Target Details
UniProt ACP17612
Gene SymbolPRKACA
Protein NamecAMP-dependent protein kinase catalytic subunit alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00069 (Pkinase)
Summary
  • Multi-target molecules 453
  • Clinical molecules 52
  • Avg pChEMBL 6.97
KEGG Pathways (72)
Top Co-occurrence Targets
Active Molecules (453)
InChIKey pChEMBL Type Targets Clinical
AOFGEEDOUASHKV 6.9 Ki 4
AUDNGNGLLRZLDR 6.9 Ki 33
GVMDVMPNOAVKJR 6.9 Ki 26 Yes
HOBMVEVXDIOMDM 6.9 Ki 18
KIOLXAWQJUDVMS 6.9 Ki 5
OEEGUWWPGAZRIJ 6.9 Ki 21
OUJZYQBEFNDJQN 6.9 Ki 71
RYYNGWLOYLRZLK 6.9 Ki 104
UMULGPSQNQMYNC 6.9 Ki 6
XFTPNRUQKBIHDT 6.9 Ki 8
OWJIKBAZUBPKGN 6.9 IC50 7
AFJRDFWMXUECEW 6.9 Kd 6
JJTVMBJRPZIZDA 6.9 IC50 4
LYJKMVFAIXOQLE 6.9 IC50 9
HFNKQEVNSGCOJV 6.8 Ki 18
MPZKHCPHRLXFAX 6.8 Ki 2
WKZTVBCDQYBGBO 6.8 IC50 16 Yes
DEEIBAOTOOOOIG 6.8 IC50 6
ACSYKUPGCXYRRO 6.8 Ki 26
BERZRFJWHSXBCR 6.8 Ki 7
CHADTINFLWZSKR 6.8 Ki 26
HBZTVQKHXVDIDE 6.8 Ki 9
HZJDBCYRQSJNLZ 6.8 Ki 7
JZTOUVBEZONDKA 6.8 Ki 80
KJGUOQMSLKZPAT 6.8 IC50 3
LCHCSKHPVCDXAU 6.8 Ki 30
MZDKLVOWGIOKTN 6.8 Ki 80
NEWAULHLLUCDPD 6.8 Ki 27
OQHALFBQFMAXFZ 6.8 Ki 9
PWIKZIKRKUUHRB 6.8 Ki 9
SKKRZILJUKYLJS 6.8 Ki 25
UFMAIBLTWQRHAK 6.8 Ki 10
VWVYILCFSYNJHF 6.8 Ki 49
AUHWQSZMVMMRLM 6.8 IC50 4
BPNNZZBLGSVSAA 6.8 IC50 7
WYHIMLBLXVJQLL 6.7 IC50 3
MCQBNMPALTYSES 6.7 IC50 3
JYRJOQGKGMHTOO 6.7 IC50 9
NGOGFTYYXHNFQH 6.7 Ki 15
UBZNLGBMKJHEFB 6.7 IC50 3
AWDORCFLUJZUQS 6.7 Ki 22
CRKQBJZCCHKEGI 6.7 Ki 20
HSMUWLLZAZCLHF 6.7 Ki 25
HXDDWVMJYDULAZ 6.7 Ki 13
KEBXAEFZLCNLJJ 6.7 Ki 13
LUPCHAFIKZSOOK 6.7 Ki 15
MTYMWGNJKDHWGN 6.7 Ki 18
NGDNKYRUKIPCLK 6.7 Ki 12
ODPGGGTTYSGTGO 6.7 Ki 153
OFPXYNMQWVCVKZ 6.7 Ki 8
2D structure