Target Details
| UniProt AC | P17612 |
|---|---|
| Gene Symbol | PRKACA |
| Protein Name | cAMP-dependent protein kinase catalytic subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 453
- Clinical molecules 52
- Avg pChEMBL 6.97
KEGG Pathways (72)
- Adrenergic signaling in cardiomyocytes
- Alcoholism
- Aldosterone synthesis and secretion
- Amoebiasis
- Amphetamine addiction
- Apelin signaling pathway
- Autophagy - animal
- Bile secretion
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cocaine addiction
- Cortisol synthesis and secretion
- Cushing syndrome
- Dilated cardiomyopathy
- Dopaminergic synapse
- Endocrine and other factor-regulated calcium reabsorption
- Endocrine resistance
- Estrogen signaling pathway
- GABAergic synapse
- Gap junction
- Gastric acid secretion
- Glucagon signaling pathway
- Glutamatergic synapse
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hormone signaling
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Insulin signaling pathway
- Long-term potentiation
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanogenesis
- Morphine addiction
- Neuroactive ligand signaling
- Olfactory transduction
- Oocyte meiosis
- Ovarian steroidogenesis
- Oxytocin signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Parkinson disease
- Pathways in cancer
- Platelet activation
- Prion disease
- Progesterone-mediated oocyte maturation
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of lipolysis in adipocytes
- Relaxin signaling pathway
- Renin secretion
- Retrograde endocannabinoid signaling
- Salivary secretion
- Serotonergic synapse
- Taste transduction
- Thermogenesis
- Thyroid hormone signaling pathway
- Thyroid hormone synthesis
- Tight junction
- Vascular smooth muscle contraction
- Vasopressin-regulated water reabsorption
- Vibrio cholerae infection
- Viral carcinogenesis
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (453)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IRGJDPZJEUYSKS
|
7.5 | IC50 | 7 | — | |
IRGJDPZJEUYSKS
|
7.5 | IC50 | 9 | — | |
IRGJDPZJEUYSKS
|
7.5 | IC50 | 9 | — | |
JTJAWKUSBMOQSN
|
7.5 | Ki | 5 | — | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
ORTCEQUUKXOFAE
|
7.5 | IC50 | 2 | — | |
BJQFSJIVYSQLSX
|
7.5 | IC50 | 4 | — | |
FUMCKNCUEAQHCV
|
7.5 | Ki | 103 | — | |
IOYGZJJCJBOPDM
|
7.5 | Ki | 8 | — | |
NIUJTENHSPPCKO
|
7.5 | Ki | 9 | — | |
QVZTZUQJFINWOX
|
7.5 | IC50 | 4 | — | |
SGHXFHRRWFLILP
|
7.5 | Ki | 29 | — | |
WAKGEHXTOOFEAE
|
7.5 | Ki | 27 | — | |
XZVLUQDUOAWQMB
|
7.5 | Ki | 4 | — | |
YOVNFNXUCOWYSG
|
7.5 | Ki | 33 | Yes | |
ZGGIYFOLDBTZIL
|
7.5 | Ki | 27 | — | |
HPWBHQIUIBFTQC
|
7.5 | IC50 | 4 | — | |
JBOUGNBDORLVHX
|
7.5 | IC50 | 2 | — | |
KKSLZAWDUQRHLJ
|
7.5 | Ki | 2 | — | |
RVSXZFNWIKKCIQ
|
7.5 | IC50 | 2 | — | |
SGHXFHRRWFLILP
|
7.4 | IC50 | 8 | — | |
JBLPUDJLELBRHC
|
7.4 | Ki | 9 | — | |
LOMGAGWJYPGDLT
|
7.4 | Ki | 8 | — | |
LRZYYIZFBXFSJB
|
7.4 | Ki | 69 | — | |
RFBPWKMQWSIPEO
|
7.4 | Ki | 28 | — | |
RGOPHVZLEMGMBZ
|
7.4 | Ki | 20 | — | |
XXSPHNFKLDJDAK
|
7.4 | Ki | 26 | — | |
YGEACCLUBSGMMJ
|
7.4 | Ki | 16 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
YOXPJLZIOXCBGO
|
7.3 | IC50 | 4 | — | |
ZAMACYCHJDCXFC
|
7.3 | IC50 | 4 | — | |
PQHAJHBMGVFBAP
|
7.3 | IC50 | 4 | — | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — | |
AQDWLHMFJHACCX
|
7.3 | Ki | 8 | — | |
CNQGNADBGYCKKV
|
7.3 | Ki | 25 | — | |
FCVHMDURXUOCFY
|
7.3 | IC50 | 7 | — | |
JMHQUQCLIVNTHT
|
7.3 | Ki | 24 | — | |
JPOSFPUHBHRUAX
|
7.3 | Ki | 40 | Yes | |
KCKXYZOBGBJZEG
|
7.3 | Ki | 36 | — | |
SJDGHXXYFFXVPE
|
7.3 | Ki | 9 | — | |
TVEREFRWBLRPPJ
|
7.3 | Ki | 15 | — | |
XMFUGSRATNLPRM
|
7.3 | Ki | 19 | — | |
XSDJOIOVIMPMHD
|
7.3 | Ki | 44 | — | |
BRIBVJICQJDZMF
|
7.3 | Kd | 2 | — | |
LIYNJKNSBUCWCZ
|
7.3 | IC50 | 3 | — | |
WXJWGWJEPVCGSC
|
7.3 | IC50 | 3 | — | |
HLXIFVDYTGEUJV
|
7.3 | IC50 | 15 | Yes | |
BPNUQXPIQBZCMR
|
7.2 | Kd | 83 | Yes | |
HOFYBOPHRAHNMK
|
7.2 | IC50 | 4 | — | |
JMGYGTNBCVNXBS
|
7.2 | IC50 | 2 | — |