6.7 Ki 2
LKVFZCXXFXGYDC 6.7 Ki 3
CLBKCGOYQYVDNB 6.7 Ki 2
BOVPSXHLLSLLHY 6.6 Ki 2
XWPMWIRSEUHFET 6.6 Ki 3
JJAOOYMOIBDGJA 6.6 Ki 2
YVQGWXFRALVDJS 6.6 Ki 3
BMJOPMWNNPSOFV 6.5 Ki 2
DSEJDNPJKDDYTK 6.5 Ki 2
JFFBDCJEPWDUJE 6.5 Ki 2
VQYAUQQZKIBVFS 6.5 Ki 2
OWSUSRRECBEBIZ 6.5 Ki 2
SOPMJELGLOZMNK 6.5 Ki 2
BYDZMKUUIQPQOJ 6.5 Ki 2
2D structure