Target Details
UniProt ACP17655
Gene SymbolCAPN2
Protein NameCalpain-2 catalytic subunit
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01067 (Calpain_III) PF13833 (EF-hand_8) PF00648 (Peptidase_C2)
Summary
  • Multi-target molecules 114
  • Clinical molecules 6
  • Avg pChEMBL 7.11
Top Co-occurrence Targets
Active Molecules (114)
InChIKey pChEMBL Type Targets Clinical
LXQHAGZZTQHHEO 9.7 Ki 3
BPXIXWUDIQQWFO 9.7 Ki 2
XVYMHUPUYXWRAO 9.7 Ki 3
UEGOQZVAGRIZMF 9.6 Ki 2
LFXDKGYPGBYESW 8.3 Ki 3
RLWHWANZNLEGCV 8.3 Ki 3
UNCOFUQMWOIDMS 8.2 Ki 3
FBLCORIGBOTKPH 8.2 Ki 3
ZWWFTIUCCNWEGY 8.2 Ki 3
YQBJQKXVOBLSJT 8.1 Ki 3
MRAGOGINUXYQRY 8.0 Ki 3
XJPDKOSJXFJJJW 7.9 Ki 3
CZZWUFZBGQIPTE 7.8 Ki 2
PAURRTCLMITPQE 7.8 Ki 3
XOOLYFKEZMFYKD 7.8 Ki 2
XJZJHBWBHUESJD 7.7 Ki 3
YLELJBQQWFIURX 7.7 Ki 3
GLEMPIVMKMAASA 7.7 Ki 3
QDIFXVWJRNFSAW 7.7 Ki 3
ABCDOWZVJWRRMY 7.6 Ki 3
BQWHGKILBWBBEZ 7.6 Ki 3
VLHHFIURJMMQSU 7.5 Ki 3
NLQSCVDOWLITDK 7.5 Ki 2
WJDCRUSBRSNMME 7.4 Ki 3
TZVQRMYLYQNBOA 7.4 Ki 2
PNRWOFORTRJIMC 7.4 Ki 2
SFXFJMNNVMLAHN 7.4 Ki 4
YXADZLOTFPFSML 7.4 Ki 3
FRACLEVIDYQZNB 7.3 Ki 3
GOYRCQFAGVGQLH 7.3 Ki 3
MSLYBTUYFAYWQS 7.3 Ki 2
WNSZSZRXSNLYSL 7.3 Ki 2
OWMWWYSNZALAER 7.3 Ki 3
GWLZMBFVBYHGBD 7.3 Ki 2
BALDEWOSOSUCAN 7.2 Ki 3
LAMTYMVWEHUWRZ 7.2 Ki 2
PRVNMMSXHWFZAQ 7.2 Ki 3
SEANAGCTCGCPQM 7.2 Ki 3
CZPUWGZBBOMJKE 7.2 Ki 2
BJVLXPNAIXTDOW 7.2 Ki 3
LKJAJQNXOPUHBI 7.2 Ki 2
RVUJRRBCTAYDMG 7.2 Ki 3
LKEAIRWHRIHIEF 7.1 Ki 2
PJJKGPCXAZFMMA 7.1 Ki 2
GLNKVXFQBYGNDP 7.1 Ki 3
LBWUIVAFNQOLOB 7.1 Ki 2
MWKSRKSEWLRPBL 7.1 Kd 1075
WSJWUIDLGZAXID 7.1 IC50 4
YYDQGTWJPADAKS 7.1 IC50 3 Yes
VPUYRFKIVDMDKL 7.1 Ki 2
2D structure